AP2013006706A0 - Napht-2-ylacetic acid derivatives to treat AIDS - Google Patents

Napht-2-ylacetic acid derivatives to treat AIDS

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Publication number
AP2013006706A0
AP2013006706A0 AP2013006706A AP2013006706A AP2013006706A0 AP 2013006706 A0 AP2013006706 A0 AP 2013006706A0 AP 2013006706 A AP2013006706 A AP 2013006706A AP 2013006706 A AP2013006706 A AP 2013006706A AP 2013006706 A0 AP2013006706 A0 AP 2013006706A0
Authority
AP
ARIPO
Prior art keywords
napht
acid derivatives
ylacetic acid
treat aids
aids
Prior art date
Application number
AP2013006706A
Other languages
English (en)
Inventor
John O Link
Kyla Bjornson
Kerim Babaoglu
Original Assignee
Gilead Sciences Inc
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44454746&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP2013006706(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of AP2013006706A0 publication Critical patent/AP2013006706A0/xx

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    • C07C59/40—Unsaturated compounds
    • C07C59/58—Unsaturated compounds containing ether groups, groups, groups, or groups
    • C07C59/64—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
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    • C07C57/58—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing halogen containing six-membered aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • C07C233/00—Carboxylic acid amides
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    • C07C233/47—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
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