CN105960400B - 氨磺酰基噻吩酰胺衍生物及其作为药物用于治疗乙型肝炎的用途 - Google Patents
氨磺酰基噻吩酰胺衍生物及其作为药物用于治疗乙型肝炎的用途 Download PDFInfo
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- CN105960400B CN105960400B CN201480028318.9A CN201480028318A CN105960400B CN 105960400 B CN105960400 B CN 105960400B CN 201480028318 A CN201480028318 A CN 201480028318A CN 105960400 B CN105960400 B CN 105960400B
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
- A61P31/22—Antivirals for DNA viruses for herpes viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Molecular Biology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP13168295.7 | 2013-05-17 | ||
| EP13168295 | 2013-05-17 | ||
| EP13185227 | 2013-09-19 | ||
| EP13185227.9 | 2013-09-19 | ||
| EP14157917 | 2014-03-05 | ||
| EP14157917.7 | 2014-03-05 | ||
| PCT/EP2014/060132 WO2014184365A1 (en) | 2013-05-17 | 2014-05-16 | Sulphamoylthiophenamide derivatives and the use thereof as medicaments for the treatment of hepatitis b |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN105960400A CN105960400A (zh) | 2016-09-21 |
| CN105960400B true CN105960400B (zh) | 2019-05-31 |
Family
ID=50729521
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN201480028318.9A Expired - Fee Related CN105960400B (zh) | 2013-05-17 | 2014-05-16 | 氨磺酰基噻吩酰胺衍生物及其作为药物用于治疗乙型肝炎的用途 |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US10160743B2 (enExample) |
| EP (1) | EP2997019B1 (enExample) |
| JP (1) | JP6441315B2 (enExample) |
| CN (1) | CN105960400B (enExample) |
| AU (1) | AU2014267235B2 (enExample) |
| BR (1) | BR112015028538A2 (enExample) |
| CA (1) | CA2909742C (enExample) |
| CY (1) | CY1122337T1 (enExample) |
| DK (1) | DK2997019T3 (enExample) |
| EA (1) | EA035500B1 (enExample) |
| ES (1) | ES2695182T3 (enExample) |
| HR (1) | HRP20181863T1 (enExample) |
| HU (1) | HUE040446T2 (enExample) |
| IL (1) | IL242141B (enExample) |
| LT (1) | LT2997019T (enExample) |
| MX (1) | MX366787B (enExample) |
| PL (1) | PL2997019T3 (enExample) |
| PT (1) | PT2997019T (enExample) |
| RS (1) | RS57999B1 (enExample) |
| SI (1) | SI2997019T1 (enExample) |
| SM (1) | SMT201800577T1 (enExample) |
| WO (1) | WO2014184365A1 (enExample) |
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| PT2961732T (pt) | 2013-02-28 | 2017-06-26 | Janssen Sciences Ireland Uc | Sulfamoil-arilamidas e utilização das mesmas como medicamentos para o tratamento de hepatite b |
| WO2014161888A1 (en) | 2013-04-03 | 2014-10-09 | Janssen R&D Ireland | N-phenyl-carboxamide derivatives and the use thereof as medicaments for the treatment of hepatitis b |
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| PT2997019T (pt) | 2013-05-17 | 2018-11-21 | Janssen Sciences Ireland Uc | Derivados de sulfamoíltiofenamida e o seu uso como medicamentos para o tratamento da hepatite b |
| UA118680C2 (uk) | 2013-07-25 | 2019-02-25 | ЯНССЕН САЙЄНСЕЗ АЙРЛЕНД ЮСі | Похідні заміщеного гліоксамідом піроламіду та їхнє застосування як лікарських препаратів для лікування гепатиту в |
| EP3060547B1 (en) | 2013-10-23 | 2017-10-11 | Janssen Sciences Ireland UC | Carboxamide derivatives and the use thereof as medicaments for the treatment of hepatitis b |
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| RU2702109C1 (ru) | 2014-02-05 | 2019-10-04 | Новира Терапьютикс, Инк. | Комбинированная терапия для лечения инфекций вгв |
| EA035848B1 (ru) | 2014-02-06 | 2020-08-20 | Янссен Сайенсиз Айрлэнд Юси | Производные сульфамоилпирроламида и их применение в качестве медикаментов для лечения гепатита b |
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- 2014-05-16 WO PCT/EP2014/060132 patent/WO2014184365A1/en not_active Ceased
- 2014-05-16 SI SI201430958T patent/SI2997019T1/sl unknown
- 2014-05-16 US US14/891,895 patent/US10160743B2/en not_active Expired - Fee Related
- 2014-05-16 HU HUE14724109A patent/HUE040446T2/hu unknown
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Also Published As
| Publication number | Publication date |
|---|---|
| JP6441315B2 (ja) | 2018-12-19 |
| CN105960400A (zh) | 2016-09-21 |
| WO2014184365A1 (en) | 2014-11-20 |
| AU2014267235B2 (en) | 2017-10-05 |
| BR112015028538A2 (pt) | 2017-07-25 |
| PT2997019T (pt) | 2018-11-21 |
| EA035500B1 (ru) | 2020-06-25 |
| AU2014267235A8 (en) | 2015-12-10 |
| MX366787B (es) | 2019-07-23 |
| HUE040446T2 (hu) | 2019-03-28 |
| IL242141B (en) | 2019-09-26 |
| EA201592198A1 (ru) | 2016-03-31 |
| HRP20181863T1 (hr) | 2018-12-28 |
| CA2909742C (en) | 2020-08-04 |
| HK1225387A1 (zh) | 2017-09-08 |
| US10160743B2 (en) | 2018-12-25 |
| US20160115149A1 (en) | 2016-04-28 |
| PL2997019T3 (pl) | 2019-03-29 |
| LT2997019T (lt) | 2018-11-26 |
| AU2014267235A1 (en) | 2015-11-12 |
| CA2909742A1 (en) | 2014-11-20 |
| CY1122337T1 (el) | 2020-07-31 |
| SMT201800577T1 (it) | 2019-01-11 |
| SI2997019T1 (sl) | 2018-12-31 |
| EP2997019A1 (en) | 2016-03-23 |
| MX2015015771A (es) | 2016-03-15 |
| RS57999B1 (sr) | 2019-01-31 |
| JP2016518437A (ja) | 2016-06-23 |
| DK2997019T3 (en) | 2018-12-03 |
| ES2695182T3 (es) | 2019-01-02 |
| EP2997019B1 (en) | 2018-08-08 |
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