UY30588A1 - Compuestos de 4-metilpiridopirimidinona - Google Patents

Compuestos de 4-metilpiridopirimidinona

Info

Publication number
UY30588A1
UY30588A1 UY30588A UY30588A UY30588A1 UY 30588 A1 UY30588 A1 UY 30588A1 UY 30588 A UY30588 A UY 30588A UY 30588 A UY30588 A UY 30588A UY 30588 A1 UY30588 A1 UY 30588A1
Authority
UY
Uruguay
Prior art keywords
compounds
methylpiridopirimidinone
alpha
methylpyridopyrimidinonna
phosphoinositide
Prior art date
Application number
UY30588A
Other languages
English (en)
Spanish (es)
Inventor
Khanh Tuan Tran
Phuong Thi Quy Le
Mary Catherine Johnson
Jacqui Elizabeth Hoffman
Mason Alan Pairish
Mitchell David Nambu
Hengmiao Cheng
Klaus Ruprecht Dress
Robert Steven Kania
Michael Bruno Plewe
Dilip Bhumralkar
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of UY30588A1 publication Critical patent/UY30588A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pyridine Compounds (AREA)
UY30588A 2006-09-15 2007-09-12 Compuestos de 4-metilpiridopirimidinona UY30588A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US84506506P 2006-09-15 2006-09-15
US94785207P 2007-07-03 2007-07-03
US95262807P 2007-07-30 2007-07-30

Publications (1)

Publication Number Publication Date
UY30588A1 true UY30588A1 (es) 2008-05-02

Family

ID=38859750

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30588A UY30588A1 (es) 2006-09-15 2007-09-12 Compuestos de 4-metilpiridopirimidinona

Country Status (41)

Country Link
US (3) US7696213B2 (enExample)
EP (1) EP2074122B9 (enExample)
JP (1) JP4718637B2 (enExample)
KR (1) KR101099926B1 (enExample)
CN (1) CN101573358B (enExample)
AP (1) AP2710A (enExample)
AR (1) AR062785A1 (enExample)
AT (1) ATE514695T1 (enExample)
AU (1) AU2007297212B8 (enExample)
BR (1) BRPI0716749B8 (enExample)
CA (1) CA2663401C (enExample)
CL (1) CL2007002682A1 (enExample)
CR (1) CR10662A (enExample)
CU (1) CU23783B7 (enExample)
CY (1) CY1111911T1 (enExample)
DK (1) DK2074122T5 (enExample)
DO (1) DOP2009000039A (enExample)
EA (1) EA016388B1 (enExample)
ES (1) ES2366489T3 (enExample)
GE (1) GEP20115306B (enExample)
GT (1) GT200700077A (enExample)
HN (1) HN2007000267A (enExample)
HR (1) HRP20110621T2 (enExample)
IL (1) IL197243A (enExample)
MA (1) MA30709B1 (enExample)
ME (1) MEP8009A (enExample)
MX (1) MX2009002927A (enExample)
MY (1) MY146420A (enExample)
NI (1) NI200900032A (enExample)
NO (1) NO342357B1 (enExample)
NZ (1) NZ575167A (enExample)
PE (1) PE20080670A1 (enExample)
PL (1) PL2074122T3 (enExample)
PT (1) PT2074122E (enExample)
RS (2) RS20090104A (enExample)
SI (1) SI2074122T1 (enExample)
TN (1) TN2009000085A1 (enExample)
TW (1) TWI334353B (enExample)
UY (1) UY30588A1 (enExample)
WO (1) WO2008032162A1 (enExample)
ZA (1) ZA200901477B (enExample)

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CN105330699B (zh) * 2014-08-13 2018-12-04 山东汇睿迪生物技术有限公司 一种含磷吡啶并[2,3-d]嘧啶-7-酮类化合物或其药学上可接受的盐、药物组合物及其应用
JP6784668B2 (ja) 2014-10-10 2020-11-11 ファイザー・インク 相乗的オーリスタチン組合せ
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Also Published As

Publication number Publication date
HK1138589A1 (en) 2010-08-27
DK2074122T5 (da) 2014-03-17
NO20091141L (no) 2009-03-31
AP2009004790A0 (en) 2009-04-30
TN2009000085A1 (fr) 2010-08-19
GT200700077A (es) 2009-08-03
MEP8009A (en) 2011-12-20
CA2663401A1 (en) 2008-03-20
CY1111911T1 (el) 2015-11-04
SI2074122T1 (sl) 2011-10-28
PE20080670A1 (es) 2008-06-14
KR101099926B1 (ko) 2011-12-28
NZ575167A (en) 2010-10-29
TW200820972A (en) 2008-05-16
AU2007297212A1 (en) 2008-03-20
JP2010503653A (ja) 2010-02-04
RS20090104A (sr) 2010-06-30
ATE514695T1 (de) 2011-07-15
US8273755B2 (en) 2012-09-25
CA2663401C (en) 2011-07-12
KR20090040389A (ko) 2009-04-23
CU20090040A7 (es) 2011-07-11
CL2007002682A1 (es) 2008-04-04
IL197243A0 (en) 2009-12-24
ES2366489T3 (es) 2011-10-20
MX2009002927A (es) 2009-03-31
EA016388B1 (ru) 2012-04-30
JP4718637B2 (ja) 2011-07-06
US7696213B2 (en) 2010-04-13
AU2007297212B2 (en) 2011-04-14
ZA200901477B (en) 2010-07-28
AU2007297212B8 (en) 2011-04-28
EP2074122B9 (en) 2013-09-11
CR10662A (es) 2009-04-17
HRP20110621T2 (hr) 2013-12-06
HRP20110621T1 (hr) 2011-09-30
US20100137279A1 (en) 2010-06-03
EA200970207A1 (ru) 2009-08-28
MY146420A (en) 2012-08-15
US20120309775A1 (en) 2012-12-06
AR062785A1 (es) 2008-12-03
US8633204B2 (en) 2014-01-21
IL197243A (en) 2013-07-31
DOP2009000039A (es) 2015-12-15
CN101573358A (zh) 2009-11-04
EP2074122A1 (en) 2009-07-01
DK2074122T3 (da) 2011-08-15
EP2074122B1 (en) 2011-06-29
TWI334353B (en) 2010-12-11
PT2074122E (pt) 2011-08-24
PL2074122T3 (pl) 2011-10-31
HN2007000267A (es) 2011-02-25
US20080090801A1 (en) 2008-04-17
BRPI0716749B8 (pt) 2021-05-25
WO2008032162A1 (en) 2008-03-20
ES2366489T9 (es) 2013-12-27
WO2008032162A8 (en) 2009-03-26
CN101573358B (zh) 2012-05-30
GEP20115306B (enExample) 2011-10-10
CU23783B7 (es) 2012-02-15
BRPI0716749A2 (pt) 2014-02-18
MA30709B1 (fr) 2009-09-01
NO342357B1 (no) 2018-05-14
RS51927B (sr) 2012-02-29
NI200900032A (es) 2010-05-14
AP2710A (en) 2013-07-30
BRPI0716749B1 (pt) 2020-10-06

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