EA200601608A1 - Способ производства твёрдой фармацевтической композиции - Google Patents

Способ производства твёрдой фармацевтической композиции

Info

Publication number
EA200601608A1
EA200601608A1 EA200601608A EA200601608A EA200601608A1 EA 200601608 A1 EA200601608 A1 EA 200601608A1 EA 200601608 A EA200601608 A EA 200601608A EA 200601608 A EA200601608 A EA 200601608A EA 200601608 A1 EA200601608 A1 EA 200601608A1
Authority
EA
Eurasian Patent Office
Prior art keywords
production
pharmaceutical composition
firm
perindopril
tablets
Prior art date
Application number
EA200601608A
Other languages
English (en)
Other versions
EA011712B1 (ru
Inventor
Изток Клобчар
Алеша Пунчух Колар
Аница Грандовец
Уршка Турк
Полона Шольмайер-Лампич
Original Assignee
Крка, Товарна Здравил, Д. Д. Ново Место
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34963866&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200601608(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE200410019845 external-priority patent/DE102004019845A1/de
Priority claimed from DE102004059521A external-priority patent/DE102004059521A1/de
Application filed by Крка, Товарна Здравил, Д. Д. Ново Место filed Critical Крка, Товарна Здравил, Д. Д. Ново Место
Publication of EA200601608A1 publication Critical patent/EA200601608A1/ru
Publication of EA011712B1 publication Critical patent/EA011712B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Abstract

Изобретение относится к способу производства твердой фармацевтической композиции периндоприла или его соли, который позволяет избежать стадии влажной грануляции и получить очень стабильные фармацевтические композиции, такие как таблетки.
EA200601608A 2004-03-29 2005-03-29 Способ производства твёрдой фармацевтической композиции EA011712B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE200410019845 DE102004019845A1 (de) 2004-03-29 2004-03-29 Verfahren zur Herstellung einer festen pharmazeutischen Zusammensetzung
DE102004059521A DE102004059521A1 (de) 2004-12-09 2004-12-09 Verfahren zur Herstellung einer festen pharmazeutischen Zusammensetzung
PCT/EP2005/003277 WO2005094793A1 (en) 2004-03-29 2005-03-29 Process for preparing a solid pharmaceutical composition

Publications (2)

Publication Number Publication Date
EA200601608A1 true EA200601608A1 (ru) 2007-02-27
EA011712B1 EA011712B1 (ru) 2009-04-28

Family

ID=34963866

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200601608A EA011712B1 (ru) 2004-03-29 2005-03-29 Способ производства твёрдой фармацевтической композиции

Country Status (14)

Country Link
US (2) US20070172524A1 (ru)
EP (1) EP1729739B1 (ru)
JP (1) JP4948392B2 (ru)
CY (1) CY1118180T1 (ru)
DK (1) DK1729739T3 (ru)
EA (1) EA011712B1 (ru)
ES (1) ES2603856T3 (ru)
HR (1) HRP20161602T1 (ru)
HU (1) HUE031058T2 (ru)
LT (1) LT1729739T (ru)
NO (1) NO20064934L (ru)
PL (1) PL1729739T3 (ru)
PT (1) PT1729739T (ru)
WO (1) WO2005094793A1 (ru)

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ES2603856T3 (es) 2004-03-29 2017-03-01 Les Laboratoires Servier Procedimiento para preparar una composición farmacéutica sólida
SI21800A (sl) * 2004-05-14 2005-12-31 Krka, Tovarna Zdravil, D.D., Novo Mesto Nov postopek sinteze perindoprila
BRPI0615607A2 (pt) * 2005-08-30 2011-05-24 Lek Pharmaceuticals composição farmacêutica compreendendo perindopril ou seus sais
RS53324B (en) * 2005-11-17 2014-10-31 Silverstone Pharma Est. STABLE FORMULATION OF AMORPHIC SALES OF PERINDOPRIL, PROCEDURE FOR THEIR PREPARATION, IN PARTICULAR INDUSTRIAL PREPARATION, AND THEIR USE IN HYPERTENSION THERAPY
EP1815857A1 (en) 2006-02-02 2007-08-08 LEK Pharmaceuticals D.D. A pharmaceutical composition comprising perindopril
EP1901739A2 (en) * 2006-04-19 2008-03-26 Teva Pharmaceutical Industries Ltd Stable pharmaceutical compositions of 2-aza-bicyclo[3.3.0]-octane-3-carboxylic acid derivatives
JP2009537538A (ja) * 2006-05-15 2009-10-29 アカドイア プハルマセウチカルス インコーポレーテッド ピマバンセリン医薬製剤
WO2008068577A2 (en) * 2006-12-01 2008-06-12 Glenmark Pharmaceuticals Limited Pharmaceutical compositions
TWI435917B (zh) 2006-12-27 2014-05-01 Fujifilm Corp 顏料分散組成物、硬化性組成物、彩色濾光片及其製造方法
US8536196B2 (en) * 2007-01-18 2013-09-17 Evolva Sa Substituted 1,3-dioxanes useful as PPAR modulators
SI22543A (sl) 2007-06-27 2008-12-31 Krka, Tovarna Zdravil, D.D., Novo Mesto Nove soli perindoprila
CN102665764A (zh) * 2009-12-22 2012-09-12 Fmc有限公司 可用作可再压实药物赋形剂的微晶纤维素和碳酸钙组合物
PL227900B1 (pl) 2012-11-15 2018-01-31 Adamed Spolka Z Ograniczona Odpowiedzialnoscia Kompozycja farmaceutyczna zawierająca inhibitor ACE i bloker kanałów wapniowych, sposób jej wytwarzania i jednostka dawkowania zawierająca tę kompozycję
WO2016178591A2 (en) 2015-05-05 2016-11-10 Gene Predit, Sa Genetic markers and treatment of male obesity
CN109700774A (zh) * 2019-03-05 2019-05-03 上药东英（江苏）药业有限公司 一种培哚普利叔丁胺片及其粉末直压工艺

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Also Published As

Publication number Publication date
JP4948392B2 (ja) 2012-06-06
PL1729739T3 (pl) 2017-04-28
NO20064934L (no) 2006-10-27
DK1729739T3 (en) 2016-10-31
LT1729739T (lt) 2016-11-10
ES2603856T3 (es) 2017-03-01
EA011712B1 (ru) 2009-04-28
US20070172524A1 (en) 2007-07-26
US20100172995A1 (en) 2010-07-08
EP1729739B1 (en) 2016-09-28
HRP20161602T1 (hr) 2016-12-30
HUE031058T2 (en) 2017-06-28
WO2005094793A1 (en) 2005-10-13
PT1729739T (pt) 2016-12-01
JP2007530623A (ja) 2007-11-01
CY1118180T1 (el) 2017-06-28
EP1729739A1 (en) 2006-12-13

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MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU