EA201290596A1 - Фармацевтический состав, содержащий один или более эфиров фумаровой кислоты в разлагаемой матрице - Google Patents

Фармацевтический состав, содержащий один или более эфиров фумаровой кислоты в разлагаемой матрице

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Publication number
EA201290596A1
EA201290596A1 EA201290596A EA201290596A EA201290596A1 EA 201290596 A1 EA201290596 A1 EA 201290596A1 EA 201290596 A EA201290596 A EA 201290596A EA 201290596 A EA201290596 A EA 201290596A EA 201290596 A1 EA201290596 A1 EA 201290596A1
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EA
Eurasian Patent Office
Prior art keywords
pharmaceutical composition
composition containing
matrix
decompated
ethers
Prior art date
Application number
EA201290596A
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English (en)
Inventor
Хенрик Нильссон
Роланд Рупп
Original Assignee
Форвард Фарма А/С
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42026676&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201290596(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Форвард Фарма А/С filed Critical Форвард Фарма А/С
Publication of EA201290596A1 publication Critical patent/EA201290596A1/ru

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/194Carboxylic acids, e.g. valproic acid having two or more carboxyl groups, e.g. succinic, maleic or phthalic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/225Polycarboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
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    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/23Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin of acids having a carboxyl group bound to a chain of seven or more carbon atoms
    • A61K31/231Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin of acids having a carboxyl group bound to a chain of seven or more carbon atoms having one or two double bonds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
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    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
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    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K9/2886Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
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    • A61P5/14Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
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Abstract

Фармацевтический состав, содержащий разлагаемую матрицу, содержащую один или более эфиров фумаровой кислоты, а также один или более контролирующих скорость агентов, при этом разложение указанной разлагаемой матрицы обеспечивает контролируемое высвобождение указанного эфира (эфиров) фумаровой кислоты.
EA201290596A 2009-01-09 2010-01-08 Фармацевтический состав, содержащий один или более эфиров фумаровой кислоты в разлагаемой матрице EA201290596A1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US14361309P 2009-01-09 2009-01-09
DKPA200900034 2009-01-09
PCT/EP2010/050172 WO2010079222A1 (en) 2009-01-09 2010-01-08 Pharmaceutical formulation comprising one or more fumaric acid esters in an erosion matrix

Publications (1)

Publication Number Publication Date
EA201290596A1 true EA201290596A1 (ru) 2013-01-30

Family

ID=42026676

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201290596A EA201290596A1 (ru) 2009-01-09 2010-01-08 Фармацевтический состав, содержащий один или более эфиров фумаровой кислоты в разлагаемой матрице

Country Status (19)

Country Link
US (5) US8906420B2 (ru)
EP (4) EP3090733A1 (ru)
JP (3) JP5788331B2 (ru)
KR (1) KR101699912B1 (ru)
CN (2) CN109044985A (ru)
CY (2) CY1114010T1 (ru)
DK (2) DK2379063T4 (ru)
EA (1) EA201290596A1 (ru)
ES (2) ES2411972T5 (ru)
HK (1) HK1180943A1 (ru)
HR (2) HRP20130480T4 (ru)
HU (1) HUE030169T2 (ru)
PL (2) PL2564839T3 (ru)
PT (2) PT2564839T (ru)
RU (2) RU2743637C2 (ru)
SI (2) SI2379063T2 (ru)
SM (1) SMT201300065B (ru)
UA (3) UA103844C2 (ru)
WO (1) WO2010079222A1 (ru)

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