DE60209343T2 - Aminosäurekomplexe von c-arylglycosiden zur behandlung von diabetes und verfahren - Google Patents
Aminosäurekomplexe von c-arylglycosiden zur behandlung von diabetes und verfahren Download PDFInfo
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- DE60209343T2 DE60209343T2 DE60209343T DE60209343T DE60209343T2 DE 60209343 T2 DE60209343 T2 DE 60209343T2 DE 60209343 T DE60209343 T DE 60209343T DE 60209343 T DE60209343 T DE 60209343T DE 60209343 T2 DE60209343 T2 DE 60209343T2
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- compounds
- inhibitor
- agent
- alkyl
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- 238000000034 method Methods 0.000 title abstract description 11
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/351—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A—HUMAN NECESSITIES
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- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
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- Dermatology (AREA)
- Ophthalmology & Optometry (AREA)
- Child & Adolescent Psychology (AREA)
- Endocrinology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Saccharide Compounds (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US28309701P | 2001-04-11 | 2001-04-11 | |
| US283097P | 2001-04-11 | ||
| PCT/US2002/011066 WO2002083066A2 (en) | 2001-04-11 | 2002-04-08 | Amino acid complexes of c-aryl glucosides for treatment of diabetes and method |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE60209343D1 DE60209343D1 (de) | 2006-04-27 |
| DE60209343T2 true DE60209343T2 (de) | 2006-10-26 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE60209343T Expired - Fee Related DE60209343T2 (de) | 2001-04-11 | 2002-04-08 | Aminosäurekomplexe von c-arylglycosiden zur behandlung von diabetes und verfahren |
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| Country | Link |
|---|---|
| US (1) | US6774112B2 (enExample) |
| EP (1) | EP1385856B1 (enExample) |
| JP (1) | JP2004536047A (enExample) |
| AT (1) | ATE318272T1 (enExample) |
| AU (1) | AU2002254567B2 (enExample) |
| CA (1) | CA2444481A1 (enExample) |
| CY (1) | CY1105038T1 (enExample) |
| DE (1) | DE60209343T2 (enExample) |
| DK (1) | DK1385856T3 (enExample) |
| ES (1) | ES2258141T3 (enExample) |
| HU (1) | HUP0600232A2 (enExample) |
| WO (1) | WO2002083066A2 (enExample) |
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| CN1020944C (zh) * | 1990-01-30 | 1993-05-26 | 阿图尔-费希尔股份公司费希尔厂 | 紧固件 |
| US9006175B2 (en) | 1999-06-29 | 2015-04-14 | Mannkind Corporation | Potentiation of glucose elimination |
| US6515117B2 (en) * | 1999-10-12 | 2003-02-04 | Bristol-Myers Squibb Company | C-aryl glucoside SGLT2 inhibitors and method |
| EP1494732B1 (en) | 2002-03-20 | 2008-01-30 | MannKind Corporation | Inhalation apparatus |
| US20080260838A1 (en) * | 2003-08-01 | 2008-10-23 | Mannkind Corporation | Glucagon-like peptide 1 (glp-1) pharmaceutical formulations |
| TWI254635B (en) | 2002-08-05 | 2006-05-11 | Yamanouchi Pharma Co Ltd | Azulene derivative and salt thereof |
| US7790681B2 (en) | 2002-12-17 | 2010-09-07 | Amylin Pharmaceuticals, Inc. | Treatment of cardiac arrhythmias with GLP-1 receptor ligands |
| AU2003299966A1 (en) * | 2003-01-03 | 2004-08-10 | Bristol-Myers Squibb Company | Methods of producing c-aryl glucoside sglt2 inhibitors |
| RS20060320A (sr) * | 2003-08-01 | 2008-08-07 | Janssen Pharmaceutica N.V., | Supstituisani indazol-o-glukozidi |
| AU2004261660A1 (en) * | 2003-08-01 | 2005-02-10 | Janssen Pharmaceutica N.V. | Substituted fused heterocyclic C-glycosides |
| EP1680131A4 (en) * | 2003-08-01 | 2009-05-27 | Janssen Pharmaceutica Nv | SUBSTITUTED INDOLE-O-GLUCOSIDES |
| MXPA06001274A (es) * | 2003-08-01 | 2006-04-11 | Tanabe Seiyaku Co | Compuestos novedosos que poseen actividad inhibitoria contra transporador dependiente de sodio. |
| TW200524951A (en) | 2003-08-01 | 2005-08-01 | Janssen Pharmaceutica Nv | Substituted benzimidazole-, benztriazole-, and benzimidazolone-O-glucosides |
| US8785403B2 (en) | 2003-08-01 | 2014-07-22 | Mitsubishi Tanabe Pharma Corporation | Glucopyranoside compound |
| JP2006514649A (ja) * | 2003-12-17 | 2006-05-11 | アミリン・ファーマシューティカルズ，インコーポレイテッド | 腎症の治療および予防のための組成物 |
| EP1581246B1 (en) * | 2003-12-17 | 2013-01-16 | Amylin Pharmaceuticals, LLC | Compositions for the treatment and prevention of nephropathy |
| EP2360165A3 (de) | 2004-03-16 | 2012-01-04 | Boehringer Ingelheim International GmbH | Glucopyranosyl-substituierte Benzol-Derivate, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung |
| CA2568640C (en) | 2004-06-04 | 2011-08-09 | Teva Pharmaceutical Industries Ltd. | Pharmaceutical composition containing irbesartan |
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2002
- 2002-04-08 ES ES02723801T patent/ES2258141T3/es not_active Expired - Lifetime
- 2002-04-08 WO PCT/US2002/011066 patent/WO2002083066A2/en not_active Ceased
- 2002-04-08 AU AU2002254567A patent/AU2002254567B2/en not_active Ceased
- 2002-04-08 AT AT02723801T patent/ATE318272T1/de not_active IP Right Cessation
- 2002-04-08 CA CA002444481A patent/CA2444481A1/en not_active Abandoned
- 2002-04-08 US US10/117,914 patent/US6774112B2/en not_active Expired - Lifetime
- 2002-04-08 DK DK02723801T patent/DK1385856T3/da active
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- 2002-04-08 EP EP02723801A patent/EP1385856B1/en not_active Expired - Lifetime
- 2002-04-08 HU HU0600232A patent/HUP0600232A2/hu unknown
- 2002-04-08 JP JP2002580871A patent/JP2004536047A/ja active Pending
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2006
- 2006-05-19 CY CY20061100657T patent/CY1105038T1/el unknown
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| CA2444481A1 (en) | 2002-10-24 |
| JP2004536047A (ja) | 2004-12-02 |
| DE60209343D1 (de) | 2006-04-27 |
| CY1105038T1 (el) | 2010-03-03 |
| DK1385856T3 (da) | 2006-05-15 |
| HUP0600232A2 (en) | 2006-08-28 |
| AU2002254567B2 (en) | 2007-10-11 |
| ES2258141T3 (es) | 2006-08-16 |
| US6774112B2 (en) | 2004-08-10 |
| US20030064935A1 (en) | 2003-04-03 |
| EP1385856A2 (en) | 2004-02-04 |
| WO2002083066A3 (en) | 2003-03-06 |
| ATE318272T1 (de) | 2006-03-15 |
| EP1385856A4 (en) | 2005-05-11 |
| WO2002083066A2 (en) | 2002-10-24 |
| EP1385856B1 (en) | 2006-02-22 |
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