ES2804202T3 - Producto intermedio sintético de Formula cristalina de (R)-1(2,2-difluorobenzo[d][1,3]dioxol-5il)-N-(1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2il)-1h-indol-5il)ciclopropanocarboxamida - Google Patents

Producto intermedio sintético de Formula cristalina de (R)-1(2,2-difluorobenzo[d][1,3]dioxol-5il)-N-(1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2il)-1h-indol-5il)ciclopropanocarboxamida Download PDF

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Publication number
ES2804202T3
ES2804202T3 ES17154840T ES17154840T ES2804202T3 ES 2804202 T3 ES2804202 T3 ES 2804202T3 ES 17154840 T ES17154840 T ES 17154840T ES 17154840 T ES17154840 T ES 17154840T ES 2804202 T3 ES2804202 T3 ES 2804202T3
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compound
vol
cftr
less
amorphous
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English (en)
Spanish (es)
Inventor
Ali Keshavarz-Shokri
Beili Zhang
Tim Edward Alcacio
Elaine Chungmin Lee
Yuegang Zhang
Mariusz Krawiec
William A Nugent
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Vertex Pharmaceuticals Inc
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Vertex Pharmaceuticals Inc
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Application filed by Vertex Pharmaceuticals Inc filed Critical Vertex Pharmaceuticals Inc
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    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
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ES17154840T 2010-03-25 2011-03-25 Producto intermedio sintético de Formula cristalina de (R)-1(2,2-difluorobenzo[d][1,3]dioxol-5il)-N-(1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2il)-1h-indol-5il)ciclopropanocarboxamida Active ES2804202T3 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US31737610P 2010-03-25 2010-03-25
US31995310P 2010-04-01 2010-04-01
US32163610P 2010-04-07 2010-04-07
US32156110P 2010-04-07 2010-04-07

Publications (1)

Publication Number Publication Date
ES2804202T3 true ES2804202T3 (es) 2021-02-04

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ID=43903962

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Application Number Title Priority Date Filing Date
ES17154840T Active ES2804202T3 (es) 2010-03-25 2011-03-25 Producto intermedio sintético de Formula cristalina de (R)-1(2,2-difluorobenzo[d][1,3]dioxol-5il)-N-(1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2il)-1h-indol-5il)ciclopropanocarboxamida
ES14172991T Active ES2845449T3 (es) 2010-03-25 2011-03-25 Dispersión sólida de forma amorfa de (R)-1(2,2-difluorobenzo[d][1,3]dioxol-5-il)-N-(1-(2,3-dihidroxipropil)-6-fluoro-2(1-hidroxi-2-metilpropan-2-il)-1h-indol-5il)-ciclopropanocarboxamida
ES20206423T Active ES2951520T3 (es) 2010-03-25 2011-03-25 Síntesis e intermedios de (R)-1-(2,2-difluorobenzo[d][1,3]dioxol-5-il)-N-(1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2-il)-1H-indol-5il)-ciclopropanocarboxamida
ES11713134.2T Active ES2604105T3 (es) 2010-03-25 2011-03-25 Formula cristalina de (r) -1 (2,2- difluorobenzo [d] [1,3] dioxol - 5yl) - n- (1- (2,3 - dihidroxipropil) - 6 - fluoro - 2- (1 - hydroxy-2-metilpropan-2il) -1h-indol-5il) cyclopropanecarboxamida

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ES14172991T Active ES2845449T3 (es) 2010-03-25 2011-03-25 Dispersión sólida de forma amorfa de (R)-1(2,2-difluorobenzo[d][1,3]dioxol-5-il)-N-(1-(2,3-dihidroxipropil)-6-fluoro-2(1-hidroxi-2-metilpropan-2-il)-1h-indol-5il)-ciclopropanocarboxamida
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