BR112017000565A2 - processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina - Google Patents

processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina

Info

Publication number
BR112017000565A2
BR112017000565A2 BR112017000565A BR112017000565A BR112017000565A2 BR 112017000565 A2 BR112017000565 A2 BR 112017000565A2 BR 112017000565 A BR112017000565 A BR 112017000565A BR 112017000565 A BR112017000565 A BR 112017000565A BR 112017000565 A2 BR112017000565 A2 BR 112017000565A2
Authority
BR
Brazil
Prior art keywords
pyrazol
pyridine
chloro
preparation
amino
Prior art date
Application number
BR112017000565A
Other languages
English (en)
Inventor
Lorsbach Beth
E Podhorez David
Roth Gary
Yang Qiang
Li Xiaoyong
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of BR112017000565A2 publication Critical patent/BR112017000565A2/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

a presente invenção refere-se a 3-(3-cloro-1h-pirazol-1-il)piridina, que é preparada por ciclização de dicloridrato de 3-hidrazinopiridina com acrilonitrila para fornecer 1-(piridin-3-il)-4,5-di-hidro-1h-pirazol-3-amina, por oxidação para fornecer 3-(3-amino-1h-pirazol-1-il)piridina, e por conversão do grupo amino em um grupo cloro por uma reação de sandmeyer.
BR112017000565A 2014-07-31 2014-10-17 processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina BR112017000565A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462031547P 2014-07-31 2014-07-31
PCT/US2014/061029 WO2016018444A1 (en) 2014-07-31 2014-10-17 Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine

Publications (1)

Publication Number Publication Date
BR112017000565A2 true BR112017000565A2 (pt) 2017-11-07

Family

ID=54609130

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112017000565A BR112017000565A2 (pt) 2014-07-31 2014-10-17 processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina

Country Status (11)

Country Link
US (3) US9249122B1 (pt)
EP (1) EP3186230A4 (pt)
JP (1) JP2017522306A (pt)
KR (1) KR20170039121A (pt)
CN (1) CN106470976A (pt)
AR (1) AR098108A1 (pt)
BR (1) BR112017000565A2 (pt)
CA (1) CA2954631A1 (pt)
IL (1) IL249988A0 (pt)
TW (1) TW201609696A (pt)
WO (1) WO2016018444A1 (pt)

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MX2016004940A (es) 2013-10-17 2016-06-28 Dow Agrosciences Llc Proceso para la preparacion de compuestos plaguicidas.
EP3057425A4 (en) 2013-10-17 2017-08-02 Dow AgroSciences LLC Processes for the preparation of pesticidal compounds
US9102654B2 (en) 2013-10-17 2015-08-11 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
WO2015058023A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
CA2925873A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
CN105636442B (zh) 2013-10-17 2018-04-27 美国陶氏益农公司 制备杀虫化合物的方法
JP2016536296A (ja) 2013-10-17 2016-11-24 ダウ アグロサイエンシィズ エルエルシー 有害生物防除性化合物の製造方法
KR20170039121A (ko) * 2014-07-31 2017-04-10 다우 아그로사이언시즈 엘엘씨 3-(3-클로로-1h-피라졸-1-일)피리딘의 제조 방법
WO2016018443A1 (en) 2014-07-31 2016-02-04 Dow Agrosciences Llc Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine
US9029555B1 (en) 2014-07-31 2015-05-12 Dow Agrosciences Llc Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine
BR112017002735A2 (pt) 2014-08-19 2017-12-19 Dow Agrosciences Llc processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina
US9085552B1 (en) 2014-09-12 2015-07-21 Dow Agrosciences Llc Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine
CN109790150A (zh) 2016-08-11 2019-05-21 拜耳作物科学股份公司 取代的吡唑啉基衍生物、其制备方法及其作为除草剂和/或植物生长调节剂的用途
EP3562807B1 (en) 2016-12-29 2022-08-03 Corteva Agriscience LLC Processes for the preparation of pesticidal compounds
US10233155B2 (en) 2016-12-29 2019-03-19 Dow Agrosciences Llc Processes for the preparation of pesticide compounds
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