BG63542B1 - Методи и междинни съединения за получаване на заместени хроманолови производни - Google Patents

Методи и междинни съединения за получаване на заместени хроманолови производни Download PDF

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Publication number
BG63542B1
BG63542B1 BG103231A BG10323199A BG63542B1 BG 63542 B1 BG63542 B1 BG 63542B1 BG 103231 A BG103231 A BG 103231A BG 10323199 A BG10323199 A BG 10323199A BG 63542 B1 BG63542 B1 BG 63542B1
Authority
BG
Bulgaria
Prior art keywords
alkyl
compound
formula
phenyl
enantiomer
Prior art date
Application number
BG103231A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG103231A (en
Inventor
Joel HAWKINS
Anthony Piscopio
Stephane Caron
Sarah KELLY
Jefrey RAGGON
Michael CASTALDI
Robert DUGGER
Sally RUGGERI
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of BG103231A publication Critical patent/BG103231A/xx
Publication of BG63542B1 publication Critical patent/BG63542B1/bg

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40Halogenated unsaturated alcohols
    • C07C33/50Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
BG103231A 1996-09-16 1999-03-09 Методи и междинни съединения за получаване на заместени хроманолови производни BG63542B1 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2637296P 1996-09-16 1996-09-16
PCT/IB1997/001024 WO1998011085A1 (en) 1996-09-16 1997-08-25 Processes and intermediates for preparing substituted chromanol derivatives

Publications (2)

Publication Number Publication Date
BG103231A BG103231A (en) 1999-12-30
BG63542B1 true BG63542B1 (bg) 2002-04-30

Family

ID=21831429

Family Applications (1)

Application Number Title Priority Date Filing Date
BG103231A BG63542B1 (bg) 1996-09-16 1999-03-09 Методи и междинни съединения за получаване на заместени хроманолови производни

Country Status (39)

Country Link
US (4) US6096906A (de)
EP (1) EP0925292B1 (de)
JP (1) JP3117730B2 (de)
KR (1) KR100339164B1 (de)
CN (1) CN1108298C (de)
AP (1) AP726A (de)
AT (1) ATE249452T1 (de)
AU (1) AU713701B2 (de)
BG (1) BG63542B1 (de)
BR (1) BR9711482A (de)
CA (1) CA2265043C (de)
CO (1) CO4600635A1 (de)
DE (1) DE69724801T2 (de)
DK (1) DK0925292T3 (de)
DZ (1) DZ2308A1 (de)
EA (1) EA002204B1 (de)
ES (1) ES2206738T3 (de)
GT (3) GT199700104A (de)
HN (1) HN1997000127A (de)
HR (1) HRP970497B1 (de)
ID (1) ID19613A (de)
IL (1) IL128732A0 (de)
IS (1) IS4980A (de)
MA (1) MA24319A1 (de)
NO (1) NO991254L (de)
NZ (1) NZ334214A (de)
OA (1) OA10995A (de)
PA (1) PA8437901A1 (de)
PE (1) PE109798A1 (de)
PL (1) PL332351A1 (de)
PT (1) PT925292E (de)
SK (1) SK31399A3 (de)
TN (1) TNSN97155A1 (de)
TR (1) TR199900592T2 (de)
TW (1) TW449579B (de)
UA (1) UA58520C2 (de)
WO (1) WO1998011085A1 (de)
YU (1) YU13299A (de)
ZA (1) ZA978291B (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6436987B1 (en) * 2000-06-08 2002-08-20 Pfizer Inc. Crystalline forms of (3S-trans)-2-[3,4-dihydro-4-hydroxy-3-(phenylmethyl)-2H-1-benzopyran-7-yl]-4-(trifluoromethyl)-benzoic acid
BR0206771A (pt) * 2001-01-30 2004-02-25 Pfizer Prod Inc Processos para a preparação de cidos cromanilbenzóicos
AU4239302A (en) * 2001-06-28 2003-01-02 Pfizer Products Inc. Benzoic acid substituted benzopyrans for the treatment of atherosclerosis
ES2551916T3 (es) 2007-07-23 2015-11-24 The Board Of Trustees Of The University Of Illinois Sistema para controlar la reactividad de los ácidos borónicos
WO2010036921A2 (en) 2008-09-26 2010-04-01 The Board Of Trustees Of The University Of Illinois Slow release of organoboronic acids in cross-coupling reactions
US8304513B2 (en) * 2009-09-02 2012-11-06 E I Du Pont De Nemours And Company Polyesters comprising fluorovinylether functionalized aromatic moieties
US8378061B2 (en) * 2009-09-02 2013-02-19 E.I. Du Pont De Nemours And Company Polyester films with improved oil repellency
TW201127822A (en) * 2009-09-02 2011-08-16 Du Pont Fluorinated 4-oxo-chroman-carboxylates
CN102612509A (zh) 2009-09-02 2012-07-25 纳幕尔杜邦公司 氟醚官能化的芳族二酯及其衍生物
CA2773142A1 (en) * 2009-09-02 2011-03-10 Neville Everton Drysdale Polyaramid comprising fluorovinylether functionalized aromatic moieties
US20110218319A1 (en) * 2009-09-02 2011-09-08 E. I. Du Pont De Nemours And Company Polyaramid films comprising fluorovinylether functionalized aromatic moieties
US8557980B2 (en) 2010-02-18 2013-10-15 The Board Of Trustees Of The University Of Illinois Methods for forming protected organoboronic acids
US10500178B2 (en) 2015-03-13 2019-12-10 The Board Of Trustees Of The Leland Stanford Junior University LTB4 inhibition to prevent and treat human lymphedema

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9119920D0 (en) * 1991-09-18 1991-10-30 Glaxo Group Ltd Chemical compounds
ES2098547T3 (es) * 1992-01-23 1997-05-01 Pfizer Benzopirano y otros antagonistas de ltb4 relacionados.
MX9300312A (es) * 1992-01-23 1993-07-31 Pfizer Antagonistas benzopiranicos y relacionado de ltb.
JPH07507811A (ja) * 1992-10-21 1995-08-31 ファイザー・インク. 鏡像異性のシス−3−(4,6−ジヒドロキシクロマン−3−イル−メチル)安息香酸
KR950704309A (ko) * 1992-10-21 1995-11-17 알렌 제이. 스피겔 벤젠융합된 하이드록시 치환-사이클로알킬 및 헤테로사이클릭 고리 화합물의 설폰아미드 유도체(sulfonamide derivatives of benzenefused hydroxy substituted cycloalkyl and heterocyclic ring compounds)
MX9702734A (es) * 1994-10-13 1997-06-28 Pfizer Benzopirano y compuestos benzocondensados, su preparacion y su uso como antagonistas de leucotrieno b4 (ltb4).
KR100232341B1 (ko) * 1994-10-13 2000-07-01 디. 제이. 우드 류코트리엔 b4(ltb4) 길항물질로서의 벤조피란 및 벤조-축합된 화합물
US5539128A (en) * 1994-11-30 1996-07-23 Pfizer Inc. Processes and intermediates for preparing cis(+)3-[4,6-dihydroxy chroman-3-ylmethyl]-4-methoxyaniline

Also Published As

Publication number Publication date
GT199700104BA (es) 1999-03-28
UA58520C2 (uk) 2003-08-15
KR20000036136A (ko) 2000-06-26
TR199900592T2 (xx) 1999-06-21
NO991254L (no) 1999-05-14
CO4600635A1 (es) 1998-05-08
AU713701B2 (en) 1999-12-09
CN1230954A (zh) 1999-10-06
HRP970497A2 (en) 1998-08-31
CA2265043C (en) 2003-01-14
IS4980A (is) 1999-02-16
AP9701083A0 (en) 1997-10-31
SK31399A3 (en) 2000-05-16
WO1998011085A1 (en) 1998-03-19
US6288242B1 (en) 2001-09-11
PL332351A1 (en) 1999-09-13
US20020042526A1 (en) 2002-04-11
DE69724801T2 (de) 2004-06-17
CN1108298C (zh) 2003-05-14
ZA978291B (en) 1999-03-15
TNSN97155A1 (fr) 2005-03-15
AU3781497A (en) 1998-04-02
AP726A (en) 1999-01-29
PT925292E (pt) 2004-01-30
DE69724801D1 (de) 2003-10-16
ATE249452T1 (de) 2003-09-15
PE109798A1 (es) 1999-01-13
NO991254D0 (no) 1999-03-15
MA24319A1 (fr) 1998-04-01
JP3117730B2 (ja) 2000-12-18
KR100339164B1 (ko) 2002-06-01
ID19613A (id) 1998-07-23
DK0925292T3 (da) 2004-01-12
US20020099227A1 (en) 2002-07-25
JP2000502726A (ja) 2000-03-07
PA8437901A1 (es) 2000-05-24
US6444826B1 (en) 2002-09-03
YU13299A (sh) 2001-03-07
EP0925292A1 (de) 1999-06-30
GT199700104AA (es) 1999-03-28
NZ334214A (en) 2000-09-29
HRP970497B1 (en) 2002-06-30
DZ2308A1 (fr) 2002-12-28
US6355825B1 (en) 2002-03-12
EP0925292B1 (de) 2003-09-10
HN1997000127A (es) 1997-12-20
BR9711482A (pt) 1999-08-24
US6096906A (en) 2000-08-01
TW449579B (en) 2001-08-11
GT199700104A (es) 1999-03-02
CA2265043A1 (en) 1998-03-19
BG103231A (en) 1999-12-30
ES2206738T3 (es) 2004-05-16
OA10995A (en) 2001-11-06
EA199900204A1 (ru) 1999-08-26
EA002204B1 (ru) 2002-02-28
IL128732A0 (en) 2000-01-31

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