CN1416425A - 1,5－苯并硫氮杂䓬及其它们作为促血清脂质降低剂的用途 - Google Patents

1,5－苯并硫氮杂䓬及其它们作为促血清脂质降低剂的用途 Download PDF

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Publication number
CN1416425A
CN1416425A CN01806160A CN01806160A CN1416425A CN 1416425 A CN1416425 A CN 1416425A CN 01806160 A CN01806160 A CN 01806160A CN 01806160 A CN01806160 A CN 01806160A CN 1416425 A CN1416425 A CN 1416425A
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alkyl
solvate
formula
group
salt
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CN01806160A
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Chinese (zh)
Inventor
I·斯塔克
M·达尔斯特伦
D·布洛姆贝里
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AstraZeneca AB
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AstraZeneca AB
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6536—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and sulfur atoms with or without oxygen atoms, as the only ring hetero atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Hematology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
CN01806160A 2000-03-08 2001-03-05 1,5－苯并硫氮杂䓬及其它们作为促血清脂质降低剂的用途 Pending CN1416425A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE00007724 2000-03-08
SE0000772A SE0000772D0 (sv) 2000-03-08 2000-03-08 Chemical compounds

Publications (1)

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CN1416425A true CN1416425A (zh) 2003-05-07

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CN01806160A Pending CN1416425A (zh) 2000-03-08 2001-03-05 1,5－苯并硫氮杂䓬及其它们作为促血清脂质降低剂的用途

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US (1) US6906058B2 (enExample)
EP (1) EP1263747B1 (enExample)
JP (1) JP5204361B2 (enExample)
KR (1) KR20020079990A (enExample)
CN (1) CN1416425A (enExample)
AT (1) ATE283266T1 (enExample)
AU (2) AU2001237556B2 (enExample)
BR (1) BR0109011A (enExample)
CA (1) CA2401055A1 (enExample)
DE (1) DE60107395T2 (enExample)
IL (1) IL151296A0 (enExample)
MX (1) MXPA02008600A (enExample)
NO (1) NO20024217L (enExample)
NZ (1) NZ520951A (enExample)
SE (1) SE0000772D0 (enExample)
WO (1) WO2001066533A1 (enExample)
ZA (1) ZA200206739B (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN106573902A (zh) * 2014-10-20 2017-04-19 Cj医药健康株式会社 新型氨基烷基苯并硫氮杂*衍生物及其用途
CN116157389A (zh) * 2020-08-03 2023-05-23 阿尔比里奥公司 苯并硫杂(二)氮杂环庚三烯化合物及其作为胆汁酸调节剂的用途

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Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN106573902A (zh) * 2014-10-20 2017-04-19 Cj医药健康株式会社 新型氨基烷基苯并硫氮杂*衍生物及其用途
CN106573902B (zh) * 2014-10-20 2019-10-08 Cj医药健康株式会社 氨基烷基苯并硫氮杂*衍生物及其用途
CN116157389A (zh) * 2020-08-03 2023-05-23 阿尔比里奥公司 苯并硫杂(二)氮杂环庚三烯化合物及其作为胆汁酸调节剂的用途

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DE60107395T2 (de) 2005-12-01
NO20024217D0 (no) 2002-09-04
BR0109011A (pt) 2003-06-03
WO2001066533A1 (en) 2001-09-13
AU3755601A (en) 2001-09-17
EP1263747B1 (en) 2004-11-24
NO20024217L (no) 2002-10-09
JP5204361B2 (ja) 2013-06-05
IL151296A0 (en) 2003-04-10
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