ZA200510194B - Benzazepine derivatives useful for the treatment of 5HT2C receptor associated diseases - Google Patents

Benzazepine derivatives useful for the treatment of 5HT2C receptor associated diseases Download PDF

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Publication number
ZA200510194B
ZA200510194B ZA200510194A ZA200510194A ZA200510194B ZA 200510194 B ZA200510194 B ZA 200510194B ZA 200510194 A ZA200510194 A ZA 200510194A ZA 200510194 A ZA200510194 A ZA 200510194A ZA 200510194 B ZA200510194 B ZA 200510194B
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South Africa
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alkyl
haloalkyl
halo
heteroaryl
aryl
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ZA200510194A
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English (en)
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Beverly W Throop
Aytes Shelley
Sengupta Dipanjan
Rey Max
Charles A Gilson Iii
Scott A Estrada
Smith Brian
Weigl Ulrich
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Arena Pharmaceticals Inc
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Publication of ZA200510194B publication Critical patent/ZA200510194B/en

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16—Benzazepines; Hydrogenated benzazepines

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  • Endocrinology (AREA)
  • Heart & Thoracic Surgery (AREA)
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ZA200510194A 2003-06-17 2005-12-14 Benzazepine derivatives useful for the treatment of 5HT2C receptor associated diseases ZA200510194B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US47928003P 2003-06-17 2003-06-17

Publications (1)

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ZA200510194B true ZA200510194B (en) 2007-02-28

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ZA200510194A ZA200510194B (en) 2003-06-17 2005-12-14 Benzazepine derivatives useful for the treatment of 5HT2C receptor associated diseases
ZA200510255A ZA200510255B (en) 2003-06-17 2005-12-15 Benzazepine derivatives useful for the treatment of 5HT2C receptor associated diseases

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ZA200510255A ZA200510255B (en) 2003-06-17 2005-12-15 Benzazepine derivatives useful for the treatment of 5HT2C receptor associated diseases

Country Status (14)

Country Link
US (3) US7704993B2 (https=)
EP (2) EP1633720A1 (https=)
JP (2) JP4782003B2 (https=)
KR (1) KR101152521B1 (https=)
CN (4) CN1805938B (https=)
AU (1) AU2004253888B2 (https=)
BR (1) BRPI0411470A (https=)
CA (2) CA2888392A1 (https=)
EA (1) EA016558B1 (https=)
IL (1) IL172334A (https=)
MX (1) MXPA05013366A (https=)
NZ (1) NZ578503A (https=)
WO (1) WO2005003096A1 (https=)
ZA (2) ZA200510194B (https=)

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JPWO2011071136A1 (ja) 2009-12-11 2013-04-22 アステラス製薬株式会社 線維筋痛症治療剤
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CA3002525A1 (en) * 2015-07-31 2017-02-09 Arena Pharmaceuticals, Inc. 5-ht2c receptor agonists and compositions and methods of use
CN105777638B (zh) * 2016-01-06 2019-07-30 北京修正创新药物研究院有限公司 氯卡色林杂质的制备方法
CN106631823B (zh) * 2016-12-20 2022-04-26 天津泰普制药有限公司 一种氯卡色林中间体的制备方法
CN107353250B (zh) * 2016-12-27 2019-11-12 开封制药(集团)有限公司 一种氯卡色林的合成方法
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