BR0311494A - Novos indóis substituìdos - Google Patents

Novos indóis substituìdos

Info

Publication number
BR0311494A
BR0311494A BR0311494-5A BR0311494A BR0311494A BR 0311494 A BR0311494 A BR 0311494A BR 0311494 A BR0311494 A BR 0311494A BR 0311494 A BR0311494 A BR 0311494A
Authority
BR
Brazil
Prior art keywords
replaced
new
new indoles
indoles replaced
indos
Prior art date
Application number
BR0311494-5A
Other languages
English (en)
Inventor
Stephen Brough
Tony Cook
Mark Dickinson
Rukhsana Rasul
Hitesh Sanganee
Simon Teague
Roger Bonnert
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BR0311494A publication Critical patent/BR0311494A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

"NOVOS INDóIS SUBSTITUìDOS". A presente invenção refere-se a indóis substituídos de fórmula (I) úteis como compostos farmacêuticos para o tratamento de distúrbios respiratórios.
BR0311494-5A 2002-05-30 2003-05-27 Novos indóis substituìdos BR0311494A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0201635A SE0201635D0 (sv) 2002-05-30 2002-05-30 Novel compounds
PCT/SE2003/000856 WO2003101961A1 (en) 2002-05-30 2003-05-27 Novel substituted indoles

Publications (1)

Publication Number Publication Date
BR0311494A true BR0311494A (pt) 2005-03-29

Family

ID=20288018

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0311494-5A BR0311494A (pt) 2002-05-30 2003-05-27 Novos indóis substituìdos

Country Status (25)

Country Link
US (1) US7166607B2 (pt)
EP (1) EP1513812B1 (pt)
JP (1) JP4485354B2 (pt)
KR (1) KR20050010507A (pt)
CN (1) CN100404505C (pt)
AR (1) AR039934A1 (pt)
AT (1) ATE501118T1 (pt)
AU (1) AU2003228201A1 (pt)
BR (1) BR0311494A (pt)
CA (1) CA2487675A1 (pt)
CO (1) CO5631431A2 (pt)
DE (1) DE60336314D1 (pt)
ES (1) ES2360936T3 (pt)
IS (1) IS7607A (pt)
MX (1) MXPA04011876A (pt)
MY (1) MY133624A (pt)
NO (1) NO20045589L (pt)
NZ (1) NZ536883A (pt)
PL (1) PL375111A1 (pt)
RU (1) RU2288914C2 (pt)
SE (1) SE0201635D0 (pt)
TW (1) TW200407305A (pt)
UA (1) UA79464C2 (pt)
WO (1) WO2003101961A1 (pt)
ZA (1) ZA200409641B (pt)

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JP4484108B2 (ja) 2002-05-16 2010-06-16 塩野義製薬株式会社 Ｐｇｄ２受容体拮抗作用を有する化合物
TW200307542A (en) 2002-05-30 2003-12-16 Astrazeneca Ab Novel compounds
SE0201635D0 (sv) 2002-05-30 2002-05-30 Astrazeneca Ab Novel compounds
SE0202241D0 (sv) 2002-07-17 2002-07-17 Astrazeneca Ab Novel Compounds
SE0301569D0 (sv) 2003-05-27 2003-05-27 Astrazeneca Ab Novel compounds
SE0302232D0 (sv) 2003-08-18 2003-08-18 Astrazeneca Ab Novel Compounds
SE0303180D0 (sv) 2003-11-26 2003-11-26 Astrazeneca Ab Novel compounds

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AU2003228201A1 (en) 2003-12-19
IS7607A (is) 2004-12-21
WO2003101961A1 (en) 2003-12-11
MY133624A (en) 2007-11-30
US7166607B2 (en) 2007-01-23
ATE501118T1 (de) 2011-03-15
JP4485354B2 (ja) 2010-06-23
EP1513812A1 (en) 2005-03-16
CO5631431A2 (es) 2006-04-28
EP1513812B1 (en) 2011-03-09
TW200407305A (en) 2004-05-16
CN100404505C (zh) 2008-07-23
ZA200409641B (en) 2006-02-22
RU2004135064A (ru) 2005-08-10
DE60336314D1 (de) 2011-04-21
RU2288914C2 (ru) 2006-12-10
KR20050010507A (ko) 2005-01-27
NZ536883A (en) 2006-08-31
AR039934A1 (es) 2005-03-09
CN1671659A (zh) 2005-09-21
NO20045589L (no) 2005-02-02
PL375111A1 (en) 2005-11-28
MXPA04011876A (es) 2005-03-31
SE0201635D0 (sv) 2002-05-30
UA79464C2 (en) 2007-06-25
JP2005538955A (ja) 2005-12-22

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