DK172397B1 - 5-Amino-8-phenyl-3H,6H-1,4,5a,8a-tetraazaacenaphthylen-3-on-forbindelser, farmaceutisk præparat og anvendelse af derivaterne til fremstilling af farmaceutisk præparat - Google Patents
5-Amino-8-phenyl-3H,6H-1,4,5a,8a-tetraazaacenaphthylen-3-on-forbindelser, farmaceutisk præparat og anvendelse af derivaterne til fremstilling af farmaceutisk præparat Download PDFInfo
- Publication number
- DK172397B1 DK172397B1 DK079589A DK79589A DK172397B1 DK 172397 B1 DK172397 B1 DK 172397B1 DK 079589 A DK079589 A DK 079589A DK 79589 A DK79589 A DK 79589A DK 172397 B1 DK172397 B1 DK 172397B1
- Authority
- DK
- Denmark
- Prior art keywords
- phenyl
- trifluoromethyl
- mixture
- tetraazaacenaphthylen
- stirred
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/16—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US15844888A | 1988-02-22 | 1988-02-22 | |
US15844888 | 1988-02-22 |
Publications (3)
Publication Number | Publication Date |
---|---|
DK79589D0 DK79589D0 (da) | 1989-02-21 |
DK79589A DK79589A (da) | 1989-08-23 |
DK172397B1 true DK172397B1 (da) | 1998-05-18 |
Family
ID=22568168
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK079589A DK172397B1 (da) | 1988-02-22 | 1989-02-21 | 5-Amino-8-phenyl-3H,6H-1,4,5a,8a-tetraazaacenaphthylen-3-on-forbindelser, farmaceutisk præparat og anvendelse af derivaterne til fremstilling af farmaceutisk præparat |
Country Status (23)
Country | Link |
---|---|
EP (1) | EP0329940B1 (de) |
JP (1) | JP2641556B2 (de) |
KR (1) | KR970009226B1 (de) |
AR (1) | AR247211A1 (de) |
AT (1) | ATE99686T1 (de) |
AU (1) | AU611769B2 (de) |
CA (1) | CA1329594C (de) |
CZ (1) | CZ284273B6 (de) |
DD (1) | DD283624A5 (de) |
DE (1) | DE68911951T2 (de) |
DK (1) | DK172397B1 (de) |
ES (1) | ES2061739T3 (de) |
FI (1) | FI89922C (de) |
HU (1) | HU203554B (de) |
IE (1) | IE64147B1 (de) |
IL (1) | IL88974A (de) |
NO (1) | NO169589C (de) |
NZ (1) | NZ228009A (de) |
PH (1) | PH26358A (de) |
PL (1) | PL158865B1 (de) |
PT (1) | PT89766B (de) |
SK (1) | SK105589A3 (de) |
ZA (1) | ZA891310B (de) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5013737A (en) * | 1988-02-22 | 1991-05-07 | American Cyanamid Company | 2,4,8-Trisubstituted-3H,6H-1,4,5A,8A-tetraazaacenaphtylene-3,5-(4H)-diones and 2,4-8-trisubstituted-4,5-dihydro-5-thioxo-3H,6H-1,4,5A,8A-tetrazaacenaphthylen-3-ones |
EP0562236A1 (de) * | 1992-03-26 | 1993-09-29 | American Cyanamid Company | Verfahren zur Synthese von 5-((substituierte)-Amino)-8-(Phenyl oder substituierte Phenyl)-3H,6H-1,4,5a,8a-Tetraazaacenaphthylen-3-Onen |
JP2001506998A (ja) * | 1996-12-19 | 2001-05-29 | アメリカン・サイアナミド・カンパニー | 好中球減少症の治療または抑制方法 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4236005A (en) * | 1979-07-02 | 1980-11-25 | American Cyanamid Company | Imidazo[1,5-a]pyrimidines |
US4713383A (en) * | 1984-10-01 | 1987-12-15 | Ciba-Geigy Corporation | Triazoloquinazoline compounds, and their methods of preparation, pharmaceutical compositions, and uses |
US4576943A (en) * | 1984-10-09 | 1986-03-18 | American Cyanamid Company | Pyrazolo[1,5-a]pyrimidines |
EP0264773A1 (de) * | 1986-10-16 | 1988-04-27 | American Cyanamid Company | 4,5-Dihydro- und 4,5,6,7-Tetrahydropyrazolo[1,5-a]pyrimidine |
-
1989
- 1989-01-16 AT AT89100657T patent/ATE99686T1/de active
- 1989-01-16 ES ES89100657T patent/ES2061739T3/es not_active Expired - Lifetime
- 1989-01-16 DE DE68911951T patent/DE68911951T2/de not_active Expired - Fee Related
- 1989-01-16 EP EP89100657A patent/EP0329940B1/de not_active Expired - Lifetime
- 1989-01-17 IL IL88974A patent/IL88974A/xx not_active IP Right Cessation
- 1989-02-16 NZ NZ228009A patent/NZ228009A/xx unknown
- 1989-02-17 CZ CS891055A patent/CZ284273B6/cs not_active IP Right Cessation
- 1989-02-17 SK SK1055-89A patent/SK105589A3/sk unknown
- 1989-02-20 PT PT89766A patent/PT89766B/pt not_active IP Right Cessation
- 1989-02-20 PH PH38218A patent/PH26358A/en unknown
- 1989-02-20 JP JP1038480A patent/JP2641556B2/ja not_active Expired - Lifetime
- 1989-02-20 CA CA000591526A patent/CA1329594C/en not_active Expired - Fee Related
- 1989-02-20 DD DD89325854A patent/DD283624A5/de unknown
- 1989-02-21 NO NO890724A patent/NO169589C/no not_active IP Right Cessation
- 1989-02-21 AU AU30172/89A patent/AU611769B2/en not_active Ceased
- 1989-02-21 AR AR89313253A patent/AR247211A1/es active
- 1989-02-21 IE IE54389A patent/IE64147B1/en not_active IP Right Cessation
- 1989-02-21 PL PL1989277837A patent/PL158865B1/pl unknown
- 1989-02-21 FI FI890826A patent/FI89922C/fi not_active IP Right Cessation
- 1989-02-21 DK DK079589A patent/DK172397B1/da not_active IP Right Cessation
- 1989-02-21 KR KR89002051A patent/KR970009226B1/ko not_active IP Right Cessation
- 1989-02-21 ZA ZA891310A patent/ZA891310B/xx unknown
- 1989-02-22 HU HU89856A patent/HU203554B/hu not_active IP Right Cessation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B1 | Patent granted (law 1993) | ||
PBP | Patent lapsed |