CN101925586B - 杂环化合物 - Google Patents

杂环化合物 Download PDF

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Publication number
CN101925586B
CN101925586B CN200980103148.5A CN200980103148A CN101925586B CN 101925586 B CN101925586 B CN 101925586B CN 200980103148 A CN200980103148 A CN 200980103148A CN 101925586 B CN101925586 B CN 101925586B
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compound
pharmaceutically acceptable
formula
independently selected
mmol
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Expired - Fee Related
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CN101925586A (zh
Inventor
拉杰什·贾殷
桑贾伊·特雷汉
加戈塔兰·达斯
尼山·辛格
格米特·考尔·南达
西塔拉姆·库马尔·马格蒂
苏迪尔·库马尔·夏尔玛
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Panacea Biotec Pharma Ltd
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Panacea Biotec Ltd
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    • C07—ORGANIC CHEMISTRY
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    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
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    • C07D487/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Reproductive Health (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Molecular Biology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Transplantation (AREA)
  • AIDS & HIV (AREA)
CN200980103148.5A 2008-01-24 2009-01-23 杂环化合物 Expired - Fee Related CN101925586B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN202DE2008 2008-01-24
IN202/DEL/2008 2008-01-24
IN688/DEL/2008 2008-03-18
IN688DE2008 2008-03-18
PCT/IN2009/000061 WO2009093269A1 (en) 2008-01-24 2009-01-23 Novel heterocyclic compounds

Publications (2)

Publication Number Publication Date
CN101925586A CN101925586A (zh) 2010-12-22
CN101925586B true CN101925586B (zh) 2014-05-07

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CN200980103148.5A Expired - Fee Related CN101925586B (zh) 2008-01-24 2009-01-23 杂环化合物

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US (1) US8455479B2 (enExample)
EP (1) EP2250157B1 (enExample)
JP (1) JP5640208B2 (enExample)
KR (1) KR20100113122A (enExample)
CN (1) CN101925586B (enExample)
AP (1) AP2010005364A0 (enExample)
AR (1) AR070520A1 (enExample)
AU (1) AU2009207297B2 (enExample)
BR (1) BRPI0906705A2 (enExample)
CA (1) CA2712685A1 (enExample)
CL (1) CL2009000135A1 (enExample)
EA (1) EA018612B1 (enExample)
PE (1) PE20091353A1 (enExample)
WO (1) WO2009093269A1 (enExample)

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US8492376B2 (en) * 2010-04-21 2013-07-23 Hoffmann-La Roche Inc. Heteroaryl-cyclohexyl-tetraazabenzo[e]azulenes
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
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CN102617566B (zh) * 2011-01-30 2015-03-04 山东轩竹医药科技有限公司 吡啶并咪唑烷衍生物
CN104230935A (zh) * 2011-04-26 2014-12-24 辽宁利锋科技开发有限公司 含有脂环结构化合物的抗肿瘤作用与应用
CN102241678B (zh) * 2011-04-26 2014-10-29 辽宁利锋科技开发有限公司 含有脂环结构化合物的抗肿瘤作用与应用
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
CN105142621A (zh) 2012-10-24 2015-12-09 国家健康科学研究所 用于预防或治疗糖尿病和促进β-细胞存活的TPL2激酶抑制剂
KR20160028241A (ko) 2014-09-03 2016-03-11 김형도 목욕탕용 순환배관 슬러지 제거방법
EP3273981B1 (en) 2015-03-24 2020-04-29 INSERM - Institut National de la Santé et de la Recherche Médicale Method and pharmaceutical composition for use in the treatment of diabetes
CA3014644A1 (en) 2016-02-15 2017-08-24 The Regents Of The University Of Michigan Fused 1,4-oxazepines and related analogs as bet bromodomain inhibitors
CN106883152A (zh) * 2017-04-07 2017-06-23 上海应用技术大学 一种β‑氨基酮的制备方法
JP7825618B2 (ja) 2020-11-06 2026-03-06 サイトキネティックス， インコーポレイテッド 二環式１，４－ジアゼパノン及びその治療的使用

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US20100311732A1 (en) 2010-12-09
CN101925586A (zh) 2010-12-22
JP5640208B2 (ja) 2014-12-17
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EP2250157A1 (en) 2010-11-17
AR070520A1 (es) 2010-04-14
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WO2009093269A1 (en) 2009-07-30
AU2009207297A1 (en) 2009-07-30
AP2010005364A0 (en) 2010-08-31
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CL2009000135A1 (es) 2009-10-09
WO2009093269A9 (en) 2009-10-15
US8455479B2 (en) 2013-06-04
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AU2009207297B2 (en) 2011-11-10
BRPI0906705A2 (pt) 2015-06-30

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