CY1114010T1 - Φαρμακευτικο σκευασμα που περιλαμβανει ενα ή περισσοτερους εστερες φουμαρικου οξεως με μητρα διαβρωσης - Google Patents

Φαρμακευτικο σκευασμα που περιλαμβανει ενα ή περισσοτερους εστερες φουμαρικου οξεως με μητρα διαβρωσης

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Publication number
CY1114010T1
CY1114010T1 CY20131100421T CY131100421T CY1114010T1 CY 1114010 T1 CY1114010 T1 CY 1114010T1 CY 20131100421 T CY20131100421 T CY 20131100421T CY 131100421 T CY131100421 T CY 131100421T CY 1114010 T1 CY1114010 T1 CY 1114010T1
Authority
CY
Cyprus
Prior art keywords
acid esters
fatty acid
erosion matrix
pharmaceutical form
erosion
Prior art date
Application number
CY20131100421T
Other languages
English (en)
Inventor
Henrik Nilsson
Roland Rupp
Original Assignee
Forward Pharma A/S
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42026676&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1114010(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Forward Pharma A/S filed Critical Forward Pharma A/S
Publication of CY1114010T1 publication Critical patent/CY1114010T1/el

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/194—Carboxylic acids, e.g. valproic acid having two or more carboxyl groups, e.g. succinic, maleic or phthalic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/225—Polycarboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/23—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin of acids having a carboxyl group bound to a chain of seven or more carbon atoms
    • A61K31/231—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin of acids having a carboxyl group bound to a chain of seven or more carbon atoms having one or two double bonds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
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    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
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  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Transplantation (AREA)
  • Inorganic Chemistry (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Ένα φαρμακευτικό σκεύασμα που περιλαμβάνει μια μήτρα διάβρωσης που περιλαμβάνει ένα ή περισσότερους εστέρες φουμαρικού οξέος καθώς και ένα ή περισσότερους παράγοντες που ελέγχουν το ρυθμό, όπου η διάβρωση της εν λόγω μήτρας διάβρωσης επιτρέπει την ελεγχόμενη αποσύνδεση του (των) εν λόγω εστέρα (εστέρων) φουμαρικού οξέος.
CY20131100421T 2009-01-09 2013-05-29 Φαρμακευτικο σκευασμα που περιλαμβανει ενα ή περισσοτερους εστερες φουμαρικου οξεως με μητρα διαβρωσης CY1114010T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US14361309P 2009-01-09 2009-01-09
DKPA200900034 2009-01-09
EP10700730.4A EP2379063B2 (en) 2009-01-09 2010-01-08 Pharmaceutical formulation comprising one or more fumaric acid esters in an erosion matrix

Publications (1)

Publication Number Publication Date
CY1114010T1 true CY1114010T1 (el) 2016-07-27

Family

ID=42026676

Family Applications (2)

Application Number Title Priority Date Filing Date
CY20131100421T CY1114010T1 (el) 2009-01-09 2013-05-29 Φαρμακευτικο σκευασμα που περιλαμβανει ενα ή περισσοτερους εστερες φουμαρικου οξεως με μητρα διαβρωσης
CY20161100739T CY1117847T1 (el) 2009-01-09 2016-07-27 Φαρμακευτικο σκευασμα που περιλαμβανει ενα ή περισσοτερους εστερες φουμαρικου οξεος σε μητρα διαβρωσης

Family Applications After (1)

Application Number Title Priority Date Filing Date
CY20161100739T CY1117847T1 (el) 2009-01-09 2016-07-27 Φαρμακευτικο σκευασμα που περιλαμβανει ενα ή περισσοτερους εστερες φουμαρικου οξεος σε μητρα διαβρωσης

Country Status (19)

Country Link
US (5) US8906420B2 (el)
EP (4) EP2564839B1 (el)
JP (3) JP5788331B2 (el)
KR (1) KR101699912B1 (el)
CN (2) CN102369001A (el)
CY (2) CY1114010T1 (el)
DK (2) DK2379063T4 (el)
EA (1) EA201290596A1 (el)
ES (2) ES2586761T3 (el)
HK (1) HK1180943A1 (el)
HR (2) HRP20130480T4 (el)
HU (1) HUE030169T2 (el)
PL (2) PL2564839T3 (el)
PT (2) PT2379063E (el)
RU (2) RU2552951C2 (el)
SI (2) SI2564839T1 (el)
SM (1) SMT201300065B (el)
UA (3) UA112975C2 (el)
WO (1) WO2010079222A1 (el)

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