DE69414590D1 - 3-(5-tetrazolyl-benzyl) aminopiperidin-derivate und tachykinin antagonisten - Google Patents

3-(5-tetrazolyl-benzyl) aminopiperidin-derivate und tachykinin antagonisten

Info

Publication number
DE69414590D1
DE69414590D1 DE69414590T DE69414590T DE69414590D1 DE 69414590 D1 DE69414590 D1 DE 69414590D1 DE 69414590 T DE69414590 T DE 69414590T DE 69414590 T DE69414590 T DE 69414590T DE 69414590 D1 DE69414590 D1 DE 69414590D1
Authority
DE
Germany
Prior art keywords
tachykinine
tetrazolyl
antagonists
benzyl
aminopiperidine derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69414590T
Other languages
English (en)
Other versions
DE69414590T2 (de
Inventor
Duncan ARMOUR
Brian Evans
Gerard Giblin
Michael Hann
Tania Hubbard
Xiao-Qing Lewell
David Middlemiss
Alan Naylor
Neil Pegg
Maria Vinader
Stephen Watson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939319606A external-priority patent/GB9319606D0/en
Priority claimed from GB9326583A external-priority patent/GB9326583D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of DE69414590D1 publication Critical patent/DE69414590D1/de
Publication of DE69414590T2 publication Critical patent/DE69414590T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DE69414590T 1993-09-22 1994-09-20 3-(5-tetrazolyl-benzyl) aminopiperidin-derivate und tachykinin antagonisten Expired - Lifetime DE69414590T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB939319606A GB9319606D0 (en) 1993-09-22 1993-09-22 Chemical compounds
GB9326583A GB9326583D0 (en) 1993-12-31 1993-12-31 Chemical compounds
PCT/EP1994/003129 WO1995008549A1 (en) 1993-09-22 1994-09-20 3-(5-tetrazolyl-benzyl)amino-piperidine derivatives and antagonists of tachykinins

Publications (2)

Publication Number Publication Date
DE69414590D1 true DE69414590D1 (de) 1998-12-17
DE69414590T2 DE69414590T2 (de) 1999-04-15

Family

ID=26303560

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69414590T Expired - Lifetime DE69414590T2 (de) 1993-09-22 1994-09-20 3-(5-tetrazolyl-benzyl) aminopiperidin-derivate und tachykinin antagonisten

Country Status (30)

Country Link
US (2) US5703240A (de)
EP (1) EP0720609B1 (de)
JP (2) JP2865872B2 (de)
CN (1) CN1061041C (de)
AP (1) AP495A (de)
AT (1) ATE173255T1 (de)
AU (1) AU681190B2 (de)
BG (1) BG62169B1 (de)
CA (1) CA2172529A1 (de)
CO (1) CO4290298A1 (de)
CZ (1) CZ285479B6 (de)
DE (1) DE69414590T2 (de)
DK (1) DK0720609T3 (de)
ES (1) ES2123829T3 (de)
FI (1) FI961270A (de)
GR (1) GR3029354T3 (de)
HK (1) HK1004219A1 (de)
HR (1) HRP940575B1 (de)
HU (1) HU217428B (de)
IL (1) IL111002A (de)
IS (1) IS4208A (de)
NO (1) NO307830B1 (de)
NZ (1) NZ273614A (de)
OA (1) OA10576A (de)
PE (1) PE18295A1 (de)
PL (1) PL179585B1 (de)
SI (1) SI0720609T1 (de)
SK (1) SK280901B6 (de)
UA (1) UA44711C2 (de)
WO (1) WO1995008549A1 (de)

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Also Published As

Publication number Publication date
NO961156D0 (no) 1996-03-21
DK0720609T3 (da) 1999-07-26
NO961156L (no) 1996-05-21
NZ273614A (en) 1997-09-22
FI961270A (fi) 1996-05-03
PL179585B1 (pl) 2000-09-29
BG62169B1 (bg) 1999-04-30
WO1995008549A1 (en) 1995-03-30
SK280901B6 (sk) 2000-09-12
PL313619A1 (en) 1996-07-08
HU9600722D0 (en) 1996-05-28
IS4208A (is) 1995-03-23
JPH09505275A (ja) 1997-05-27
NO307830B1 (no) 2000-06-05
OA10576A (en) 2002-06-03
FI961270A0 (fi) 1996-03-19
PE18295A1 (es) 1995-07-27
HRP940575B1 (en) 2000-06-30
HU217428B (hu) 2000-01-28
AU681190B2 (en) 1997-08-21
AP495A (en) 1996-05-28
CN1061041C (zh) 2001-01-24
EP0720609A1 (de) 1996-07-10
AP9400671A0 (en) 1994-10-31
US5843966A (en) 1998-12-01
ATE173255T1 (de) 1998-11-15
BG100487A (bg) 1996-12-31
IL111002A (en) 1998-09-24
AU7697494A (en) 1995-04-10
GR3029354T3 (en) 1999-05-28
SK38396A3 (en) 1997-02-05
CN1135218A (zh) 1996-11-06
JPH11106341A (ja) 1999-04-20
CZ285479B6 (cs) 1999-08-11
SI0720609T1 (en) 1999-02-28
HRP940575A2 (en) 1997-02-28
CZ83096A3 (en) 1996-09-11
IL111002A0 (en) 1994-11-28
CO4290298A1 (es) 1996-04-17
US5703240A (en) 1997-12-30
ES2123829T3 (es) 1999-01-16
CA2172529A1 (en) 1995-03-30
JP2865872B2 (ja) 1999-03-08
UA44711C2 (uk) 2002-03-15
DE69414590T2 (de) 1999-04-15
HUT75648A (en) 1997-05-28
EP0720609B1 (de) 1998-11-11
HK1004219A1 (en) 1998-11-20

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