AU2002254567B2 - Amino acid complexes of C-aryl glucosides for treatment of diabetes and method - Google Patents

Amino acid complexes of C-aryl glucosides for treatment of diabetes and method Download PDF

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Publication number
AU2002254567B2
AU2002254567B2 AU2002254567A AU2002254567A AU2002254567B2 AU 2002254567 B2 AU2002254567 B2 AU 2002254567B2 AU 2002254567 A AU2002254567 A AU 2002254567A AU 2002254567 A AU2002254567 A AU 2002254567A AU 2002254567 B2 AU2002254567 B2 AU 2002254567B2
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AU
Australia
Prior art keywords
agent
inhibitor
compounds
compound
alkyl
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Ceased
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AU2002254567A
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AU2002254567A1 (en
Inventor
Jack Z. Gougoutas
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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Publication of AU2002254567A1 publication Critical patent/AU2002254567A1/en
Application granted granted Critical
Publication of AU2002254567B2 publication Critical patent/AU2002254567B2/en
Priority to AU2008200159A priority Critical patent/AU2008200159A1/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
AU2002254567A 2001-04-11 2002-04-08 Amino acid complexes of C-aryl glucosides for treatment of diabetes and method Ceased AU2002254567B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2008200159A AU2008200159A1 (en) 2001-04-11 2008-01-11 Amino acid complexes of C-aryl glucosides for treatment of diabetes and method

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28309701P 2001-04-11 2001-04-11
US60/283,097 2001-04-11
PCT/US2002/011066 WO2002083066A2 (en) 2001-04-11 2002-04-08 Amino acid complexes of c-aryl glucosides for treatment of diabetes and method

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU2008200159A Division AU2008200159A1 (en) 2001-04-11 2008-01-11 Amino acid complexes of C-aryl glucosides for treatment of diabetes and method

Publications (2)

Publication Number Publication Date
AU2002254567A1 AU2002254567A1 (en) 2003-04-17
AU2002254567B2 true AU2002254567B2 (en) 2007-10-11

Family

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Family Applications (1)

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AU2002254567A Ceased AU2002254567B2 (en) 2001-04-11 2002-04-08 Amino acid complexes of C-aryl glucosides for treatment of diabetes and method

Country Status (12)

Country Link
US (1) US6774112B2 (enExample)
EP (1) EP1385856B1 (enExample)
JP (1) JP2004536047A (enExample)
AT (1) ATE318272T1 (enExample)
AU (1) AU2002254567B2 (enExample)
CA (1) CA2444481A1 (enExample)
CY (1) CY1105038T1 (enExample)
DE (1) DE60209343T2 (enExample)
DK (1) DK1385856T3 (enExample)
ES (1) ES2258141T3 (enExample)
HU (1) HUP0600232A2 (enExample)
WO (1) WO2002083066A2 (enExample)

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JP2004536047A (ja) 2004-12-02
DE60209343D1 (de) 2006-04-27
CY1105038T1 (el) 2010-03-03
DK1385856T3 (da) 2006-05-15
HUP0600232A2 (en) 2006-08-28
ES2258141T3 (es) 2006-08-16
US6774112B2 (en) 2004-08-10
DE60209343T2 (de) 2006-10-26
US20030064935A1 (en) 2003-04-03
EP1385856A2 (en) 2004-02-04
WO2002083066A3 (en) 2003-03-06
ATE318272T1 (de) 2006-03-15
EP1385856A4 (en) 2005-05-11
WO2002083066A2 (en) 2002-10-24
EP1385856B1 (en) 2006-02-22

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