YU32799A - Novi prostaglandini agonisti, njihove smeše i kompleti koji ih sadrže - Google Patents

Novi prostaglandini agonisti, njihove smeše i kompleti koji ih sadrže

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Publication number
YU32799A
YU32799A YU32799A YU32799A YU32799A YU 32799 A YU32799 A YU 32799A YU 32799 A YU32799 A YU 32799A YU 32799 A YU32799 A YU 32799A YU 32799 A YU32799 A YU 32799A
Authority
YU
Yugoslavia
Prior art keywords
agonists
prostaglandines
compositions
new
kits containing
Prior art date
Application number
YU32799A
Other languages
English (en)
Inventor
Kimberly O'keefe Cameron
Hua Zhu Ke
Bruce Allen Lefker
Robert Louis Rosati
David Duane Thompson
Original Assignee
Pfizer Inc.
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Filing date
Publication date
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of YU32799A publication Critical patent/YU32799A/sh

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    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
    • C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
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    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane

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Abstract

Opisana su nova jedinjenja formule (I) u kojima, na primer, A je sulfonil ili acil grupa, B je N ili CH, M sadrži neki prsten, a K i Q su vezujuće grupe, farmaceutski sastavi koji sadrže takve prostaglandin agoniste i kompleti korisni u tretmanu koštanih poremećaja uključujući osteoporozu.[Prostaglandin agonists of formula (I), in which, for example, A is a sulphonyl or acyl group, B is N or CH, M contains a ring and K and Q are linking groups, methods of using such prostaglandin agonists, pharmaceutical compositions containing such prostaglandin agonists and kits useful for the treatment of bone disorders including osteoporosis.
YU32799A 1996-12-20 1997-11-10 Novi prostaglandini agonisti, njihove smeše i kompleti koji ih sadrže YU32799A (sh)

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US6288120B1 (en) 2001-09-11
CA2275479C (en) 2007-05-08
HUP0000739A2 (hu) 2000-09-28
BR9714155A (pt) 2000-05-02
EA003529B1 (ru) 2003-06-26
CZ223399A3 (cs) 2000-08-16
EP0946501A1 (en) 1999-10-06
JP2000514827A (ja) 2000-11-07
AR010843A1 (es) 2000-07-12
AU721260B2 (en) 2000-06-29
CA2275479A1 (en) 1998-07-02
EA200200806A1 (ru) 2003-02-27
EP0946501B1 (en) 2006-05-31
PT946501E (pt) 2006-10-31
KR100311566B1 (ko) 2001-11-03
IS5055A (is) 1999-05-21
KR20000057684A (ko) 2000-09-25
DZ2375A1 (fr) 2002-12-28
HUP0000739A3 (en) 2001-02-28
DK0946501T3 (da) 2006-10-02
PL192670B1 (pl) 2006-11-30
SA05260204B1 (ar) 2008-07-14
US20030105092A1 (en) 2003-06-05
OA11065A (en) 2002-11-15
US20020016368A1 (en) 2002-02-07
JP2005068154A (ja) 2005-03-17
US6998423B2 (en) 2006-02-14
IL130306A (en) 2008-12-29
MA24425A1 (fr) 1998-07-01
TR199901366T2 (xx) 1999-09-21
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ATE327976T1 (de) 2006-06-15
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SA97180721A (ar) 2005-12-03
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ZA9711437B (en) 1999-06-21
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PA8443001A1 (es) 2000-05-24
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MY141384A (en) 2010-04-30
PE47499A1 (es) 1999-05-13
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WO1998028264A1 (en) 1998-07-02
JP3679418B2 (ja) 2005-08-03
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