BG107056A - Азетидинови производни, тяхното получаване и фармацевтични състави, които ги съдържат - Google Patents

Азетидинови производни, тяхното получаване и фармацевтични състави, които ги съдържат Download PDF

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Publication number
BG107056A
BG107056A BG107056A BG10705602A BG107056A BG 107056 A BG107056 A BG 107056A BG 107056 A BG107056 A BG 107056A BG 10705602 A BG10705602 A BG 10705602A BG 107056 A BG107056 A BG 107056A
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BG
Bulgaria
Prior art keywords
radical
methyl
formula
chlorophenyl
hydrogen atom
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BG107056A
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Bulgarian (bg)
English (en)
Inventor
Daniel Achard
Herve Bouchard
Jean Bouquerel
Bruno Filoche
Serge Grisoni
Augustin Hittinger
Michael Myers
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Aventis Pharma S.A.
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Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.
Publication of BG107056A publication Critical patent/BG107056A/bg

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Addiction (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Hematology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Child & Adolescent Psychology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Immunology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Nutrition Science (AREA)
  • Otolaryngology (AREA)
BG107056A 2000-03-03 2002-09-03 Азетидинови производни, тяхното получаване и фармацевтични състави, които ги съдържат BG107056A (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0002775A FR2805818B1 (fr) 2000-03-03 2000-03-03 Derives d'azetidine, leur preparation et les compositions pharmaceutiques les contenant
PCT/FR2001/000600 WO2001064632A1 (fr) 2000-03-03 2001-03-01 Derives d'azetidine, leur preparation et les compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
BG107056A true BG107056A (bg) 2003-07-31

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BG107056A BG107056A (bg) 2000-03-03 2002-09-03 Азетидинови производни, тяхното получаване и фармацевтични състави, които ги съдържат

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EP (1) EP1263720B1 (pt)
JP (1) JP2003525268A (pt)
KR (1) KR100786411B1 (pt)
CN (1) CN1185213C (pt)
AR (1) AR027608A1 (pt)
AT (1) ATE432919T1 (pt)
AU (2) AU3752501A (pt)
BG (1) BG107056A (pt)
BR (1) BR0108871A (pt)
CA (1) CA2400116A1 (pt)
CY (1) CY1109343T1 (pt)
CZ (1) CZ20022931A3 (pt)
DE (1) DE60138872D1 (pt)
DK (1) DK1263720T3 (pt)
DZ (1) DZ3313A1 (pt)
EA (1) EA006583B1 (pt)
EE (1) EE05104B1 (pt)
ES (1) ES2328104T3 (pt)
FR (1) FR2805818B1 (pt)
HR (1) HRP20020711A2 (pt)
HU (1) HUP0301404A3 (pt)
IL (2) IL151428A0 (pt)
MA (1) MA26877A1 (pt)
ME (1) MEP24608A (pt)
MX (1) MXPA02008360A (pt)
NO (1) NO324505B1 (pt)
NZ (1) NZ521075A (pt)
OA (1) OA12220A (pt)
PL (1) PL357534A1 (pt)
PT (1) PT1263720E (pt)
RS (1) RS50417B (pt)
SI (1) SI1263720T1 (pt)
SK (1) SK12452002A3 (pt)
TW (1) TWI230153B (pt)
UA (1) UA72593C2 (pt)
WO (1) WO2001064632A1 (pt)
ZA (1) ZA200206905B (pt)

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WO2003007887A2 (en) 2001-07-20 2003-01-30 Merck & Co., Inc. Substituted imidazoles as cannabinoid receptor modulators
FR2833842B1 (fr) * 2001-12-21 2004-02-13 Aventis Pharma Sa Compositions pharmaceutiques a base de derives d'azetidine
EP1496838B1 (en) 2002-03-12 2010-11-03 Merck Sharp & Dohme Corp. Substituted amides
US7105526B2 (en) 2002-06-28 2006-09-12 Banyu Pharmaceuticals Co., Ltd. Benzimidazole derivatives
AU2003250117B2 (en) 2002-07-29 2007-05-10 F. Hoffmann-La Roche Ag Novel benzodioxoles
PL378244A1 (pl) 2003-01-02 2006-03-20 F. Hoffmann-La Roche Ag Pirolilotiazole i ich zastosowanie jako odwrotnych agonistów receptora CB 1
CN101012193A (zh) 2003-01-02 2007-08-08 霍夫曼-拉罗奇有限公司 新cb 1受体反激动剂
US7772188B2 (en) 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
EP1611120A4 (en) * 2003-04-07 2008-04-23 Cortical Pty Ltd NEW M THODES FOR THE TREATMENT OF INFLAMMATORY DISEASES
FR2854633B1 (fr) * 2003-05-07 2005-06-24 Sanofi Synthelabo Derives de piperidinyl-et piperazinyl-alkylcarbamates, leur preparation et leur application en therapeutique
US7485732B2 (en) * 2003-06-11 2009-02-03 Merck & Co., Inc. Substituted 3-alkyl and 3-alkenyl azetidine derivatives
MXPA05013733A (es) 2003-06-20 2006-03-08 Hoffmann La Roche 2-aminobenzotiazoles como agonistas inversos del receptor de cb1.
GB0320983D0 (en) * 2003-09-08 2003-10-08 Biofocus Plc Compound libraries
JP4765627B2 (ja) 2003-09-22 2011-09-07 Ｍｓｄ株式会社 新規ピペリジン誘導体
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