AU2003304237A1 - Gel-stabilized nanoparticulate active agent compositions - Google Patents

Gel-stabilized nanoparticulate active agent compositions

Info

Publication number
AU2003304237A1
AU2003304237A1 AU2003304237A AU2003304237A AU2003304237A1 AU 2003304237 A1 AU2003304237 A1 AU 2003304237A1 AU 2003304237 A AU2003304237 A AU 2003304237A AU 2003304237 A AU2003304237 A AU 2003304237A AU 2003304237 A1 AU2003304237 A1 AU 2003304237A1
Authority
AU
Australia
Prior art keywords
active agent
solid
nanoparticulate active
gel
dosage form
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003304237A
Other languages
English (en)
Other versions
AU2003304237A8 (en
Inventor
David A. Czekai
Simon L. Mcgurk
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Perrigo Pharma International DAC
Original Assignee
Elan Pharma International Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Elan Pharma International Ltd filed Critical Elan Pharma International Ltd
Publication of AU2003304237A8 publication Critical patent/AU2003304237A8/xx
Publication of AU2003304237A1 publication Critical patent/AU2003304237A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Zoology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Yarns And Mechanical Finishing Of Yarns Or Ropes (AREA)
AU2003304237A 2002-09-11 2003-09-11 Gel-stabilized nanoparticulate active agent compositions Abandoned AU2003304237A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40958702P 2002-09-11 2002-09-11
US60/409,587 2002-09-11
PCT/US2003/028380 WO2005000265A2 (en) 2002-09-11 2003-09-11 Gel-stabilized nanoparticulate active agent compositions

Publications (2)

Publication Number Publication Date
AU2003304237A8 AU2003304237A8 (en) 2005-01-13
AU2003304237A1 true AU2003304237A1 (en) 2005-01-13

Family

ID=33551184

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003304237A Abandoned AU2003304237A1 (en) 2002-09-11 2003-09-11 Gel-stabilized nanoparticulate active agent compositions

Country Status (13)

Country Link
US (1) US7713551B2 (cg-RX-API-DMAC7.html)
EP (1) EP1553927B9 (cg-RX-API-DMAC7.html)
JP (1) JP4878839B2 (cg-RX-API-DMAC7.html)
AT (1) ATE487470T1 (cg-RX-API-DMAC7.html)
AU (1) AU2003304237A1 (cg-RX-API-DMAC7.html)
CA (1) CA2498207C (cg-RX-API-DMAC7.html)
CY (1) CY1110949T1 (cg-RX-API-DMAC7.html)
DE (1) DE60334924D1 (cg-RX-API-DMAC7.html)
DK (1) DK1553927T3 (cg-RX-API-DMAC7.html)
ES (1) ES2355723T3 (cg-RX-API-DMAC7.html)
PT (1) PT1553927E (cg-RX-API-DMAC7.html)
SI (1) SI1553927T1 (cg-RX-API-DMAC7.html)
WO (1) WO2005000265A2 (cg-RX-API-DMAC7.html)

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US20050031691A1 (en) 2005-02-10
EP1553927B9 (en) 2011-09-21
AU2003304237A8 (en) 2005-01-13
EP1553927A2 (en) 2005-07-20
CA2498207C (en) 2012-03-13
WO2005000265A3 (en) 2005-05-12
JP4878839B2 (ja) 2012-02-15
ES2355723T3 (es) 2011-03-30
WO2005000265A2 (en) 2005-01-06
DK1553927T3 (da) 2011-01-31
JP2006514688A (ja) 2006-05-11
DE60334924D1 (de) 2010-12-23
CA2498207A1 (en) 2005-01-06
EP1553927B1 (en) 2010-11-10
CY1110949T1 (el) 2015-06-10
SI1553927T1 (sl) 2010-12-31
PT1553927E (pt) 2010-11-22
US7713551B2 (en) 2010-05-11

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