EA200401289A1 - Новые противоинфекционные соединения, способы их получения и фармацевтические композиции, содержащие эти соединения - Google Patents
Новые противоинфекционные соединения, способы их получения и фармацевтические композиции, содержащие эти соединенияInfo
- Publication number
- EA200401289A1 EA200401289A1 EA200401289A EA200401289A EA200401289A1 EA 200401289 A1 EA200401289 A1 EA 200401289A1 EA 200401289 A EA200401289 A EA 200401289A EA 200401289 A EA200401289 A EA 200401289A EA 200401289 A1 EA200401289 A1 EA 200401289A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- methods
- pharmaceutical compositions
- compositions containing
- connections
- production
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
Настоящее изобретение относится к новым противоинфекционным соединениям, к способам их получения и к фармацевтическим композициям, содержащим указанные соединения.Отчет о международном поиске был опубликован 2003.11.13.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN310MU2002 | 2002-04-01 | ||
PCT/IN2003/000081 WO2003082864A2 (en) | 2002-04-01 | 2003-03-26 | Antiinfectve compounds, process for their preparation and pharmaceutical compositions containing them |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200401289A1 true EA200401289A1 (ru) | 2005-04-28 |
Family
ID=28460710
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200401289A EA200401289A1 (ru) | 2002-04-01 | 2003-03-26 | Новые противоинфекционные соединения, способы их получения и фармацевтические композиции, содержащие эти соединения |
Country Status (8)
Country | Link |
---|---|
US (1) | US20060229316A1 (ru) |
EP (1) | EP1495021A2 (ru) |
AU (1) | AU2003231920A1 (ru) |
BR (1) | BR0308837A (ru) |
CA (1) | CA2478502A1 (ru) |
EA (1) | EA200401289A1 (ru) |
WO (1) | WO2003082864A2 (ru) |
ZA (1) | ZA200406844B (ru) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2513416A1 (en) * | 2002-08-22 | 2004-03-04 | Orchid Chemicals & Pharmaceuticals Ltd. | Novel antibacterial agents |
AU2002953533A0 (en) * | 2002-12-24 | 2003-01-16 | Arthron Limited | Fc receptor modulating compounds and compositions |
US20040204463A1 (en) * | 2003-04-01 | 2004-10-14 | Harris Christina Renee | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
US20080139574A1 (en) * | 2006-11-30 | 2008-06-12 | Cadila Healthcare Limited | Novel quinoline derivatives |
RU2478619C2 (ru) | 2006-12-11 | 2013-04-10 | Ривайва Фармасьютикалс, Инк. | Композиции, синтез и способы применения ингибиторов холинэстеразы на основе инданона |
WO2008148851A1 (en) | 2007-06-08 | 2008-12-11 | Janssen Pharmaceutica N.V. | Piperidine/piperazine derivatives |
PE20090362A1 (es) | 2007-06-08 | 2009-04-04 | Janssen Pharmaceutica Nv | Derivados de piperidina/piperazina como moduladores de dgat |
JP5443342B2 (ja) | 2007-06-08 | 2014-03-19 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | ピペリジン/ピペラジン誘導体 |
JO2972B1 (en) | 2007-06-08 | 2016-03-15 | جانسين فارماسوتيكا ان. في | Piperidine / piperazine derivatives |
CA2692255A1 (en) * | 2007-06-22 | 2008-12-31 | Orchid Research Laboratories Limited | Novel compounds and their use |
WO2009147170A2 (en) | 2008-06-05 | 2009-12-10 | Janssen Pharmaceutica Nv | Drug combinations comprising a dgat inhibitor and a ppar-agonist |
FR3123565A1 (fr) * | 2021-06-04 | 2022-12-09 | Institut Des Sciences Et Industries Du Vivant Et De L'environnement - Agroparistech | Nouvelles molecules derivees de furanacrylates et 5-hydroxymethyl furanacrylates presentant des proprietes filtre uv-b et/ou antimicrobiennes |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SK283420B6 (sk) * | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
GB9614236D0 (en) * | 1996-07-06 | 1996-09-04 | Zeneca Ltd | Chemical compounds |
BR9910971A (pt) * | 1998-06-05 | 2001-02-13 | Astrazeneca Ab | Composto, processos para a preparação de um composto e para produzir um efeito antibacteriano em um animal de sangue quente, uso de um composto, e, composição farmacêutica |
US20010047004A1 (en) * | 2000-02-10 | 2001-11-29 | Hester Jackson B. | Oxazolidinone thioamides with piperazine amide substituents |
US6642238B2 (en) * | 2000-02-10 | 2003-11-04 | Pharmacia And Upjohn Company | Oxazolidinone thioamides with piperazine amide substituents |
NZ523700A (en) * | 2000-07-17 | 2004-11-26 | Ranbaxy Lab Ltd | Oxazolidinone derivatives as antimicrobials |
US20040204463A1 (en) * | 2003-04-01 | 2004-10-14 | Harris Christina Renee | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
-
2003
- 2003-03-26 US US10/509,892 patent/US20060229316A1/en not_active Abandoned
- 2003-03-26 AU AU2003231920A patent/AU2003231920A1/en not_active Abandoned
- 2003-03-26 EP EP03745394A patent/EP1495021A2/en not_active Withdrawn
- 2003-03-26 CA CA002478502A patent/CA2478502A1/en not_active Abandoned
- 2003-03-26 EA EA200401289A patent/EA200401289A1/ru unknown
- 2003-03-26 WO PCT/IN2003/000081 patent/WO2003082864A2/en not_active Application Discontinuation
- 2003-03-26 BR BR0308837-5A patent/BR0308837A/pt not_active IP Right Cessation
-
2004
- 2004-08-27 ZA ZA200406844A patent/ZA200406844B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
BR0308837A (pt) | 2005-02-01 |
AU2003231920A8 (en) | 2003-10-13 |
EP1495021A2 (en) | 2005-01-12 |
WO2003082864A2 (en) | 2003-10-09 |
CA2478502A1 (en) | 2003-10-09 |
WO2003082864A3 (en) | 2003-11-13 |
ZA200406844B (en) | 2006-05-31 |
US20060229316A1 (en) | 2006-10-12 |
AU2003231920A1 (en) | 2003-10-13 |
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