CS240966B2 - Preparation method of 1-ethoxycarbonyloxyethylester of 6-(d-(-)-alfa-amino-phenylacetoamido)penicilane acid - Google Patents

Preparation method of 1-ethoxycarbonyloxyethylester of 6-(d-(-)-alfa-amino-phenylacetoamido)penicilane acid Download PDF

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Publication number
CS240966B2
CS240966B2 CS834857A CS485783A CS240966B2 CS 240966 B2 CS240966 B2 CS 240966B2 CS 834857 A CS834857 A CS 834857A CS 485783 A CS485783 A CS 485783A CS 240966 B2 CS240966 B2 CS 240966B2
Authority
CS
Czechoslovakia
Prior art keywords
alpha
formula
acid
ester
preparation
Prior art date
Application number
CS834857A
Other languages
Czech (cs)
English (en)
Other versions
CS485783A2 (en
Inventor
Luigi Ratti
Drek R Palmer
Robert G Tyson
Original Assignee
Astra Laekemedel Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Laekemedel Ab filed Critical Astra Laekemedel Ab
Priority to CS849086A priority Critical patent/CS251087B2/cs
Priority to CS849085A priority patent/CS251086B2/cs
Publication of CS485783A2 publication Critical patent/CS485783A2/cs
Publication of CS240966B2 publication Critical patent/CS240966B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/96—Esters of carbonic or haloformic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CS834857A 1982-06-29 1983-06-29 Preparation method of 1-ethoxycarbonyloxyethylester of 6-(d-(-)-alfa-amino-phenylacetoamido)penicilane acid CS240966B2 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
CS849086A CS251087B2 (cs) 1982-06-29 1984-11-27 Způsob výroby ethoxykarbonyloxyethylesteru kyseliny 6- [D-(—) -ar-amino-a-fenylacetamido)penicilanové
CS849085A CS251086B2 (cs) 1982-11-16 1984-11-27 Zp&iob výroby ethoxykarbonyloxyethylesteru penicilinu G

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT22141/82A IT1190897B (it) 1982-06-29 1982-06-29 Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico

Publications (2)

Publication Number Publication Date
CS485783A2 CS485783A2 (en) 1985-06-13
CS240966B2 true CS240966B2 (en) 1986-03-13

Family

ID=11192093

Family Applications (1)

Application Number Title Priority Date Filing Date
CS834857A CS240966B2 (en) 1982-06-29 1983-06-29 Preparation method of 1-ethoxycarbonyloxyethylester of 6-(d-(-)-alfa-amino-phenylacetoamido)penicilane acid

Country Status (12)

Country Link
US (1) US4619785A (ru)
JP (1) JPS5920287A (ru)
BE (1) BE897161A (ru)
CA (1) CA1236450A (ru)
CS (1) CS240966B2 (ru)
IT (1) IT1190897B (ru)
LT (1) LT2254B (ru)
PH (1) PH21849A (ru)
PL (1) PL140499B1 (ru)
RO (1) RO86529B (ru)
SU (1) SU1245262A3 (ru)
ZA (1) ZA834370B (ru)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE43833T1 (de) * 1982-11-04 1989-06-15 Astra Laekemedel Ab Verfahren zur herstellung des 1'ethoxycarbonyloxyethylestersvon benzylpenicillin.
IL67637A0 (en) * 1983-01-07 1983-05-15 Orvet Bv Preparation of 1'-ethoxycarbonyl-oxyethyl esters of penicillins and novel intermediates
IL67177A (en) * 1982-11-04 1985-08-30 Orvet Bv 1-bromoethyl ethyl carbonate,methods for its preparation and 1-bromoethylchloroformate and 1-bromoethylbromoformate obtained as intermediates
JPS6124595A (ja) * 1984-07-10 1986-02-03 株式会社　鍾根堂 α−アミノベンジルペニシリンのエステル化合物の製造方法
JPH0740661B2 (ja) * 1985-09-11 1995-05-01 セイコーエプソン株式会社 自動選局回路
CN103450224A (zh) * 2013-08-29 2013-12-18 东北制药集团股份有限公司 一种头孢噻利δ3异构体的制备方法

Family Cites Families (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB991586A (en) * 1963-02-28 1965-05-12 Beecham Res Lab Process for the preparation of penicillins
GB1033257A (en) * 1964-04-23 1966-06-22 Beecham Group Ltd Penicillins
CH516593A (de) * 1967-09-29 1971-12-15 Leo Pharm Prod Ltd Verfahren zur Herstellung von neuen Estern von a-Aminobenzyl-penicillin
US3697507A (en) * 1968-09-26 1972-10-10 Leo Pharm Prod Ltd Esters of {60 -aminobenzylpenicillin
GB1302917A (ru) * 1970-07-14 1973-01-10
US3873521A (en) * 1970-09-17 1975-03-25 Astra Laekemedel Ab Esters of {60 -amino penicillins
IE35648B1 (en) * 1970-09-25 1976-04-14 Beecham Group Ltd Penicillins
BE756806A (en) * 1970-09-29 1971-03-29 Vnii Antibiotikov Process for 6-(d(-)-alpha-amino-phenylacet- - amido)-penicillanic acid
GB1347979A (en) * 1970-11-12 1974-02-27 Beecham Group Ltd Penicillins
DE2161420A1 (de) * 1970-12-30 1972-07-27 Toyama Chemical Co. Ltd., Tokio Penicillinderivate und Verfahren zu deren Herstellung
GB1390754A (en) * 1971-06-09 1975-04-16 Beecham Group Ltd Penicillin and cephalosporin esters
GB1377817A (en) * 1971-06-09 1974-12-18 Beecham Group Ltd Penicillins and cephalosporins
GB1364672A (en) * 1971-06-09 1974-08-29 Beecham Group Ltd Penicillins
DE2228670A1 (de) * 1971-06-15 1973-01-11 Yamanouchi Pharma Co Ltd Neue oxymethylesterderivate von penicillin und cephalosporin
GB1433131A (en) * 1972-03-13 1976-04-22 Astra Laekemedel Ab Penicillins
GB1426717A (en) * 1972-03-13 1976-03-03 Astra Laekemedel Ab Penicillins
GB1426869A (en) * 1972-03-13 1976-03-03 Astra Laekemedel Ab Penicillins
GB1425571A (en) * 1972-03-13 1976-02-18 Astra Laekemedel Ab Penicillins and cephaosporins
GB1427139A (en) * 1972-03-13 1976-03-10 Astra Laekemedel Ab Penicillins
SE397981B (sv) * 1973-02-19 1977-11-28 Astra Laekemedel Ab Nya tetraalkylammoniumsalter av 6-aminopenicillansyra och av bensylpenicillin avsedda att anvendas som mellanprodukter vid framstellning av vissa estrar av 6-aminopenicillansyra och av bensylpenicillin
GB1435847A (en) * 1973-07-17 1976-05-19 Landerlan Sa Lab Esters of alpha-alkylidene-aminobenzyl penicillins
YU125575A (en) * 1974-05-20 1982-05-31 Lilly Co Eli Process for obtaining 3-cephalosporinic esters
GB1598568A (en) * 1977-04-19 1981-09-23 Glaxo Lab Ltd Esters of(6r,7r)-3-carbamoyloxymethyl-7-((z)-2-(fur-2-yl)-2-methoxyiminoacetamido)-ceph-3-em-4-carboxylic acid
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
SE449103B (sv) * 1979-03-05 1987-04-06 Pfizer Sett att framstella penicillansyra-1,1-dioxid samt estrar derav
GB2111043B (en) * 1980-12-12 1985-02-06 Ciba Geigy Ag Novel cephalosporin esters

Also Published As

Publication number Publication date
PH21849A (en) 1988-03-17
LT2254B (lt) 1993-11-15
US4619785A (en) 1986-10-28
ZA834370B (en) 1984-03-28
SU1245262A3 (ru) 1986-07-15
RO86529A (ro) 1985-03-15
PL140499B1 (en) 1987-04-30
IT8222141A0 (it) 1982-06-29
IT8222141A1 (it) 1983-12-29
RO86529B (ro) 1985-04-01
BE897161A (fr) 1983-12-29
CS485783A2 (en) 1985-06-13
IT1190897B (it) 1988-02-24
PL242730A1 (en) 1985-03-12
JPH045032B2 (ru) 1992-01-30
CA1236450A (en) 1988-05-10
JPS5920287A (ja) 1984-02-01

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