AP120A - Quinuclidine therapeutic agents - Google Patents

Quinuclidine therapeutic agents Download PDF

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Publication number
AP120A
AP120A APAP/P/1989/000152A AP8900152A AP120A AP 120 A AP120 A AP 120A AP 8900152 A AP8900152 A AP 8900152A AP 120 A AP120 A AP 120A
Authority
AP
ARIPO
Prior art keywords
cis
carbon atoms
quinuclidine
methylamino
compound
Prior art date
Application number
APAP/P/1989/000152A
Other languages
English (en)
Other versions
AP8900152A0 (en
Inventor
Iii John Adams Lowe
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of AP8900152A0 publication Critical patent/AP8900152A0/xx
Application granted granted Critical
Publication of AP120A publication Critical patent/AP120A/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
APAP/P/1989/000152A 1988-11-23 1989-11-22 Quinuclidine therapeutic agents AP120A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US1988/004205 WO1990005525A1 (en) 1988-11-23 1988-11-23 Quinuclidine derivatives as substance p antagonists

Publications (2)

Publication Number Publication Date
AP8900152A0 AP8900152A0 (en) 1990-01-31
AP120A true AP120A (en) 1991-02-20

Family

ID=22209014

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/1989/000152A AP120A (en) 1988-11-23 1989-11-22 Quinuclidine therapeutic agents

Country Status (29)

Country Link
US (1) US5162339A (zh)
EP (1) EP0409931B1 (zh)
JP (1) JPH0647589B2 (zh)
KR (1) KR900701782A (zh)
CN (1) CN1026111C (zh)
AP (1) AP120A (zh)
AR (1) AR246522A1 (zh)
AT (1) ATE101608T1 (zh)
AU (1) AU617906B2 (zh)
CA (1) CA2003441C (zh)
DD (1) DD285605A5 (zh)
DE (1) DE68913194T2 (zh)
EG (1) EG19301A (zh)
ES (1) ES2062504T3 (zh)
FI (1) FI903656A0 (zh)
HU (1) HU900517D0 (zh)
IE (1) IE893730L (zh)
IL (1) IL92336A0 (zh)
MA (1) MA21682A1 (zh)
MX (1) MX18467A (zh)
MY (1) MY105061A (zh)
NZ (1) NZ231461A (zh)
OA (1) OA10023A (zh)
PH (1) PH26590A (zh)
PL (1) PL161864B1 (zh)
PT (1) PT92361B (zh)
WO (2) WO1990005525A1 (zh)
YU (1) YU47097B (zh)
ZA (1) ZA898901B (zh)

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CA2003441A1 (en) 1990-05-23
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US5162339A (en) 1992-11-10
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