BRPI9612950B1 - - Google Patents

Info

Publication number
BRPI9612950B1
BRPI9612950B1 BRPI9612950A BRPI9612950B1 BR PI9612950 B1 BRPI9612950 B1 BR PI9612950B1 BR PI9612950 A BRPI9612950 A BR PI9612950A BR PI9612950 B1 BRPI9612950 B1 BR PI9612950B1
Authority
BR
Brazil
Prior art keywords
powder
particles
active
inhaler
carrier particles
Prior art date
Application number
Other languages
English (en)
Portuguese (pt)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10768844&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI9612950(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of BRPI9612950B1 publication Critical patent/BRPI9612950B1/pt
Publication of BRPI9612950B8 publication Critical patent/BRPI9612950B8/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7012Compounds having a free or esterified carboxyl group attached, directly or through a carbon chain, to a carbon atom of the saccharide radical, e.g. glucuronic acid, neuraminic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/12Aerosols; Foams
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Dispersion Chemistry (AREA)
  • Pulmonology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Otolaryngology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Manufacturing Of Micro-Capsules (AREA)
BRPI9612950A 1995-01-31 1996-01-31 pó para uso em inaladores de pó seco. BRPI9612950B8 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GBGB9501841.2A GB9501841D0 (en) 1995-01-31 1995-01-31 Improvements in and relating to carrier particles for use in dry powder inhalers
GBGB9521937.4A GB9521937D0 (en) 1995-01-31 1995-10-26 Improvementsin and relating to carrier particles for use in dry powder inhailers
PCT/GB1996/000215 WO1996023485A1 (en) 1995-01-31 1996-01-31 Carrier particles for use in dry powder inhalers
BRPI9607490A BR9607490B8 (pt) 1995-01-31 1996-01-31 pó para uso em inaladores de pó seco e partículas para o uso no mesmo.

Publications (2)

Publication Number Publication Date
BRPI9612950B1 true BRPI9612950B1 (enExample) 2011-08-23
BRPI9612950B8 BRPI9612950B8 (pt) 2018-04-17

Family

ID=10768844

Family Applications (3)

Application Number Title Priority Date Filing Date
BRPI9612950-6A BR9612950B1 (pt) 1995-01-31 1996-01-31 pó para uso em inaladores de pó seco.
BRPI9607490A BR9607490B8 (pt) 1995-01-31 1996-01-31 pó para uso em inaladores de pó seco e partículas para o uso no mesmo.
BRPI9612950A BRPI9612950B8 (pt) 1995-01-31 1996-01-31 pó para uso em inaladores de pó seco.

Family Applications Before (2)

Application Number Title Priority Date Filing Date
BRPI9612950-6A BR9612950B1 (pt) 1995-01-31 1996-01-31 pó para uso em inaladores de pó seco.
BRPI9607490A BR9607490B8 (pt) 1995-01-31 1996-01-31 pó para uso em inaladores de pó seco e partículas para o uso no mesmo.

Country Status (32)

Country Link
US (5) US6153224A (enExample)
EP (6) EP0806938B1 (enExample)
JP (1) JP4042867B2 (enExample)
KR (1) KR100500694B1 (enExample)
CN (1) CN1303974C (enExample)
AT (3) ATE256450T1 (enExample)
AU (1) AU699131B2 (enExample)
BG (1) BG101858A (enExample)
BR (3) BR9612950B1 (enExample)
CA (1) CA2211874C (enExample)
CZ (1) CZ294259B6 (enExample)
DE (2) DE69636961T2 (enExample)
DK (3) DK0806938T3 (enExample)
EA (1) EA000352B1 (enExample)
EE (1) EE9700176A (enExample)
ES (3) ES2375007T3 (enExample)
FI (1) FI119676B (enExample)
GB (2) GB9501841D0 (enExample)
GE (1) GEP19991687B (enExample)
HU (1) HU229965B1 (enExample)
IS (1) IS4531A (enExample)
MX (1) MX9705847A (enExample)
NO (1) NO324037B1 (enExample)
NZ (1) NZ300654A (enExample)
PL (1) PL186757B1 (enExample)
PT (3) PT1232745E (enExample)
SI (2) SI1232745T1 (enExample)
SK (1) SK282630B6 (enExample)
TR (1) TR199700722T1 (enExample)
UA (1) UA61051C2 (enExample)
WO (1) WO1996023485A1 (enExample)
ZA (1) ZA96721B (enExample)

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* Cited by examiner, † Cited by third party
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