WO2008126797A1 - 微粉砕化有機化合物粒子の製造方法 - Google Patents

微粉砕化有機化合物粒子の製造方法 Download PDF

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Publication number
WO2008126797A1
WO2008126797A1 PCT/JP2008/056799 JP2008056799W WO2008126797A1 WO 2008126797 A1 WO2008126797 A1 WO 2008126797A1 JP 2008056799 W JP2008056799 W JP 2008056799W WO 2008126797 A1 WO2008126797 A1 WO 2008126797A1
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WIPO (PCT)
Prior art keywords
organic compound
compound particle
poorly water
producing
medical use
Prior art date
Application number
PCT/JP2008/056799
Other languages
English (en)
French (fr)
Inventor
Takashi Hirokawa
Takahiro Tada
Original Assignee
Activus Pharma Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Activus Pharma Co., Ltd. filed Critical Activus Pharma Co., Ltd.
Priority to CN2008800084620A priority Critical patent/CN101636150B/zh
Priority to EP08739905.1A priority patent/EP2143423B1/en
Priority to KR1020097014759A priority patent/KR101369061B1/ko
Priority to ES08739905.1T priority patent/ES2563979T3/es
Priority to JP2009509328A priority patent/JP5317960B2/ja
Priority to CA2679929A priority patent/CA2679929C/en
Publication of WO2008126797A1 publication Critical patent/WO2008126797A1/ja
Priority to IL201169A priority patent/IL201169A/en
Priority to US12/585,786 priority patent/US8226983B2/en
Priority to US13/484,460 priority patent/US20120237768A1/en
Priority to IL223087A priority patent/IL223087A/en

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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
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    • Y10T428/29—Coated or structually defined flake, particle, cell, strand, strand portion, rod, filament, macroscopic fiber or mass thereof
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Abstract

　本発明は、難水溶性であり、かつ、結晶性である有機化合物の微粉砕化粒子の製造方法、及び、該製造方法により製造された微粉砕化有機化合物粒子の提供することを目的とする。特に、本発明は、難水溶性医療用有機化合物を、生理学的に許容される塩及び生理学的に許容されるポリオールと混合して、前記有機化合物を湿式粉砕することを特徴とする、難水溶性医療用有機化合物微粒子の製造方法、及び該製造方法により得られる難水溶性医療用有機化合物微粒子を提供することを目的とする。
PCT/JP2008/056799 2007-04-06 2008-04-04 微粉砕化有機化合物粒子の製造方法 WO2008126797A1 (ja)

Priority Applications (10)

Application Number Priority Date Filing Date Title
CN2008800084620A CN101636150B (zh) 2007-04-06 2008-04-04 难水溶性医疗用有机化合物微粒子的制造方法
EP08739905.1A EP2143423B1 (en) 2007-04-06 2008-04-04 Method for producing pulverized organic compound particle
KR1020097014759A KR101369061B1 (ko) 2007-04-06 2008-04-04 미분쇄화 유기 화합물 입자의 제조 방법
ES08739905.1T ES2563979T3 (es) 2007-04-06 2008-04-04 Método para producción de partículas de compuesto orgánico pulverizadas
JP2009509328A JP5317960B2 (ja) 2007-04-06 2008-04-04 微粉砕化有機化合物粒子の製造方法
CA2679929A CA2679929C (en) 2007-04-06 2008-04-04 Method for producing finely pulverized organic compound particle
IL201169A IL201169A (en) 2007-04-06 2009-09-24 A method for producing crushed particles of organic compound
US12/585,786 US8226983B2 (en) 2007-04-06 2009-09-24 Method for producing pulverized organic compound particle
US13/484,460 US20120237768A1 (en) 2007-04-06 2012-05-31 Method for producing pulverized organic compound particle
IL223087A IL223087A (en) 2007-04-06 2012-11-18 Thin crushed organic compound particles

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JP2007-100902 2007-04-06
JP2007100902 2007-04-06
JP2007-210370 2007-08-10
JP2007210370 2007-08-10

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CA (1) CA2679929C (ja)
ES (1) ES2563979T3 (ja)
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WO2011001214A1 (en) * 2009-06-30 2011-01-06 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi Surface amorphization of phenprobamate
WO2011118960A2 (ko) 2010-03-22 2011-09-29 (주)바이오시네틱스 나노입자 제조방법
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CN101636150A (zh) 2010-01-27
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CA2679929C (en) 2014-12-16
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KR20100014315A (ko) 2010-02-10
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