PT66780A - PROCESS FOR THE PREPARATION OF 5-AROIL-1,2-DIHYDRO-3H-PIRROLE (1,2-ALPHA) PIRROLE-1-CARBOXILIC ACID DERIVATIVES - Google Patents

PROCESS FOR THE PREPARATION OF 5-AROIL-1,2-DIHYDRO-3H-PIRROLE (1,2-ALPHA) PIRROLE-1-CARBOXILIC ACID DERIVATIVES

Info

Publication number
PT66780A
PT66780A PT66780A PT6678077A PT66780A PT 66780 A PT66780 A PT 66780A PT 66780 A PT66780 A PT 66780A PT 6678077 A PT6678077 A PT 6678077A PT 66780 A PT66780 A PT 66780A
Authority
PT
Portugal
Prior art keywords
pirrole
aroil
dihydro
alpha
preparation
Prior art date
Application number
PT66780A
Other languages
French (fr)
Portuguese (pt)
Other versions
PT66780B (en
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27107410&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT66780(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US05/771,286 external-priority patent/US4089969A/en
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of PT66780A publication Critical patent/PT66780A/en
Publication of PT66780B publication Critical patent/PT66780B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
PT66780A 1976-07-14 1977-07-08 PROCESS FOR THE PREPARATION OF 5-AROIL-1,2-DIHYDRO-3H-PIRROLE / 1,2-ALPHA / PIRROLE-1-CARBOXILIC ACID DERIVATIVES PT66780B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US70490976A 1976-07-14 1976-07-14
US05/771,286 US4089969A (en) 1976-07-14 1977-02-23 5-Aroyl-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof

Publications (2)

Publication Number Publication Date
PT66780A true PT66780A (en) 1977-08-01
PT66780B PT66780B (en) 1978-12-18

Family

ID=27107410

Family Applications (1)

Application Number Title Priority Date Filing Date
PT66780A PT66780B (en) 1976-07-14 1977-07-08 PROCESS FOR THE PREPARATION OF 5-AROIL-1,2-DIHYDRO-3H-PIRROLE / 1,2-ALPHA / PIRROLE-1-CARBOXILIC ACID DERIVATIVES

Country Status (27)

Country Link
JP (1) JPS539788A (en)
AR (1) AR224997A1 (en)
CA (1) CA1102809A (en)
CH (3) CH641458A5 (en)
CS (1) CS204954B2 (en)
DE (2) DE2731678A1 (en)
DK (1) DK151886C (en)
ES (2) ES460706A1 (en)
FI (1) FI63406C (en)
FR (2) FR2358406A1 (en)
GB (1) GB1554075A (en)
GR (1) GR61111B (en)
HK (1) HK15981A (en)
HU (1) HU174224B (en)
IE (1) IE45253B1 (en)
IL (2) IL52493A (en)
IT (1) IT1117313B (en)
MX (1) MX163202B (en)
MY (1) MY8100357A (en)
NL (2) NL186318C (en)
NO (1) NO147564C (en)
NZ (1) NZ184610A (en)
PL (4) PL109390B1 (en)
PT (1) PT66780B (en)
SE (1) SE434643B (en)
SU (1) SU695558A3 (en)
YU (1) YU40816B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4140698A (en) * 1977-07-25 1979-02-20 Syntex (Usa) Inc. 1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles
JPS55124633A (en) * 1979-03-19 1980-09-25 Sohachi Takeuchi Manufacturing method of tubular vessel
US4344943A (en) * 1980-06-09 1982-08-17 Syntex (U.S.A.) Inc. 6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo[1,2-a]-pyrrole-1-carboxylic acids and derivatives thereof
US4353829A (en) * 1980-11-21 1982-10-12 Syntex (U.S.A.) Inc. Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters
US4511724A (en) * 1982-06-10 1985-04-16 Merck & Co., Inc. 5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents
JPS5910589A (en) * 1982-06-10 1984-01-20 メルク　エンド　カムパニー　インコーポレーテツド Antiinflammatory and analgesic novel 5-(pyrrol-2-oyl)-1,2-dihydro-3h-pyrrolo(1,2-a) pyrrole derivative
US4874871A (en) * 1987-03-25 1989-10-17 Syntex (U.S.A.) Inc. Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds
JPH0739418B2 (en) * 1987-09-10 1995-05-01 久光製薬株式会社 Novel 3-aroyl-6,7-dihydro-5H-pyrrolo [1,2-c] imidazole-7-carboxylic acid derivative
JP2649168B2 (en) * 1988-02-25 1997-09-03 久光製薬株式会社 Novel 5,6-diphenyl-1,2-dihydro-3H-pyrrolo [1,2-a] pyrrole-1-carboxylic acid derivatives
IT1250691B (en) * 1991-07-22 1995-04-21 Giancarlo Santus THERAPEUTIC COMPOSITIONS FOR INTRANASAL ADMINISTRATION INCLUDING KETOROLAC.
WO1993009768A1 (en) * 1991-11-11 1993-05-27 Hisamitsu Pharmaceutical Co., Inc. Fomentation containing ketorolac
DE4300697C1 (en) * 1993-01-13 1994-05-19 Roemmers Sa New 2-pyrrolidino-ethyl ester of ketorolac - useful as analgesic, antiinflammatory and antipyretic agent with low ulcerogenicity
US5622948A (en) * 1994-12-01 1997-04-22 Syntex (U.S.A.) Inc. Pyrrole pyridazine and pyridazinone anti-inflammatory agents
JP2008210666A (en) * 2007-02-27 2008-09-11 Okamura Corp Lighting system in merchandise display shelf

Also Published As

Publication number Publication date
SE7708141L (en) 1978-01-15
NL930021I1 (en) 1993-05-03
PL109390B1 (en) 1980-05-31
MX163202B (en) 1992-02-20
IL52493A0 (en) 1977-10-31
ES470214A1 (en) 1979-09-16
PL124445B1 (en) 1983-01-31
JPS6254109B2 (en) 1987-11-13
NL7707651A (en) 1978-01-17
NO772494L (en) 1978-01-17
AU2697577A (en) 1979-01-18
NO147564B (en) 1983-01-24
CA1102809A (en) 1981-06-09
SU695558A3 (en) 1979-10-30
FI63406B (en) 1983-02-28
FR2375234A1 (en) 1978-07-21
IT1117313B (en) 1986-02-17
AU513384B2 (en) 1980-11-27
CH646973A5 (en) 1984-12-28
NO147564C (en) 1983-05-18
DK307577A (en) 1978-01-15
DE2760330C2 (en) 1989-06-15
HU174224B (en) 1979-11-28
IE45253L (en) 1978-01-14
HK15981A (en) 1981-05-01
FI63406C (en) 1983-06-10
NL186318C (en) 1990-11-01
CS204954B2 (en) 1981-04-30
MY8100357A (en) 1981-12-31
YU172177A (en) 1983-09-30
FR2358406B1 (en) 1981-04-17
IL52493A (en) 1982-02-28
DK151886C (en) 1988-06-06
FR2358406A1 (en) 1978-02-10
IE45253B1 (en) 1982-07-14
NZ184610A (en) 1979-03-28
DE2731678C2 (en) 1989-06-08
PL199603A1 (en) 1978-04-24
PL124711B1 (en) 1983-02-28
CH641458A5 (en) 1984-02-29
SE434643B (en) 1984-08-06
NL930021I2 (en) 1997-03-03
AR224997A1 (en) 1982-02-15
GR61111B (en) 1978-09-12
DK151886B (en) 1988-01-11
NL186318B (en) 1990-06-01
JPS539788A (en) 1978-01-28
FI772153A (en) 1978-01-15
PT66780B (en) 1978-12-18
ES460706A1 (en) 1978-12-01
DE2731678A1 (en) 1978-03-16
CH646972A5 (en) 1984-12-28
PL124444B1 (en) 1983-01-31
GB1554075A (en) 1979-10-17
FR2375234B1 (en) 1980-11-07
IL58779A0 (en) 1980-02-29
YU40816B (en) 1986-06-30

Similar Documents

Publication Publication Date Title
RO80265A (en) PROCESS FOR THE PREPARATION OF BETA-CARBOLINE-3-CARBOXYLICIDE ACID DERIVATIVES
RO75256A (en) PROCESS FOR THE PREPARATION OF 1,2,3, THIAZOLE-5-CARBOXYLIC ACID DERIVATIVES
RO75478A (en) PROCEDURE FOR THE PREPARATION OF ALPROCED ACID DERIVATIVES FOR THE PREPARATION OF ALPHA-PHENOYPROPIONIC ACID DERIVATIVES PHA-PHENOXYPROPIONIC
RO70687A (en) PROCESS FOR THE PREPARATION OF PHENOXYPHENOXYPROPIONIC ACID DERIVATIVES
RO70264A (en) PROCESS FOR THE PREPARATION OF 1-ALKYL-5-AROYLPYROL-2-ACETIC ACID DERIVATIVES
RO78013A (en) PROCESS FOR THE PREPARATION OF THIAZONCARBOXYLIC OR MORPHOLINCARBOXYLIC THIAZOLIDINCARBOXYLIC ACID DEDIVES
PT66780A (en) PROCESS FOR THE PREPARATION OF 5-AROIL-1,2-DIHYDRO-3H-PIRROLE (1,2-ALPHA) PIRROLE-1-CARBOXILIC ACID DERIVATIVES
BE890223A (en) PROCESS FOR THE PREPARATION OF QUINOLEINE-CARBOXYLIC ACID DERIVATIVES
PT67004B (en) PROCESS FOR THE PREPARATION OF 7-ACILAMINE-8-OXO-3-OXA-1-AZABICICLE- / 4,2,0 / -OCTANE-2-CARBOXIC ACID DERIVATIVES
PT67088A (en) PROCESS FOR THE PREPARATION OF (PHENYL-3-AMINO-2-PROPIONYLOXY) -2-ACETIC ACID DERIVATIVES
RO79837A (en) PROCESS FOR THE PREPARATION OF CYANHYDRIC ACID
RO77179A (en) PROCESS FOR THE PREPARATION OF 3,4-DIHYDRO-2-METHYL-4-OXO-2H-1,2-BENZOTHIAZIN-O-CARBOXYLIC ACID CHLORAMIDES
RO69916A (en) PROCESS FOR THE PREPARATION OF 3,7-DIMETHYLOCY-2-EN-OIC ACID NITRYL
BE880031A (en) PROCESS FOR THE PREPARATION OF 1 ALPHA, 3 BETA-DIHYDROXY-DELTA 5-STEROIDES
BE861693A (en) PROCESS FOR REDUCTION OF 2,5-DICETOGLUCONIC ACID
RO81937A (en) PROCESS FOR THE PREPARATION OF 7 BETA-AMINOTHIAZOLYLACETAMIDO-3-CEPHEM-4-CARBOXYLIC ACID DERIVATIVES
BE865774A (en) PROCESS FOR THE PREPARATION OF 1-AMINO-8-NAPHTOL-3,6-DISULPHONIC ACID ("H" ACID)
PT74813A (en) PROCESS FOR THE PREPARATION OF 1,4-THIAZAN CARBOXYLIC ACID DERIVATIVES
FR2353558A1 (en) PROCESS FOR THE PREPARATION OF 7-AMINO-D3-DESACETOXYCEPHALOSPORANIC ACID DERIVATIVES
BE873495A (en) PROCESS FOR THE PREPARATION OF 2,4-DIFLUORO-6-AMINO-S-TRIAZINE
BE820267A (en) PROCESS FOR THE PREPARATION OF P. ISOBUTYL-HYDRATROPIC ACID
BE877887A (en) PROCESS FOR THE PREPARATION OF DERIVATIVES OF BENZOXAZOLYL-PROPIONIC ACID
FR2351983A1 (en) PROCESS FOR THE PREPARATION OF CEPHALOSPORANIC ACID DERIVATIVES
BE858002A (en) PROCESS FOR PREPARING DERIVATIVES OF EPOXY-1,2-PROPYLPHOSPHONIC ACID
RO73287A (en) PROCESS FOR THE PREPARATION OF ESTERS OF N, N-DIMETHYL-O-PYRAZOLYLCARBAMINIC ACID