SE434643B - ANALOGY PROCEDURE FOR PREPARING 5-AROYL-1,2-DIHYDRO-3H-PYRROLO (1,2-A) -PYRROL-1-CARBONIC ACID DERIVATIVES - Google Patents

ANALOGY PROCEDURE FOR PREPARING 5-AROYL-1,2-DIHYDRO-3H-PYRROLO (1,2-A) -PYRROL-1-CARBONIC ACID DERIVATIVES

Info

Publication number
SE434643B
SE434643B SE7708141A SE7708141A SE434643B SE 434643 B SE434643 B SE 434643B SE 7708141 A SE7708141 A SE 7708141A SE 7708141 A SE7708141 A SE 7708141A SE 434643 B SE434643 B SE 434643B
Authority
SE
Sweden
Prior art keywords
aroyl
pyrrol
pyrrolo
dihydro
preparing
Prior art date
Application number
SE7708141A
Other languages
Swedish (sv)
Other versions
SE7708141L (en
Inventor
J M Muchowski
A F Kluge
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27107410&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SE434643(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US05/771,286 external-priority patent/US4089969A/en
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of SE7708141L publication Critical patent/SE7708141L/en
Publication of SE434643B publication Critical patent/SE434643B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
SE7708141A 1976-07-14 1977-07-13 ANALOGY PROCEDURE FOR PREPARING 5-AROYL-1,2-DIHYDRO-3H-PYRROLO (1,2-A) -PYRROL-1-CARBONIC ACID DERIVATIVES SE434643B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US70490976A 1976-07-14 1976-07-14
US05/771,286 US4089969A (en) 1976-07-14 1977-02-23 5-Aroyl-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof

Publications (2)

Publication Number Publication Date
SE7708141L SE7708141L (en) 1978-01-15
SE434643B true SE434643B (en) 1984-08-06

Family

ID=27107410

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7708141A SE434643B (en) 1976-07-14 1977-07-13 ANALOGY PROCEDURE FOR PREPARING 5-AROYL-1,2-DIHYDRO-3H-PYRROLO (1,2-A) -PYRROL-1-CARBONIC ACID DERIVATIVES

Country Status (27)

Country Link
JP (1) JPS539788A (en)
AR (1) AR224997A1 (en)
CA (1) CA1102809A (en)
CH (3) CH641458A5 (en)
CS (1) CS204954B2 (en)
DE (2) DE2760330C2 (en)
DK (1) DK151886C (en)
ES (2) ES460706A1 (en)
FI (1) FI63406C (en)
FR (2) FR2358406A1 (en)
GB (1) GB1554075A (en)
GR (1) GR61111B (en)
HK (1) HK15981A (en)
HU (1) HU174224B (en)
IE (1) IE45253B1 (en)
IL (2) IL52493A (en)
IT (1) IT1117313B (en)
MX (1) MX163202B (en)
MY (1) MY8100357A (en)
NL (2) NL186318C (en)
NO (1) NO147564C (en)
NZ (1) NZ184610A (en)
PL (4) PL124445B1 (en)
PT (1) PT66780B (en)
SE (1) SE434643B (en)
SU (1) SU695558A3 (en)
YU (1) YU40816B (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4140698A (en) * 1977-07-25 1979-02-20 Syntex (Usa) Inc. 1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles
JPS55124633A (en) * 1979-03-19 1980-09-25 Sohachi Takeuchi Manufacturing method of tubular vessel
US4344943A (en) * 1980-06-09 1982-08-17 Syntex (U.S.A.) Inc. 6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo[1,2-a]-pyrrole-1-carboxylic acids and derivatives thereof
US4353829A (en) * 1980-11-21 1982-10-12 Syntex (U.S.A.) Inc. Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters
JPS5910589A (en) * 1982-06-10 1984-01-20 メルク　エンド　カムパニー　インコーポレーテツド Antiinflammatory and analgesic novel 5-(pyrrol-2-oyl)-1,2-dihydro-3h-pyrrolo(1,2-a) pyrrole derivative
US4511724A (en) * 1982-06-10 1985-04-16 Merck & Co., Inc. 5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents
US4874871A (en) * 1987-03-25 1989-10-17 Syntex (U.S.A.) Inc. Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds
JPH0739418B2 (en) * 1987-09-10 1995-05-01 久光製薬株式会社 Novel 3-aroyl-6,7-dihydro-5H-pyrrolo [1,2-c] imidazole-7-carboxylic acid derivative
JP2649168B2 (en) * 1988-02-25 1997-09-03 久光製薬株式会社 Novel 5,6-diphenyl-1,2-dihydro-3H-pyrrolo [1,2-a] pyrrole-1-carboxylic acid derivatives
IT1250691B (en) * 1991-07-22 1995-04-21 Giancarlo Santus THERAPEUTIC COMPOSITIONS FOR INTRANASAL ADMINISTRATION INCLUDING KETOROLAC.
AU669492B2 (en) * 1991-11-11 1996-06-13 Hisamitsu Pharmaceutical Co., Inc. Fomentation containing ketorolac
DE4300697C1 (en) * 1993-01-13 1994-05-19 Roemmers Sa New 2-pyrrolidino-ethyl ester of ketorolac - useful as analgesic, antiinflammatory and antipyretic agent with low ulcerogenicity
US5622948A (en) * 1994-12-01 1997-04-22 Syntex (U.S.A.) Inc. Pyrrole pyridazine and pyridazinone anti-inflammatory agents
JP2008210666A (en) * 2007-02-27 2008-09-11 Okamura Corp Lighting device for merchandise display shelf
KR20230131182A (en) * 2020-12-16 2023-09-12 뉴 프런티어 랩스 엘엘씨 Dicarboxylic acid esters to induce analgesic effects

Also Published As

Publication number Publication date
HU174224B (en) 1979-11-28
IL52493A0 (en) 1977-10-31
DE2760330C2 (en) 1989-06-15
MX163202B (en) 1992-02-20
FI772153A7 (en) 1978-01-15
GB1554075A (en) 1979-10-17
AU2697577A (en) 1979-01-18
SE7708141L (en) 1978-01-15
FI63406B (en) 1983-02-28
IT1117313B (en) 1986-02-17
FI63406C (en) 1983-06-10
NL7707651A (en) 1978-01-17
NZ184610A (en) 1979-03-28
YU40816B (en) 1986-06-30
DK307577A (en) 1978-01-15
NL930021I2 (en) 1997-03-03
PL109390B1 (en) 1980-05-31
NL186318C (en) 1990-11-01
PT66780B (en) 1978-12-18
NO772494L (en) 1978-01-17
AR224997A1 (en) 1982-02-15
CH646972A5 (en) 1984-12-28
PL124444B1 (en) 1983-01-31
CH641458A5 (en) 1984-02-29
PL124711B1 (en) 1983-02-28
NO147564B (en) 1983-01-24
FR2375234A1 (en) 1978-07-21
NO147564C (en) 1983-05-18
SU695558A3 (en) 1979-10-30
DE2731678C2 (en) 1989-06-08
FR2375234B1 (en) 1980-11-07
GR61111B (en) 1978-09-12
HK15981A (en) 1981-05-01
JPS539788A (en) 1978-01-28
PL124445B1 (en) 1983-01-31
JPS6254109B2 (en) 1987-11-13
PL199603A1 (en) 1978-04-24
DK151886C (en) 1988-06-06
NL930021I1 (en) 1993-05-03
AU513384B2 (en) 1980-11-27
CA1102809A (en) 1981-06-09
NL186318B (en) 1990-06-01
FR2358406A1 (en) 1978-02-10
ES470214A1 (en) 1979-09-16
ES460706A1 (en) 1978-12-01
IE45253L (en) 1978-01-14
DE2731678A1 (en) 1978-03-16
FR2358406B1 (en) 1981-04-17
DK151886B (en) 1988-01-11
MY8100357A (en) 1981-12-31
IL52493A (en) 1982-02-28
CS204954B2 (en) 1981-04-30
IE45253B1 (en) 1982-07-14
CH646973A5 (en) 1984-12-28
YU172177A (en) 1983-09-30
IL58779A0 (en) 1980-02-29
PT66780A (en) 1977-08-01

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