CZ416291A3 - Derivatives of cis, endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid, process of their preparation, compounds in which said derivatives are contained and their use - Google Patents

Derivatives of cis, endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid, process of their preparation, compounds in which said derivatives are contained and their use Download PDF

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Publication number
CZ416291A3
CZ416291A3 CS914162A CS416291A CZ416291A3 CZ 416291 A3 CZ416291 A3 CZ 416291A3 CS 914162 A CS914162 A CS 914162A CS 416291 A CS416291 A CS 416291A CZ 416291 A3 CZ416291 A3 CZ 416291A3
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CZ
Czechia
Prior art keywords
compound
formula
hydrogen
endo
cis
Prior art date
Application number
CS914162A
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Czech (cs)
English (en)
Inventor
Volker Dr Teetz
Rolf Prof Dr Geiger
Hansjorg Dr Urbach
Reinhard Dr Becker
Bernward Dr Scholkens
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Hoechst Ag
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25797115&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CZ416291(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of CZ416291A3 publication Critical patent/CZ416291A3/cs

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CS914162A 1981-11-05 1991-12-30 Derivatives of cis, endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid, process of their preparation, compounds in which said derivatives are contained and their use CZ416291A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3143946 1981-11-05
DE19823226768 DE3226768A1 (de) 1981-11-05 1982-07-17 Derivate der cis, endo-2-azabicyclo-(3.3.0)-octan-3-carbonsaeure, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung

Publications (1)

Publication Number Publication Date
CZ416291A3 true CZ416291A3 (en) 1993-09-15

Family

ID=25797115

Family Applications (1)

Application Number Title Priority Date Filing Date
CS914162A CZ416291A3 (en) 1981-11-05 1991-12-30 Derivatives of cis, endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid, process of their preparation, compounds in which said derivatives are contained and their use

Country Status (31)

Country Link
US (4) US4727160A (es)
EP (2) EP0079022B1 (es)
JP (3) JPH02104526A (es)
KR (1) KR890000007B1 (es)
AR (1) AR240675A1 (es)
AU (3) AU565200B2 (es)
BG (1) BG60532B2 (es)
CA (1) CA1187087A (es)
CS (1) CS247159B2 (es)
CZ (1) CZ416291A3 (es)
DD (2) DD219480A5 (es)
DE (3) DE3226768A1 (es)
DK (2) DK166624C (es)
DZ (1) DZ473A1 (es)
ES (3) ES8307746A1 (es)
FI (1) FI81087C (es)
GR (1) GR77381B (es)
HK (1) HK74889A (es)
HU (2) HU186339B (es)
IE (1) IE56476B1 (es)
IL (1) IL67172A (es)
JO (1) JO1224B1 (es)
LU (1) LU88260I2 (es)
MA (1) MA19639A1 (es)
NL (1) NL930039I2 (es)
NO (2) NO156940C (es)
NZ (1) NZ202378A (es)
PH (2) PH22417A (es)
PT (1) PT75792A (es)
SG (1) SG1189G (es)
SU (1) SU1277895A3 (es)

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