FR2839646B1 - Utilisation de derives de quinoleine a effet anti-integrase et ses applications - Google Patents
Utilisation de derives de quinoleine a effet anti-integrase et ses applicationsInfo
- Publication number
- FR2839646B1 FR2839646B1 FR0206126A FR0206126A FR2839646B1 FR 2839646 B1 FR2839646 B1 FR 2839646B1 FR 0206126 A FR0206126 A FR 0206126A FR 0206126 A FR0206126 A FR 0206126A FR 2839646 B1 FR2839646 B1 FR 2839646B1
- Authority
- FR
- France
- Prior art keywords
- applications
- quinoline derivatives
- integrase
- effect
- integrase effect
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Virology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Tropical Medicine & Parasitology (AREA)
- AIDS & HIV (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biotechnology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Quinoline Compounds (AREA)
Priority Applications (9)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0206126A FR2839646B1 (fr) | 2002-05-17 | 2002-05-17 | Utilisation de derives de quinoleine a effet anti-integrase et ses applications |
AU2003251047A AU2003251047A1 (en) | 2002-05-17 | 2003-05-15 | Use of quinoline derivatives with anti-integrase effect and applications thereof |
PCT/FR2003/001487 WO2003096965A2 (fr) | 2002-05-17 | 2003-05-15 | Derives de quinoleine a effet anti-integrase et leurs applications comme antiviraux |
EP03752821A EP1507532A2 (fr) | 2002-05-17 | 2003-05-15 | Utilisation de derives de quinoleine a effet anti-integrase et ses applications |
CA002489102A CA2489102A1 (fr) | 2002-05-17 | 2003-05-15 | Derives de quinoleine a effet anti-integrase et leurs applications comme antiviraux |
JP2004504964A JP2005531554A (ja) | 2002-05-17 | 2003-05-15 | 抗インテグラーゼ作用をもつキノリン誘導体類の利用およびそれらの応用 |
US10/514,631 US7479497B2 (en) | 2002-05-17 | 2003-05-15 | Use of quinoline derivatives with anti-integrase effect and applications thereof |
IL16526903A IL165269A0 (en) | 2002-05-17 | 2003-05-15 | Use of quinoline derivatives with anti-integrase effect and applications thereof |
US12/042,628 US20080161350A1 (en) | 2002-05-17 | 2008-03-05 | Use of quinoline derivatives with anti-integrase effect and applications thereof |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0206126A FR2839646B1 (fr) | 2002-05-17 | 2002-05-17 | Utilisation de derives de quinoleine a effet anti-integrase et ses applications |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2839646A1 FR2839646A1 (fr) | 2003-11-21 |
FR2839646B1 true FR2839646B1 (fr) | 2008-04-11 |
Family
ID=29286592
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR0206126A Expired - Fee Related FR2839646B1 (fr) | 2002-05-17 | 2002-05-17 | Utilisation de derives de quinoleine a effet anti-integrase et ses applications |
Country Status (8)
Country | Link |
---|---|
US (2) | US7479497B2 (fr) |
EP (1) | EP1507532A2 (fr) |
JP (1) | JP2005531554A (fr) |
AU (1) | AU2003251047A1 (fr) |
CA (1) | CA2489102A1 (fr) |
FR (1) | FR2839646B1 (fr) |
IL (1) | IL165269A0 (fr) |
WO (1) | WO2003096965A2 (fr) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20080280849A1 (en) * | 2005-06-01 | 2008-11-13 | Herve Leh | Synergic Combinations Comprising a Quinoline Compound and Other Hiv Infection Therapeutic Agents |
KR20100108337A (ko) * | 2007-11-15 | 2010-10-06 | 베링거 인겔하임 인터내셔날 게엠베하 | 사람 면역결핍 바이러스 복제의 억제제 |
ES2381234T3 (es) * | 2007-11-15 | 2012-05-24 | Gilead Sciences, Inc. | Inhibidores de la replicación del virus de la inmunodeficiencia humana |
WO2009062308A1 (fr) * | 2007-11-16 | 2009-05-22 | Boehringer Ingelheim International Gmbh | Inhibiteurs de la réplication du virus de l'immunodéficience humaine |
CA2707418C (fr) * | 2007-11-16 | 2013-11-19 | Boehringer Ingelheim International Gmbh | Inhibiteurs de la replication du virus de l'immunodeficience humaine |
CA2793959C (fr) | 2010-03-25 | 2019-06-04 | Oregon Health & Science University | Glycoproteines du cmv et vecteurs recombines |
SG186821A1 (en) * | 2010-07-02 | 2013-02-28 | Gilead Sciences Inc | 2 -quinolinyl- acetic acid derivatives as hiv antiviral compounds |
UY33480A (es) | 2010-07-02 | 2012-02-29 | Gilead Sciences Inc | Compuestos terapeuticos, composicion farmaceutica que lo comprende, metodo de tratamiento y su uso para la manufactura de un medicamento. |
ES2615734T3 (es) | 2011-04-21 | 2017-06-08 | Gilead Sciences, Inc. | Compuestos de benzotiazol y su uso farmacéutico |
HUE037408T2 (hu) | 2011-06-10 | 2018-08-28 | Univ Oregon Health & Science | CMV glikoproteinek és rekombináns vektorok |
BR112014013224B1 (pt) | 2011-11-30 | 2023-03-07 | Emory University | Inibidores de jak antivirais úteis no tratamento ou prevenção de infecções retrovirais e outras infecções virais |
US9284323B2 (en) | 2012-01-04 | 2016-03-15 | Gilead Sciences, Inc. | Naphthalene acetic acid derivatives against HIV infection |
WO2013103724A1 (fr) | 2012-01-04 | 2013-07-11 | Gilead Sciences, Inc. | Dérivés d'acide 2-(tert-butoxy)-2-(7-méthylquinoléin-6-yl)acétique pour traiter le sida |
BR112014018990A8 (pt) | 2012-04-20 | 2017-07-11 | Gilead Sciences Inc | Derivados de ácido benzotiazol-6-il acético e seu uso para tratamento de uma infecção |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2761687B1 (fr) * | 1997-04-08 | 2000-09-15 | Centre Nat Rech Scient | Derives de quinoleines, possedant notamment des proprietes antivirales, leurs preparations et leurs applications biologiques |
FR2830863B1 (fr) * | 2001-10-12 | 2004-01-30 | Bioalliance Pharma | Derives de quinoleine, procede de synthese, et medicaments renfermant ces derives |
-
2002
- 2002-05-17 FR FR0206126A patent/FR2839646B1/fr not_active Expired - Fee Related
-
2003
- 2003-05-15 WO PCT/FR2003/001487 patent/WO2003096965A2/fr active Application Filing
- 2003-05-15 IL IL16526903A patent/IL165269A0/xx unknown
- 2003-05-15 EP EP03752821A patent/EP1507532A2/fr not_active Ceased
- 2003-05-15 AU AU2003251047A patent/AU2003251047A1/en not_active Abandoned
- 2003-05-15 CA CA002489102A patent/CA2489102A1/fr not_active Abandoned
- 2003-05-15 US US10/514,631 patent/US7479497B2/en not_active Expired - Fee Related
- 2003-05-15 JP JP2004504964A patent/JP2005531554A/ja active Pending
-
2008
- 2008-03-05 US US12/042,628 patent/US20080161350A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
FR2839646A1 (fr) | 2003-11-21 |
US20050261336A1 (en) | 2005-11-24 |
CA2489102A1 (fr) | 2003-11-27 |
WO2003096965A2 (fr) | 2003-11-27 |
AU2003251047A8 (en) | 2003-12-02 |
WO2003096965A3 (fr) | 2004-04-22 |
US20080161350A1 (en) | 2008-07-03 |
AU2003251047A1 (en) | 2003-12-02 |
US7479497B2 (en) | 2009-01-20 |
IL165269A0 (en) | 2005-12-18 |
JP2005531554A (ja) | 2005-10-20 |
EP1507532A2 (fr) | 2005-02-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TQ | Partial transmission of property | ||
RM | Correction of a material error | ||
ST | Notification of lapse |
Effective date: 20130131 |