DK0720609T3 - 3-(5-Tetrazolylbenzyl)aminoperidinderivater og antagonister for tachykininer - Google Patents

3-(5-Tetrazolylbenzyl)aminoperidinderivater og antagonister for tachykininer

Info

Publication number
DK0720609T3
DK0720609T3 DK94927627T DK94927627T DK0720609T3 DK 0720609 T3 DK0720609 T3 DK 0720609T3 DK 94927627 T DK94927627 T DK 94927627T DK 94927627 T DK94927627 T DK 94927627T DK 0720609 T3 DK0720609 T3 DK 0720609T3
Authority
DK
Denmark
Prior art keywords
aminoperidine
tetrazolylbenzyl
tachykinins
antagonists
derivatives
Prior art date
Application number
DK94927627T
Other languages
Danish (da)
English (en)
Inventor
Duncan Robert Armour
Brian Evans
Gerard Martin Paul Giblin
Michael Menteith Hann
Maria Victoria Vinader
Stephen Watson
Neil Anthony Pegg
Alan Naylor
Xiao-Qing Lewell
David Middlemiss
Stephen Paul Watson
Tania Hubbard
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939319606A external-priority patent/GB9319606D0/en
Priority claimed from GB9326583A external-priority patent/GB9326583D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of DK0720609T3 publication Critical patent/DK0720609T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DK94927627T 1993-09-22 1994-09-20 3-(5-Tetrazolylbenzyl)aminoperidinderivater og antagonister for tachykininer DK0720609T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB939319606A GB9319606D0 (en) 1993-09-22 1993-09-22 Chemical compounds
GB9326583A GB9326583D0 (en) 1993-12-31 1993-12-31 Chemical compounds
PCT/EP1994/003129 WO1995008549A1 (en) 1993-09-22 1994-09-20 3-(5-tetrazolyl-benzyl)amino-piperidine derivatives and antagonists of tachykinins

Publications (1)

Publication Number Publication Date
DK0720609T3 true DK0720609T3 (da) 1999-07-26

Family

ID=26303560

Family Applications (1)

Application Number Title Priority Date Filing Date
DK94927627T DK0720609T3 (da) 1993-09-22 1994-09-20 3-(5-Tetrazolylbenzyl)aminoperidinderivater og antagonister for tachykininer

Country Status (29)

Country Link
US (2) US5703240A (cs)
EP (1) EP0720609B1 (cs)
JP (2) JP2865872B2 (cs)
CN (1) CN1061041C (cs)
AP (1) AP495A (cs)
AT (1) ATE173255T1 (cs)
AU (1) AU681190B2 (cs)
BG (1) BG62169B1 (cs)
CA (1) CA2172529A1 (cs)
CO (1) CO4290298A1 (cs)
CZ (1) CZ285479B6 (cs)
DE (1) DE69414590T2 (cs)
DK (1) DK0720609T3 (cs)
ES (1) ES2123829T3 (cs)
FI (1) FI961270A7 (cs)
GR (1) GR3029354T3 (cs)
HR (1) HRP940575B1 (cs)
HU (1) HU217428B (cs)
IL (1) IL111002A (cs)
IS (1) IS4208A (cs)
NO (1) NO307830B1 (cs)
NZ (1) NZ273614A (cs)
OA (1) OA10576A (cs)
PE (1) PE18295A1 (cs)
PL (1) PL179585B1 (cs)
SI (1) SI0720609T1 (cs)
SK (1) SK280901B6 (cs)
UA (1) UA44711C2 (cs)
WO (1) WO1995008549A1 (cs)

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Also Published As

Publication number Publication date
OA10576A (en) 2002-06-03
UA44711C2 (uk) 2002-03-15
IS4208A (is) 1995-03-23
DE69414590D1 (de) 1998-12-17
EP0720609A1 (en) 1996-07-10
PL313619A1 (en) 1996-07-08
US5703240A (en) 1997-12-30
DE69414590T2 (de) 1999-04-15
HK1004219A1 (en) 1998-11-20
AP495A (en) 1996-05-28
BG62169B1 (bg) 1999-04-30
IL111002A (en) 1998-09-24
CZ285479B6 (cs) 1999-08-11
HRP940575B1 (en) 2000-06-30
SK38396A3 (en) 1997-02-05
AP9400671A0 (en) 1994-10-31
HU217428B (hu) 2000-01-28
ES2123829T3 (es) 1999-01-16
AU7697494A (en) 1995-04-10
US5843966A (en) 1998-12-01
ATE173255T1 (de) 1998-11-15
GR3029354T3 (en) 1999-05-28
CO4290298A1 (es) 1996-04-17
CZ83096A3 (en) 1996-09-11
BG100487A (bg) 1996-12-31
HUT75648A (en) 1997-05-28
JP2865872B2 (ja) 1999-03-08
FI961270A0 (fi) 1996-03-19
PE18295A1 (es) 1995-07-27
WO1995008549A1 (en) 1995-03-30
FI961270A7 (fi) 1996-05-03
PL179585B1 (pl) 2000-09-29
JPH11106341A (ja) 1999-04-20
CN1135218A (zh) 1996-11-06
JPH09505275A (ja) 1997-05-27
HRP940575A2 (en) 1997-02-28
AU681190B2 (en) 1997-08-21
SI0720609T1 (en) 1999-02-28
HU9600722D0 (en) 1996-05-28
EP0720609B1 (en) 1998-11-11
NO307830B1 (no) 2000-06-05
CN1061041C (zh) 2001-01-24
NO961156L (no) 1996-05-21
NZ273614A (en) 1997-09-22
CA2172529A1 (en) 1995-03-30
SK280901B6 (sk) 2000-09-12
NO961156D0 (no) 1996-03-21
IL111002A0 (en) 1994-11-28

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