ES2634490T3 - Derivados de ácido napht-2-ylacetico para tratar el sida - Google Patents
Derivados de ácido napht-2-ylacetico para tratar el sida Download PDFInfo
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- ES2634490T3 ES2634490T3 ES11738878.5T ES11738878T ES2634490T3 ES 2634490 T3 ES2634490 T3 ES 2634490T3 ES 11738878 T ES11738878 T ES 11738878T ES 2634490 T3 ES2634490 T3 ES 2634490T3
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- napht
- acid derivatives
- ylacetic acid
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- C07C59/40—Unsaturated compounds
- C07C59/58—Unsaturated compounds containing ether groups, groups, groups, or groups
- C07C59/64—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
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- C07C57/58—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing halogen containing six-membered aromatic rings
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
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- C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
- C07C233/46—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
- C07C233/47—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
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- C07C255/57—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and carboxyl groups, other than cyano groups, bound to the carbon skeleton
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- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
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- C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
- C07C311/16—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom
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- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
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- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
Abstract
Un compuesto seleccionado del grupo que consiste en: **Fórmula** o una sal farmacéuticamente aceptable del mismo.
Description
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Claims (1)
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Applications Claiming Priority (3)
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US36131410P | 2010-07-02 | 2010-07-02 | |
US361314P | 2010-07-02 | ||
PCT/US2011/042880 WO2012003497A1 (en) | 2010-07-02 | 2011-07-01 | Napht- 2 -ylacetic acid derivatives to treat aids |
Publications (1)
Publication Number | Publication Date |
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ES2634490T3 true ES2634490T3 (es) | 2017-09-28 |
Family
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ES11738878.5T Active ES2634490T3 (es) | 2010-07-02 | 2011-07-01 | Derivados de ácido napht-2-ylacetico para tratar el sida |
Country Status (27)
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US (1) | US9102614B2 (es) |
EP (1) | EP2588450B1 (es) |
JP (2) | JP5984218B2 (es) |
KR (1) | KR20130135826A (es) |
CN (1) | CN103140474A (es) |
AP (1) | AP2013006706A0 (es) |
AR (1) | AR082079A1 (es) |
AU (1) | AU2011274322B2 (es) |
BR (1) | BR112013000043A2 (es) |
CA (1) | CA2802308C (es) |
CL (1) | CL2012003722A1 (es) |
CO (1) | CO6660497A2 (es) |
CR (1) | CR20130045A (es) |
EA (1) | EA201291300A1 (es) |
EC (1) | ECSP13012417A (es) |
ES (1) | ES2634490T3 (es) |
IL (1) | IL223558A0 (es) |
MA (1) | MA34397B1 (es) |
MX (1) | MX2012015097A (es) |
NZ (1) | NZ604598A (es) |
PE (1) | PE20130385A1 (es) |
PT (1) | PT2588450T (es) |
SG (1) | SG186820A1 (es) |
TW (1) | TWI453208B (es) |
UY (1) | UY33480A (es) |
WO (1) | WO2012003497A1 (es) |
ZA (1) | ZA201209596B (es) |
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PT2588450T (pt) | 2017-08-03 |
PE20130385A1 (es) | 2013-03-30 |
ZA201209596B (en) | 2015-06-24 |
CO6660497A2 (es) | 2013-04-30 |
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EA201291300A1 (ru) | 2013-06-28 |
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JP5984218B2 (ja) | 2016-09-06 |
AU2011274322B2 (en) | 2015-08-13 |
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IL223558A0 (en) | 2013-03-05 |
JP2013535426A (ja) | 2013-09-12 |
BR112013000043A2 (pt) | 2019-09-24 |
CA2802308C (en) | 2018-08-28 |
CL2012003722A1 (es) | 2014-03-21 |
SG186820A1 (en) | 2013-02-28 |
MX2012015097A (es) | 2013-05-28 |
AP2013006706A0 (en) | 2013-02-28 |
UY33480A (es) | 2012-02-29 |
WO2012003497A1 (en) | 2012-01-05 |
EP2588450A1 (en) | 2013-05-08 |
CN103140474A (zh) | 2013-06-05 |
CR20130045A (es) | 2013-05-16 |
US9102614B2 (en) | 2015-08-11 |
AU2011274322A1 (en) | 2013-01-10 |
NZ604598A (en) | 2014-12-24 |
AR082079A1 (es) | 2012-11-07 |
EP2588450B1 (en) | 2017-05-24 |
CA2802308A1 (en) | 2012-01-05 |
TWI453208B (zh) | 2014-09-21 |
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