AR006012A1 - Tabletas que contienen antibioticos de beta-lactamas y un metodo para obtenerlas - Google Patents

Tabletas que contienen antibioticos de beta-lactamas y un metodo para obtenerlas

Info

Publication number
AR006012A1
AR006012A1 ARP970100776A ARP970100776A AR006012A1 AR 006012 A1 AR006012 A1 AR 006012A1 AR P970100776 A ARP970100776 A AR P970100776A AR P970100776 A ARP970100776 A AR P970100776A AR 006012 A1 AR006012 A1 AR 006012A1
Authority
AR
Argentina
Prior art keywords
tablets
weight
tablets containing
containing beta
obtaining
Prior art date
Application number
ARP970100776A
Other languages
English (en)
Original Assignee
Astellas Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astellas Pharma Inc filed Critical Astellas Pharma Inc
Publication of AR006012A1 publication Critical patent/AR006012A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A61K31/546Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Organic Chemistry (AREA)
  • Biophysics (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Zoology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Seasonings (AREA)

Abstract

Tabletas conteniendo antibiótico beta-lactam capaz de ser tomadas oralmente en la forma de dispersiones que resultan de la fácil desintegración por símismas al ser vertidas en agua en un vaso así como un método de producción de dichas tabletas.Las tabletas de esta invención comprenden, en base de cadatableta, de 60-85% por peso de un antibiótico de beta-lactan, 1-10%por peso de hidroxipropilcelulosa de sustitución baja y/o polivinilpirrolidona unida através como un desintegrador, y 0,5-2% po r peso de un aglutinante. Los gránulos a seer comprimidos para producir tabletas se preparan utilizando agua o unasolución acuosa de etanol o similar.
ARP970100776A 1996-02-29 1997-02-27 Tabletas que contienen antibioticos de beta-lactamas y un metodo para obtenerlas AR006012A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP4274396 1996-02-29
JP32026496 1996-11-29

Publications (1)

Publication Number Publication Date
AR006012A1 true AR006012A1 (es) 1999-07-21

Family

ID=26382481

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP970100776A AR006012A1 (es) 1996-02-29 1997-02-27 Tabletas que contienen antibioticos de beta-lactamas y un metodo para obtenerlas

Country Status (24)

Country Link
US (4) US6423341B1 (es)
EP (2) EP0890359B1 (es)
JP (1) JP3180350B2 (es)
KR (1) KR20040058360A (es)
CN (2) CN1136853C (es)
AR (1) AR006012A1 (es)
AT (2) ATE216887T1 (es)
AU (1) AU724946B2 (es)
BR (1) BR9707780A (es)
CA (1) CA2248179C (es)
DE (2) DE69712332T2 (es)
DK (2) DK0890359T3 (es)
EA (1) EA001089B1 (es)
ES (2) ES2231369T3 (es)
HK (1) HK1015684A1 (es)
HU (1) HU227821B1 (es)
IL (1) IL125214A0 (es)
MX (1) MX9806265A (es)
NZ (2) NZ330864A (es)
PT (2) PT890359E (es)
TR (1) TR199801680T2 (es)
TW (1) TW473393B (es)
WO (1) WO1997031639A1 (es)
ZA (1) ZA971584B (es)

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Also Published As

Publication number Publication date
DE69732312T2 (de) 2006-04-06
AU724946B2 (en) 2000-10-05
BR9707780A (pt) 1999-07-27
KR20040058360A (ko) 2004-07-03
NZ330864A (en) 2001-07-27
DE69712332D1 (de) 2002-06-06
EA001089B1 (ru) 2000-10-30
CN1409995A (zh) 2003-04-16
MX9806265A (es) 1998-12-31
CA2248179A1 (en) 1997-09-04
TR199801680T2 (xx) 1999-02-22
IL125214A0 (en) 1999-03-12
EA199800775A1 (ru) 1999-02-25
EP0890359B1 (en) 2002-05-02
CA2248179C (en) 2007-09-18
EP0890359A4 (es) 1999-01-13
ATE287218T1 (de) 2005-02-15
EP1166651B1 (en) 2005-01-19
DK1166651T3 (da) 2005-05-30
ES2173420T3 (es) 2002-10-16
US20020192281A1 (en) 2002-12-19
EP1166651A1 (en) 2002-01-02
HU227821B1 (en) 2012-03-28
US20020051816A1 (en) 2002-05-02
HUP9901877A3 (en) 2000-04-28
US20070134325A1 (en) 2007-06-14
JP3180350B2 (ja) 2001-06-25
PT1166651E (pt) 2005-04-29
DE69732312D1 (de) 2005-02-24
ATE216887T1 (de) 2002-05-15
NZ512609A (en) 2003-03-28
EP0890359A1 (en) 1999-01-13
AU1734797A (en) 1997-09-16
PT890359E (pt) 2003-03-31
DE69732312T8 (de) 2006-07-27
ZA971584B (en) 1997-09-10
US20030129227A1 (en) 2003-07-10
WO1997031639A1 (fr) 1997-09-04
HUP9901877A1 (hu) 1999-12-28
DK0890359T3 (da) 2002-07-01
CN1212626A (zh) 1999-03-31
DE69712332T2 (de) 2002-10-02
CN1136853C (zh) 2004-02-04
TW473393B (en) 2002-01-21
US6423341B1 (en) 2002-07-23
HK1015684A1 (en) 1999-10-22
ES2231369T3 (es) 2005-05-16

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