UY31134A1 - Derivados de piperidina/piperazina (i) - Google Patents

Derivados de piperidina/piperazina (i)

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Publication number
UY31134A1
UY31134A1 UY31134A UY31134A UY31134A1 UY 31134 A1 UY31134 A1 UY 31134A1 UY 31134 A UY31134 A UY 31134A UY 31134 A UY31134 A UY 31134A UY 31134 A1 UY31134 A1 UY 31134A1
Authority
UY
Uruguay
Prior art keywords
piperidine
piperazine derivatives
compounds
dgat inhibitor
medicaments
Prior art date
Application number
UY31134A
Other languages
English (en)
Inventor
Braeken Mirielle
Davidenko Petr Vladimirivich
Roevens Peter Walter Maria
Waepenaert Katharina Antonia Germania J M De
Berwaer Monique Jenny Marie
Buyck Christophe Francis Robert Nestor
Coesemans Erwin
Van Lommen Guy Rosalia Eguren
Joannes Theodorus Mari Linders
Lieven Meerpoel
Jean Pierre Andre Mar Bongartz
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38616252&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY31134(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of UY31134A1 publication Critical patent/UY31134A1/es

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/451—Non condensed piperidines, e.g. piperocaine having a carbocyclic group directly attached to the heterocyclic ring, e.g. glutethimide, meperidine, loperamide, phencyclidine, piminodine
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Abstract

La invencion se refiere a un inhibidor de DGAT de formula incluyendo sus isomeros esteroquímicos, donde a representa CH o N; la línea punteada representa un enlace opcional en caso que A sea un átomo de carbono. También se refiere a métodos para preparar tales compuestos, a composiciones farmacéuticas y al uso como medicamentos, como inhibidor de DGAT, de dichos compuestos.
UY31134A 2007-06-08 2008-06-09 Derivados de piperidina/piperazina (i) UY31134A1 (es)

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US9227935B2 (en) 2016-01-05
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TW200916449A (en) 2009-04-16
US8946228B2 (en) 2015-02-03
CA2687243C (en) 2016-07-12
RU2478628C2 (ru) 2013-04-10
AU2008258558A1 (en) 2008-12-11
WO2008148849A3 (en) 2009-04-16
TWI438197B (zh) 2014-05-21
CA2687243A1 (en) 2008-12-11
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AU2008258558B2 (en) 2013-11-07
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US20150087629A1 (en) 2015-03-26
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JP2010529085A (ja) 2010-08-26
PA8783401A1 (es) 2009-01-23
WO2008148849A2 (en) 2008-12-11
ES2522617T3 (es) 2014-11-17
AR066153A1 (es) 2009-07-29
US20100210618A1 (en) 2010-08-19
PE20090820A1 (es) 2009-06-27
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