SE0301569D0 - Novel compounds - Google Patents

Novel compounds

Info

Publication number
SE0301569D0
SE0301569D0 SE0301569A SE0301569A SE0301569D0 SE 0301569 D0 SE0301569 D0 SE 0301569D0 SE 0301569 A SE0301569 A SE 0301569A SE 0301569 A SE0301569 A SE 0301569A SE 0301569 D0 SE0301569 D0 SE 0301569D0
Authority
SE
Sweden
Prior art keywords
novel compounds
novel
compounds
Prior art date
Application number
SE0301569A
Other languages
English (en)
Inventor
Roger Bonnert
Rukhsana Rasul
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Priority to SE0301569A priority Critical patent/SE0301569D0/sv
Publication of SE0301569D0 publication Critical patent/SE0301569D0/sv
Priority to SE0302305A priority patent/SE0302305D0/sv
Priority to TW099109193A priority patent/TW201024261A/zh
Priority to TW093114113A priority patent/TWI328004B/zh
Priority to ARP040101792A priority patent/AR044552A1/es
Priority to DK04734774T priority patent/DK1656346T3/da
Priority to AT08165755T priority patent/ATE502010T1/de
Priority to EP04734774A priority patent/EP1656346B1/en
Priority to JP2006532212A priority patent/JP4541361B2/ja
Priority to DE602004020072T priority patent/DE602004020072D1/de
Priority to KR1020117009790A priority patent/KR20110050754A/ko
Priority to SI200431874T priority patent/SI2281815T1/sl
Priority to DE602004031894T priority patent/DE602004031894D1/de
Priority to CN2004800146027A priority patent/CN1795174B/zh
Priority to SI200431120T priority patent/SI1656346T1/sl
Priority to AT10180348T priority patent/ATE552243T1/de
Priority to EP10180348A priority patent/EP2281815B1/en
Priority to AT04734774T priority patent/ATE425965T1/de
Priority to PT08165755T priority patent/PT2025670E/pt
Priority to DK08165755.3T priority patent/DK2025670T3/da
Priority to BRPI0410711A priority patent/BRPI0410711B8/pt
Priority to AU2004242624A priority patent/AU2004242624B2/en
Priority to ES10180348T priority patent/ES2382606T3/es
Priority to PL08165755T priority patent/PL2025670T3/pl
Priority to EP08165755A priority patent/EP2025670B1/en
Priority to PCT/SE2004/000808 priority patent/WO2004106302A1/en
Priority to KR1020057022513A priority patent/KR101067586B1/ko
Priority to SI200431669T priority patent/SI2025670T1/sl
Priority to CN2011102633202A priority patent/CN102391171A/zh
Priority to PT04734774T priority patent/PT1656346E/pt
Priority to ES04734774T priority patent/ES2322650T3/es
Priority to US10/558,228 priority patent/US7687535B2/en
Priority to RU2005137403/04A priority patent/RU2361860C2/ru
Priority to PT10180348T priority patent/PT2281815E/pt
Priority to MYPI20041992A priority patent/MY144483A/en
Priority to PL10180348T priority patent/PL2281815T3/pl
Priority to ES08165755T priority patent/ES2361485T3/es
Priority to DK10180348.4T priority patent/DK2281815T3/da
Priority to MXPA05012680A priority patent/MXPA05012680A/es
Priority to UAA200511010A priority patent/UA84701C2/ru
Priority to CA2526866A priority patent/CA2526866C/en
Priority to PL04734774T priority patent/PL1656346T3/pl
Priority to NZ543722A priority patent/NZ543722A/xx
Priority to KR1020117009788A priority patent/KR101067535B1/ko
Priority to IL171928A priority patent/IL171928A/en
Priority to CO05118882A priority patent/CO5630030A2/es
Priority to ZA200509598A priority patent/ZA200509598B/en
Priority to IS8189A priority patent/IS2722B/is
Priority to NO20056130A priority patent/NO20056130L/no
Priority to HK06111158.9A priority patent/HK1090635A1/xx
Priority to IL194872A priority patent/IL194872A0/en
Priority to US12/397,618 priority patent/US20090163518A1/en
Priority to HR20090281T priority patent/HRP20090281T1/xx
Priority to CY20091100564T priority patent/CY1109104T1/el
Priority to HK11107570.0A priority patent/HK1149563A1/xx
Priority to HK09105852.7A priority patent/HK1126773A1/xx
Priority to JP2010082748A priority patent/JP2010155862A/ja
Priority to IS8920A priority patent/IS8920A/is
Priority to US13/047,280 priority patent/US20110263614A1/en
Priority to IL212265A priority patent/IL212265A0/en
Priority to IL212371A priority patent/IL212371A0/en
Priority to HR20110359T priority patent/HRP20110359T1/hr
Priority to CY20111100464T priority patent/CY1111469T1/el
Priority to US13/344,051 priority patent/US20120178764A1/en
Priority to HRP20120390TT priority patent/HRP20120390T1/hr
Priority to CY20121100486T priority patent/CY1112853T1/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/16Central respiratory analeptics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
SE0301569A 2003-05-27 2003-05-27 Novel compounds SE0301569D0 (sv)

Priority Applications (66)

Application Number Priority Date Filing Date Title
SE0301569A SE0301569D0 (sv) 2003-05-27 2003-05-27 Novel compounds
SE0302305A SE0302305D0 (sv) 2003-05-27 2003-08-27 Novel Compounds
TW099109193A TW201024261A (en) 2003-05-27 2004-05-19 Substituted indoles and preparation and use thereof
TW093114113A TWI328004B (en) 2003-05-27 2004-05-19 Substituted indoles and use thereof
ARP040101792A AR044552A1 (es) 2003-05-27 2004-05-24 Derivados del indol,composiciones farmaceuticas que los contienen y procesos para su preparacion, de utilidad para el tratamiento de trastornos respiratorios
DK04734774T DK1656346T3 (da) 2003-05-27 2004-05-25 1,2,3,4-tetrasubstituerede indol til behandling af luftvejssygdomme
AT08165755T ATE502010T1 (de) 2003-05-27 2004-05-25 Verwendung von 3-phenylthio-1h-indol-1-essigsäure-derivate als modulatoren der crth2-rezeptor- aktivität
EP04734774A EP1656346B1 (en) 2003-05-27 2004-05-25 1,2,3,4-tetrasubstituted indole for the treatment of respiratory diseases
JP2006532212A JP4541361B2 (ja) 2003-05-27 2004-05-25 新規3位硫黄置換インドール
DE602004020072T DE602004020072D1 (de) 2003-05-27 2004-05-25 1,2,3,4-tetrasubstituiertes indol zur behandlung von atemwegserkrankungen
KR1020117009790A KR20110050754A (ko) 2003-05-27 2004-05-25 신규한 치환된 3-황 인돌
SI200431874T SI2281815T1 (sl) 2003-05-27 2004-05-25 Vmesna spojina etil estra 4-(acetilamino)-3-((4-klorofenil)tio)-2-metil-1H-indol-1-ocetne kisline
DE602004031894T DE602004031894D1 (de) 2003-05-27 2004-05-25 Verwendung von 3-Phenylthio-1H-indol-1-essigsäure-Derivate als Modulatoren der CRTh2-Rezeptor-Aktivität
CN2004800146027A CN1795174B (zh) 2003-05-27 2004-05-25 取代的3-硫吲哚
SI200431120T SI1656346T1 (sl) 2003-05-27 2004-05-25 1,2,3,4-tetrasubstituiran indol za zdravljenje respiratornih bolezni
AT10180348T ATE552243T1 (de) 2003-05-27 2004-05-25 4-(acetylamino)-3-ä(4-chlorophenyl)thioü-2-meth l-1h-indole-1-essigsäure-ethyl-ester zwischenverbindung
EP10180348A EP2281815B1 (en) 2003-05-27 2004-05-25 4-(Acetylamino)-3-[(4-chlorophenyl)thio]-2-methyl-1H-indole-1-acetic acid ethyl ester intermediate compound
AT04734774T ATE425965T1 (de) 2003-05-27 2004-05-25 1,2,3,4-tetrasubstituiertes indol zur behandlung von atemwegserkrankungen
PT08165755T PT2025670E (pt) 2003-05-27 2004-05-25 Utiliza??o de derivados do ?cido 3-feniltio-1h-indole-1-ac?tico como moduladores da actividade dos receptores crth2
DK08165755.3T DK2025670T3 (da) 2003-05-27 2004-05-25 Anvendelse af 3-phenylthio-1H-indol-1-eddikesyre-derivater som modulatorer af CRTh2-receptor aktivitet
BRPI0410711A BRPI0410711B8 (pt) 2003-05-27 2004-05-25 ácido 4-(acetilamina)-3-[(4-clorofenil)tio]-2-metil-1h-indol-1-acético
AU2004242624A AU2004242624B2 (en) 2003-05-27 2004-05-25 Novel substituted 3-sulfur indoles
ES10180348T ES2382606T3 (es) 2003-05-27 2004-05-25 Compuesto intermedio éster etílico del ácido 4-(acetilamino)-3-[(4-clorofenil)tio]-2-metil-1H-indol-acético
PL08165755T PL2025670T3 (pl) 2003-05-27 2004-05-25 Zastosowanie pochodnych kwasu 3-fenylotio-1H-indolo-1-octowego jako modulatorów aktywności receptora CRTh2
EP08165755A EP2025670B1 (en) 2003-05-27 2004-05-25 Use of 3-phenylthio-1H-indole-1-acetic acid derivatives as modulators of CRTh2 receptor activity
PCT/SE2004/000808 WO2004106302A1 (en) 2003-05-27 2004-05-25 Novel substituted 3-sulfur indoles
KR1020057022513A KR101067586B1 (ko) 2003-05-27 2004-05-25 신규한 치환된 3-황 인돌
SI200431669T SI2025670T1 (sl) 2003-05-27 2004-05-25 Uporaba derivatov 3-feniltio-1H-indol-1-ocetne kisline kot modulatorjev aktivnosti CRTh2 receptorja
CN2011102633202A CN102391171A (zh) 2003-05-27 2004-05-25 新型取代的3-硫吲哚
PT04734774T PT1656346E (pt) 2003-05-27 2004-05-25 Indole 1,2,3,4-tetrassubstituído para o tratamento de doenças respiratórias
ES04734774T ES2322650T3 (es) 2003-05-27 2004-05-25 Indol 1,2,3,4-tetrasustituido para el tratamiento de enfermedades respiratorias.
US10/558,228 US7687535B2 (en) 2003-05-27 2004-05-25 Substituted 3-sulfur indoles
RU2005137403/04A RU2361860C2 (ru) 2003-05-27 2004-05-25 Новые замещенные 3-сера-индолы
PT10180348T PT2281815E (pt) 2003-05-27 2004-05-25 Composto intermediário de éster etílico do ácido 4-(acetilamino)-3-[(4-clorofenil)tio]-2-metil-1h-indole- 1-acético
MYPI20041992A MY144483A (en) 2003-05-27 2004-05-25 1,2,3,4-tetrasubstituted indole for the treatment of respiratory diseases
PL10180348T PL2281815T3 (pl) 2003-05-27 2004-05-25 Związek pośredni, ester etylowy kwasu 4-(acetyloamino)-3-[(4-chlorofenylo}tio]-2-metylo-1H-indolooctowego
ES08165755T ES2361485T3 (es) 2003-05-27 2004-05-25 Uso de derivados de ácido 3-feniltio-1h-indol-acético como moduladores de la actividad del receptor crth2.
DK10180348.4T DK2281815T3 (da) 2003-05-27 2004-05-25 4-(Acetylamino)-3-[(4-chlorophenyl)thio]-2-methyl-1H-indole-1-acetic acid ethyl ester intermediate compound
MXPA05012680A MXPA05012680A (es) 2003-05-27 2004-05-25 Indoles novedosos de 3-azufre sustituidos.
UAA200511010A UA84701C2 (ru) 2003-05-27 2004-05-25 Замещенные индолы, способ их получения, их использования
CA2526866A CA2526866C (en) 2003-05-27 2004-05-25 Substituted 3-sulfur indoles for treating a disease mediated by crth2
PL04734774T PL1656346T3 (pl) 2003-05-27 2004-05-25 1,2,3,4-Tetrapodstawiony indol do leczenia chorób dróg oddechowych
NZ543722A NZ543722A (en) 2003-05-27 2004-05-25 Novel substituted 3-sulfur indoles
KR1020117009788A KR101067535B1 (ko) 2003-05-27 2004-05-25 신규한 치환된 3-황 인돌
IL171928A IL171928A (en) 2003-05-27 2005-11-14 Compounds of 4 - (acetylamino) - 3 - [(4 - chlorophenyl) thio] - 2 - methyl - 1H - indole - 1 - acetic acid, salts and their solvates, and their uses in the preparation of medicine
CO05118882A CO5630030A2 (es) 2003-05-27 2005-11-23 Acido 4-(acetilamino)-3-{(4-clorofenil)tio}-2-metil-1h-indol-1-acetico y composicion farmaceutica que lo contiene
ZA200509598A ZA200509598B (en) 2003-05-27 2005-11-28 Novel substituted 3-sulfur indoles
IS8189A IS2722B (is) 2003-05-27 2005-12-20 1, 2, 3, 4- Tetrasetin indól til meðhöndlunar á öndunarfærasjúkdómum
NO20056130A NO20056130L (no) 2003-05-27 2005-12-22 Nye substituerte 3-svovelindoler
HK06111158.9A HK1090635A1 (en) 2003-05-27 2006-10-11 Substituted 3-sulfur indoles
IL194872A IL194872A0 (en) 2003-05-27 2008-10-23 Novel substituted 3-sulfur indoles
US12/397,618 US20090163518A1 (en) 2003-05-27 2009-03-04 Novel Compounds
HR20090281T HRP20090281T1 (en) 2003-05-27 2009-05-15 1,2,3,4-tetrasubstituted indole for the treatment of respiratory diseases
CY20091100564T CY1109104T1 (el) 2003-05-27 2009-05-28 1,2,3,4 τετρα-υποκατεστημενη ινδολη για την αντιμετωπιση ασθενειων του αναπνευστικου
HK11107570.0A HK1149563A1 (sv) 2003-05-27 2009-06-30
HK09105852.7A HK1126773A1 (sv) 2003-05-27 2009-06-30
JP2010082748A JP2010155862A (ja) 2003-05-27 2010-03-31 新規3位硫黄置換インドール
IS8920A IS8920A (is) 2003-05-27 2010-08-09 3-(Fenýl eða kínólyl)þíó- 1H-idnól-1-ediksýru afleður sem mótarar á virkni CRTh2 vitaka.
US13/047,280 US20110263614A1 (en) 2003-05-27 2011-03-14 Novel compounds
IL212265A IL212265A0 (en) 2003-05-27 2011-04-11 Novel compounds
IL212371A IL212371A0 (en) 2003-05-27 2011-04-14 Novel compounds
HR20110359T HRP20110359T1 (hr) 2003-05-27 2011-05-16 Upotreba derivata 3-feniltio-1h-indol-1-octene kiseline kao modulatora crth2 receptorske aktivnosti
CY20111100464T CY1111469T1 (el) 2003-05-27 2011-05-16 ΧΡΗΣΗ ΠΑΡΑΓΩΓΩΝ 3-ΦΑΙΝΥΛΘΕΙΟ-1Η-ΙΝΔΟΛΗ-1-ΟΞΙΚΟΥ ΟΞΕΟΣ ΩΣ ΡΥΘΜΙΣΤΕΣ ΤΗΣ ΔΡΑΣΗΣ ΤΟΥ ΥΠΟΔΟΧΕΑ CRTh2
US13/344,051 US20120178764A1 (en) 2003-05-27 2012-01-05 Novel Compounds
HRP20120390TT HRP20120390T1 (hr) 2003-05-27 2012-05-10 Intermedijarni spoj etil estera 4-(acetilamino)-3-[(4-klorofenil)tio]-2-metil-1h-indol-1-octene kiseline
CY20121100486T CY1112853T1 (el) 2003-05-27 2012-05-29 Ενδιαμεση ενωση 4-(ακετυλαμινο)-3-[(4-χλωροφαινυλ)θειο]-2-μεθυλ-1η-ινδολη-1-οξικο οξυ αιθυλεστερα

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0301569A SE0301569D0 (sv) 2003-05-27 2003-05-27 Novel compounds
SE0302305A SE0302305D0 (sv) 2003-05-27 2003-08-27 Novel Compounds

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RU2005137403A (ru) 2006-05-27
BRPI0410711B1 (pt) 2018-09-25
PT2281815E (pt) 2012-05-24
KR20110050754A (ko) 2011-05-16
BRPI0410711B8 (pt) 2021-05-25
IL194872A0 (en) 2011-08-01
SI2025670T1 (sl) 2011-06-30
CY1111469T1 (el) 2015-08-05
PL2025670T3 (pl) 2011-07-29
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CO5630030A2 (es) 2006-04-28
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ATE502010T1 (de) 2011-04-15

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