BR112022015771A2 - Compostos tetracíclicos para tratar a infecção por hiv - Google Patents

Compostos tetracíclicos para tratar a infecção por hiv

Info

Publication number
BR112022015771A2
BR112022015771A2 BR112022015771A BR112022015771A BR112022015771A2 BR 112022015771 A2 BR112022015771 A2 BR 112022015771A2 BR 112022015771 A BR112022015771 A BR 112022015771A BR 112022015771 A BR112022015771 A BR 112022015771A BR 112022015771 A2 BR112022015771 A2 BR 112022015771A2
Authority
BR
Brazil
Prior art keywords
compounds
hiv infection
tetracyclic compounds
treat hiv
tetracyclic
Prior art date
Application number
BR112022015771A
Other languages
English (en)
Inventor
Jiang Lan
w lin David
L Mitchell Michael
Roberts Ezra
M Schwarzwalder Gregg
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of BR112022015771A2 publication Critical patent/BR112022015771A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/22—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed systems contains four or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • AIDS & HIV (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

COMPOSTOS TETRACÍCLICOS PARA TRATAR A INFECÇÃO POR HIV A presente invenção refere-se, de modo geral, a certos compostos tetracíclicos, composições farmacêuticas compreendendo os ditos compostos e métodos de preparo e uso dos ditos compostos e composições farmacêuticas. Os compostos da invenção são úteis no tratamento ou na prevenção da infecção pelo vírus da imunodeficiência humana (HIV).
BR112022015771A 2020-02-24 2021-02-23 Compostos tetracíclicos para tratar a infecção por hiv BR112022015771A2 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US202062980857P 2020-02-24 2020-02-24
US202063036268P 2020-06-08 2020-06-08
US202063128670P 2020-12-21 2020-12-21
PCT/US2021/019179 WO2021173522A1 (en) 2020-02-24 2021-02-23 Tetracyclic compounds for treating hiv infection

Publications (1)

Publication Number Publication Date
BR112022015771A2 true BR112022015771A2 (pt) 2022-10-11

Family

ID=74885056

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112022015771A BR112022015771A2 (pt) 2020-02-24 2021-02-23 Compostos tetracíclicos para tratar a infecção por hiv

Country Status (15)

Country Link
US (2) US11697652B2 (pt)
EP (1) EP4110783A1 (pt)
JP (2) JP7453399B2 (pt)
CN (1) CN115151545A (pt)
AU (2) AU2021225809B2 (pt)
BR (1) BR112022015771A2 (pt)
CA (1) CA3166480A1 (pt)
CO (1) CO2022011947A2 (pt)
CR (1) CR20220418A (pt)
DO (1) DOP2022000171A (pt)
IL (1) IL295677A (pt)
MX (1) MX2022009871A (pt)
PE (1) PE20221569A1 (pt)
TW (2) TWI777425B (pt)
WO (1) WO2021173522A1 (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI4196479T1 (sl) 2021-01-19 2024-01-31 Gilead Sciences, Inc. Substituirane piridotriazinske spojine in njihove uporabe
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Publication number Publication date
EP4110783A1 (en) 2023-01-04
TW202140481A (zh) 2021-11-01
WO2021173522A1 (en) 2021-09-02
CR20220418A (es) 2022-10-10
DOP2022000171A (es) 2022-10-16
PE20221569A1 (es) 2022-10-06
JP7453399B2 (ja) 2024-03-19
US20240010650A1 (en) 2024-01-11
CO2022011947A2 (es) 2022-08-30
AU2023266279A1 (en) 2023-12-07
CN115151545A (zh) 2022-10-04
AU2021225809B2 (en) 2023-08-24
AU2021225809A1 (en) 2022-10-13
TWI777425B (zh) 2022-09-11
MX2022009871A (es) 2022-08-19
TW202248199A (zh) 2022-12-16
US11697652B2 (en) 2023-07-11
CA3166480A1 (en) 2021-09-02
IL295677A (en) 2022-10-01
JP2023514635A (ja) 2023-04-06
US20210284642A1 (en) 2021-09-16
JP2023184696A (ja) 2023-12-28

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