CS208114B2 - Method of making the new 4-substituted thiazol-2-exan acids - Google Patents
Method of making the new 4-substituted thiazol-2-exan acids Download PDFInfo
- Publication number
- CS208114B2 CS208114B2 CS794390A CS439079A CS208114B2 CS 208114 B2 CS208114 B2 CS 208114B2 CS 794390 A CS794390 A CS 794390A CS 439079 A CS439079 A CS 439079A CS 208114 B2 CS208114 B2 CS 208114B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- thiazole
- acid
- hydrogen
- oxamic acid
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19782828091 DE2828091A1 (de) | 1978-06-27 | 1978-06-27 | 4-substituierte thiazoloxamsaeuren sowie ihre salze und ester |
Publications (1)
Publication Number | Publication Date |
---|---|
CS208114B2 true CS208114B2 (en) | 1981-08-31 |
Family
ID=6042852
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS794390A CS208114B2 (en) | 1978-06-27 | 1979-06-26 | Method of making the new 4-substituted thiazol-2-exan acids |
Country Status (36)
Country | Link |
---|---|
US (1) | US4238496A (fr) |
JP (1) | JPS557290A (fr) |
AT (1) | AT373884B (fr) |
AU (1) | AU525312B2 (fr) |
BE (1) | BE877293A (fr) |
BG (1) | BG30324A3 (fr) |
CA (1) | CA1246071A (fr) |
CH (1) | CH644370A5 (fr) |
CS (1) | CS208114B2 (fr) |
DD (1) | DD144542A5 (fr) |
DE (1) | DE2828091A1 (fr) |
DK (1) | DK147940C (fr) |
ES (1) | ES481917A1 (fr) |
FI (1) | FI69456C (fr) |
FR (1) | FR2429787A1 (fr) |
GB (1) | GB2023580B (fr) |
GR (1) | GR69231B (fr) |
HK (1) | HK66285A (fr) |
HU (1) | HU178996B (fr) |
IE (1) | IE48357B1 (fr) |
IL (1) | IL57659A0 (fr) |
IT (1) | IT1120443B (fr) |
LU (1) | LU81424A1 (fr) |
MY (1) | MY8600653A (fr) |
NL (1) | NL7904957A (fr) |
NO (1) | NO151500C (fr) |
NZ (1) | NZ190842A (fr) |
PH (1) | PH17226A (fr) |
PL (1) | PL117333B1 (fr) |
PT (1) | PT69822A (fr) |
RO (1) | RO77553A (fr) |
SE (1) | SE446182B (fr) |
SG (1) | SG61985G (fr) |
SU (1) | SU791237A3 (fr) |
YU (1) | YU41645B (fr) |
ZA (1) | ZA793176B (fr) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4321372A (en) * | 1980-06-16 | 1982-03-23 | Pfizer Inc. | Antiulcer thiazol-2-ylcarbamoyl-carboxylic acids, esters and amides |
DE3027528A1 (de) * | 1980-07-19 | 1982-02-18 | Basf Ag, 6700 Ludwigshafen | Ueberbrueckte thiazolyloxamidsaeure-derivate, verfahren zu ihrer herstellung und diese enthaltende therapeutische mittel |
DE3027527A1 (de) | 1980-07-19 | 1982-02-18 | Basf Ag, 6700 Ludwigshafen | Neue oxamidsaeure-derivate, verfahren zu ihrer herstellung und diese enthaltende therapeutische mittel |
FR2494272A1 (fr) * | 1980-11-19 | 1982-05-21 | Fabre Sa Pierre | Derives de l'acide thiazolyl-2 oxamique substitues en position 4 par un radical thienyle ou furyle, leur preparation et leur utilisation comme medicaments |
DE3135250A1 (de) * | 1981-09-05 | 1983-03-17 | Basf Ag, 6700 Ludwigshafen | Tricyclische thiazolyloxamate, verfahren zu ihrer herstellung und diese enthaltende therapeutische mittel |
ATE38224T1 (de) * | 1983-09-01 | 1988-11-15 | Boehringer Ingelheim Ltd | Diazin-ethenylphenyloxamidsaeuren und deren ester und salze. |
US4788198A (en) * | 1983-09-01 | 1988-11-29 | Boehringer Ingelheim Pharmaceuticals, Inc. | Diazine-ethyenylphenyl oxamic acids and esters and salts thereof |
US4681884A (en) * | 1983-09-01 | 1987-07-21 | Boehringer Ingelheim Pharmaceuticals, Inc. | Diazine-ethenylphenyl oxamic acids and esters and salts thereof |
IT1204959B (it) * | 1987-03-25 | 1989-03-10 | Zambon Farmaceutici Spa | Composti dotati di attivita' antiallergica |
IT1204960B (it) * | 1987-03-25 | 1989-03-10 | Zambon Farmaceutici Spa | Composti dotati di attivita' antiallergica |
DE3807232A1 (de) * | 1988-03-05 | 1989-09-14 | Bayer Ag | Substituierte acrylsaeureester |
JPH0667836B2 (ja) * | 1989-03-01 | 1994-08-31 | 東洋紡績株式会社 | アミド系化合物からなる抗アレルギー剤 |
FR2671552B1 (fr) * | 1991-01-15 | 1993-05-07 | Pf Medicament | Procede de preparation de thiazolyl-2 oxamates d'alkyle. |
EP1027050B1 (fr) * | 1997-10-27 | 2004-01-14 | Takeda Chemical Industries, Ltd. | 1,3-thiazoles comme antagonistes des recepteurs de l'adenosine a3 pour le traitement de l'allergie, de l'asthme et du diabete |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1062245B (de) * | 1957-10-17 | 1959-07-30 | Ciba Geigy | Verfahren zur Herstellung von 2-Amino-4-pyridyl-(2')-thiazol und seinen Salzen |
FR1526074A (fr) * | 1967-03-22 | 1968-05-24 | Rech S Ind S O R I Soc D | Méthoxy-phényl-amino-2-thiazoles, leurs amides et leurs procédés de préparation |
BE795907A (fr) * | 1972-02-25 | 1973-06-18 | Luso Farmaco Inst | 2-amino-4-arylthiazoles 5-substitues et leur preparation |
US3966965A (en) * | 1973-03-23 | 1976-06-29 | American Home Products Corporation | Oxamic acid derivatives for the prevention of immediate type hypersensitivity reactions |
US4054666A (en) * | 1973-03-23 | 1977-10-18 | American Home Products Corporation | Compositions and methods of treating immediate hypersensitivity reactions with thiazolyl oxamic acid derivatives |
FR2429210A1 (fr) * | 1978-06-19 | 1980-01-18 | Fabre Sa Pierre | Derives de phenyl-4 thiazolyl-2 oxamates utiles dans le traitement de l'asthme |
-
1978
- 1978-06-27 DE DE19782828091 patent/DE2828091A1/de active Granted
-
1979
- 1979-06-18 GR GR59370A patent/GR69231B/el unknown
- 1979-06-18 US US06/049,173 patent/US4238496A/en not_active Expired - Lifetime
- 1979-06-19 AT AT0431879A patent/AT373884B/de active
- 1979-06-20 SU SU792776204A patent/SU791237A3/ru active
- 1979-06-22 DD DD79213848A patent/DD144542A5/de not_active IP Right Cessation
- 1979-06-22 CH CH588679A patent/CH644370A5/de not_active IP Right Cessation
- 1979-06-25 LU LU81424A patent/LU81424A1/de unknown
- 1979-06-25 BG BG7944041A patent/BG30324A3/xx unknown
- 1979-06-25 FI FI792006A patent/FI69456C/fi not_active IP Right Cessation
- 1979-06-25 YU YU1497/79A patent/YU41645B/xx unknown
- 1979-06-25 IT IT49533/79A patent/IT1120443B/it active
- 1979-06-26 SE SE7905608A patent/SE446182B/sv not_active IP Right Cessation
- 1979-06-26 CS CS794390A patent/CS208114B2/cs unknown
- 1979-06-26 RO RO7997961A patent/RO77553A/fr unknown
- 1979-06-26 DK DK269879A patent/DK147940C/da not_active IP Right Cessation
- 1979-06-26 PL PL1979216608A patent/PL117333B1/pl unknown
- 1979-06-26 HU HU79BO1794A patent/HU178996B/hu not_active IP Right Cessation
- 1979-06-26 AU AU48397/79A patent/AU525312B2/en not_active Ceased
- 1979-06-26 NZ NZ190842A patent/NZ190842A/xx unknown
- 1979-06-26 CA CA000330575A patent/CA1246071A/fr not_active Expired
- 1979-06-26 NO NO792139A patent/NO151500C/no unknown
- 1979-06-26 PH PH22688A patent/PH17226A/en unknown
- 1979-06-26 PT PT69822A patent/PT69822A/pt unknown
- 1979-06-26 GB GB7922155A patent/GB2023580B/en not_active Expired
- 1979-06-26 ES ES481917A patent/ES481917A1/es not_active Expired
- 1979-06-26 JP JP8062879A patent/JPS557290A/ja active Granted
- 1979-06-26 ZA ZA793176A patent/ZA793176B/xx unknown
- 1979-06-26 IL IL57659A patent/IL57659A0/xx not_active IP Right Cessation
- 1979-06-26 NL NL7904957A patent/NL7904957A/nl not_active Application Discontinuation
- 1979-06-26 BE BE0/195981A patent/BE877293A/fr not_active IP Right Cessation
- 1979-06-27 FR FR7916627A patent/FR2429787A1/fr active Granted
- 1979-08-08 IE IE1200/79A patent/IE48357B1/en not_active IP Right Cessation
-
1985
- 1985-08-23 SG SG619/85A patent/SG61985G/en unknown
- 1985-09-05 HK HK662/85A patent/HK66285A/xx unknown
-
1986
- 1986-12-30 MY MY653/86A patent/MY8600653A/xx unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
KR100371297B1 (ko) | 치환된티아졸리딘디온유도체 | |
CS208114B2 (en) | Method of making the new 4-substituted thiazol-2-exan acids | |
US4581363A (en) | Furo-(3,4-C)-pyridine derivatives and therapeutic compositions containing the same | |
EP0984934B1 (fr) | Nouveaux chelateurs du fer (iii) agissant par la voie orale | |
US4735950A (en) | Furo-(3,4-C)-pyridine derivatives and therapeutic composition containing the same | |
NL7909024A (nl) | 1,4-dihydropyridinen en werkwijzen voor het bereiden en toepassen van deze verbindingen. | |
KR100608416B1 (ko) | 2-(n-시아노이미노)티아졸리딘-4-온 유도체 | |
CZ279917B6 (cs) | Thiazolidinové sloučeniny obsahující chinonovou skupinu, způsob výroby a farmaceutické prostředky s jejich obsahem | |
CZ284238B6 (cs) | Substituované beta-diketony, způsob jejich výroby a farmaceutický přípravek, který je obsahuje | |
CS226020B2 (en) | Method of preparing pyridine and pyrimidine derivatives | |
US3467715A (en) | 2,4-diloweralkanoyl phloroglucinol derivatives | |
US3883546A (en) | S-heterocyclic derivatives of phosphine or phosphite gold mercaptides | |
JPS60104084A (ja) | 4H‐ベンゾ〔4,5〕シクロヘプタ〔1,2‐b〕チオフエン誘導体 | |
NL7906339A (nl) | Hydroxyalkaanzuurderivaten en werkwijzen voor het bereiden en toepassen van deze derivaten. | |
KR820001995B1 (ko) | 4-치환티아졸-2-옥삼산의 제조방법 | |
US3766245A (en) | 3,5-dialkoxyalkoxy-4-substituted benzoic acid esters | |
US4820837A (en) | 1-hydroxy-oxo-5H-pyrido(3,2-a)phenoxazine-3-carboxylic acid esters | |
RU2068415C1 (ru) | 5,7-диокси-2-метил-8-/4-(3-окси-1-(1-пропил)пиперидинил/-4н-1-бензопиран-4-он или его стереоизомеры или фармакологически приемлемые кислотно-аддитивные соли и способ их получения | |
KR970003126B1 (ko) | 디티올란 유도체 | |
US4427683A (en) | Antiinflammatory 2'-pyridyl-1'-oxide carbothiolate and carbodithioate compounds | |
US3947565A (en) | Anti-arthritic compositions comprising s-heterocyclic derivatives of phosphine or phosphite gold mercaptides and methods of producing anti-arthritic activity | |
IL43667A (en) | 2,7 bis-dialkylaminoalkyl esters and ethers of 9-benzylidenefluorene | |
JP2003505357A (ja) | ビス第4アンモニウム塩の前駆体及び駆虫活性をもつプロドラッグとしてのその応用 | |
HUT68502A (en) | 1-(4-oxo-thiazolidin-2-yliden)-isothiosemicarbazide derivatives, pharmaceutical preparations containing them and their preparations | |
KR820000097B1 (ko) | 피리도[2,1-b] 퀴나졸린 유도체의 제조방법 |