DK173330B1 - Pyrido(3,2,1-ij)-1,3,4-benzoxadiazin-derivater, en fremgangsmåde til fremstilling deraf, disse forbindelser til anvendelse - Google Patents

Pyrido(3,2,1-ij)-1,3,4-benzoxadiazin-derivater, en fremgangsmåde til fremstilling deraf, disse forbindelser til anvendelse Download PDF

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Publication number
DK173330B1
DK173330B1 DK198704772A DK477287A DK173330B1 DK 173330 B1 DK173330 B1 DK 173330B1 DK 198704772 A DK198704772 A DK 198704772A DK 477287 A DK477287 A DK 477287A DK 173330 B1 DK173330 B1 DK 173330B1
Authority
DK
Denmark
Prior art keywords
methyl
dihydro
pyrido
compound
oxo
Prior art date
Application number
DK198704772A
Other languages
Danish (da)
English (en)
Other versions
DK477287D0 (da
DK477287A (da
Inventor
Masahiro Aoki
Miyako Kamata
Tatsuo Ohtsuka
Nobuo Shimma
Kazuteru Yokose
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK477287D0 publication Critical patent/DK477287D0/da
Publication of DK477287A publication Critical patent/DK477287A/da
Application granted granted Critical
Publication of DK173330B1 publication Critical patent/DK173330B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/58—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK198704772A 1986-09-12 1987-09-11 Pyrido(3,2,1-ij)-1,3,4-benzoxadiazin-derivater, en fremgangsmåde til fremstilling deraf, disse forbindelser til anvendelse DK173330B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP86112619 1986-09-12
EP86112619 1986-09-12

Publications (3)

Publication Number Publication Date
DK477287D0 DK477287D0 (da) 1987-09-11
DK477287A DK477287A (da) 1988-03-13
DK173330B1 true DK173330B1 (da) 2000-07-24

Family

ID=8195410

Family Applications (1)

Application Number Title Priority Date Filing Date
DK198704772A DK173330B1 (da) 1986-09-12 1987-09-11 Pyrido(3,2,1-ij)-1,3,4-benzoxadiazin-derivater, en fremgangsmåde til fremstilling deraf, disse forbindelser til anvendelse

Country Status (22)

Country Link
JP (3) JPH0696578B2 (ja)
KR (1) KR960002857B1 (ja)
CN (1) CN1017800B (ja)
AT (1) AT389119B (ja)
AU (1) AU602534B2 (ja)
CA (1) CA1336905C (ja)
CZ (1) CZ281195B6 (ja)
DK (1) DK173330B1 (ja)
DZ (1) DZ1124A1 (ja)
FI (1) FI86428C (ja)
HU (1) HU199481B (ja)
IE (1) IE61624B1 (ja)
IL (1) IL83814A (ja)
MC (1) MC1850A1 (ja)
MX (1) MX8302A (ja)
NO (1) NO169125C (ja)
NZ (1) NZ221681A (ja)
PH (1) PH23930A (ja)
PT (1) PT85686B (ja)
SK (1) SK278990B6 (ja)
ZA (1) ZA876636B (ja)
ZW (1) ZW16387A1 (ja)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZW16387A1 (en) * 1986-09-12 1988-05-25 Hoffmann La Roche Tricyclic compounds
EP1757598A4 (en) 2004-05-13 2010-07-21 Daiichi Seiyaku Co SUBSTITUTED PYRROLIDINE DERIVATIVE
US7563805B2 (en) * 2005-05-19 2009-07-21 Daiichi Pharmaceutical Co., Ltd. Tri-, tetra-substituted-3-aminopyrrolidine derivative
EP2383271B1 (en) 2006-03-13 2013-07-10 Kyorin Pharmaceutical Co., Ltd. Aminoquinolones as GSK-3 Inhibitors
KR101563018B1 (ko) 2007-09-11 2015-10-23 교린 세이야꾸 가부시키 가이샤 Ｇｓｋ-３ 억제제로서의 시아노아미노퀴놀론 및 테트라졸로아미노퀴놀론
CN102344457B (zh) 2007-09-12 2015-07-22 杏林制药株式会社 作为 gsk-3 抑制剂的螺环状氨基喹诺酮
FR2928150A1 (fr) * 2008-02-29 2009-09-04 Vetoquinol Sa Sa Nouveaux derives 7-substitues de 3-carboxy-oxadiazino-quinolones, leur preparation et leur application comme anti-bacteriens
EP2145891A1 (en) * 2008-07-09 2010-01-20 Vetoquinol S.A. 9-substituted-5-carboxy-oxadiazino-quinolone derivatives, their preparation and their application as anti-bacterials
CA2755120C (en) 2009-03-11 2017-05-16 Kyorin Pharmaceutical Co., Ltd. 7-cycloalkylaminoquinolones as gsk-3 inhibitors
CN107522718B (zh) * 2017-09-14 2019-11-08 浙江国邦药业有限公司 一种马波沙星的合成方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZW16387A1 (en) * 1986-09-12 1988-05-25 Hoffmann La Roche Tricyclic compounds

Also Published As

Publication number Publication date
CN1017800B (zh) 1992-08-12
AU7811487A (en) 1988-03-17
CZ281195B6 (cs) 1996-07-17
DZ1124A1 (fr) 2004-09-13
NZ221681A (en) 1990-12-21
CZ660487A3 (en) 1996-04-17
JPH0826030B2 (ja) 1996-03-13
NO169125B (no) 1992-02-03
JPH0819120B2 (ja) 1996-02-28
CA1336905C (en) 1995-09-05
JPH07138256A (ja) 1995-05-30
JPH0696578B2 (ja) 1994-11-30
PH23930A (en) 1990-01-23
KR880003954A (ko) 1988-06-01
ZA876636B (en) 1988-07-27
MC1850A1 (fr) 1988-09-30
IE872444L (en) 1988-03-12
MX8302A (es) 1993-12-01
NO169125C (no) 1992-05-13
HUT47294A (en) 1989-02-28
PT85686A (en) 1987-10-01
DK477287D0 (da) 1987-09-11
JPS63132891A (ja) 1988-06-04
AU602534B2 (en) 1990-10-18
FI86428C (fi) 1992-08-25
FI86428B (fi) 1992-05-15
DK477287A (da) 1988-03-13
FI873940A0 (fi) 1987-09-11
FI873940A (fi) 1988-03-13
KR960002857B1 (ko) 1996-02-27
IL83814A (en) 1991-09-16
IE61624B1 (en) 1994-11-16
PT85686B (pt) 1990-05-31
HU199481B (en) 1990-02-28
ATA263887A (de) 1989-03-15
CN87106838A (zh) 1988-05-11
SK660487A3 (en) 1998-05-06
ZW16387A1 (en) 1988-05-25
JPH07138262A (ja) 1995-05-30
NO873816L (no) 1988-03-14
AT389119B (de) 1989-10-25
NO873816D0 (no) 1987-09-11
SK278990B6 (sk) 1998-05-06

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
CTFF Application for supplementary protection certificate (spc) filed

Free format text: CA 2000 00020, 20001024, EXPIRES: 20100210

PUP Patent expired