ATE531697T1 - Neuartige imidazolinylmethyl-aryl-sulfonamide - Google Patents
Neuartige imidazolinylmethyl-aryl-sulfonamideInfo
- Publication number
- ATE531697T1 ATE531697T1 AT09708902T AT09708902T ATE531697T1 AT E531697 T1 ATE531697 T1 AT E531697T1 AT 09708902 T AT09708902 T AT 09708902T AT 09708902 T AT09708902 T AT 09708902T AT E531697 T1 ATE531697 T1 AT E531697T1
- Authority
- AT
- Austria
- Prior art keywords
- novel
- methyl aryl
- aryl sulfonamides
- imidazolinyl
- imidazolinyl methyl
- Prior art date
Links
- -1 IMIDAZOLINYL METHYL Chemical class 0.000 title 1
- 229940124530 sulfonamide Drugs 0.000 title 1
- 150000003456 sulfonamides Chemical class 0.000 title 1
- 239000003814 drug Substances 0.000 abstract 1
- 239000004031 partial agonist Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
- 229940124597 therapeutic agent Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D233/24—Radicals substituted by nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2583608P | 2008-02-04 | 2008-02-04 | |
| PCT/EP2009/050837 WO2009098133A1 (en) | 2008-02-04 | 2009-01-26 | Novel imidazolinylmethyl aryl sulfonamides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE531697T1 true ATE531697T1 (de) | 2011-11-15 |
Family
ID=40456344
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT09708902T ATE531697T1 (de) | 2008-02-04 | 2009-01-26 | Neuartige imidazolinylmethyl-aryl-sulfonamide |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20090197933A1 (de) |
| EP (1) | EP2238115B1 (de) |
| JP (1) | JP2011511023A (de) |
| KR (1) | KR20100096266A (de) |
| CN (1) | CN101925579A (de) |
| AT (1) | ATE531697T1 (de) |
| AU (1) | AU2009211503A1 (de) |
| BR (1) | BRPI0907495A2 (de) |
| CA (1) | CA2711724A1 (de) |
| IL (1) | IL206763A0 (de) |
| MX (1) | MX2010008019A (de) |
| WO (1) | WO2009098133A1 (de) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2022047052A1 (en) * | 2020-08-27 | 2022-03-03 | Curasen Therapeutics, Inc. | α1A-ADRENERGIC RECEPTOR AGONISTS AND METHODS OF USE |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG72827A1 (en) * | 1997-06-23 | 2000-05-23 | Hoffmann La Roche | Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives |
| NZ535823A (en) * | 2002-04-23 | 2007-07-27 | Hoffmann La Roche | Imidazolin-2-ylmethyl substituted aralkylsulfonamides |
-
2009
- 2009-01-26 JP JP2010545427A patent/JP2011511023A/ja active Pending
- 2009-01-26 CN CN200980102956XA patent/CN101925579A/zh active Pending
- 2009-01-26 AT AT09708902T patent/ATE531697T1/de active
- 2009-01-26 BR BRPI0907495-3A patent/BRPI0907495A2/pt not_active IP Right Cessation
- 2009-01-26 AU AU2009211503A patent/AU2009211503A1/en not_active Abandoned
- 2009-01-26 MX MX2010008019A patent/MX2010008019A/es not_active Application Discontinuation
- 2009-01-26 KR KR1020107016883A patent/KR20100096266A/ko not_active Ceased
- 2009-01-26 WO PCT/EP2009/050837 patent/WO2009098133A1/en not_active Ceased
- 2009-01-26 EP EP09708902A patent/EP2238115B1/de not_active Not-in-force
- 2009-01-26 CA CA2711724A patent/CA2711724A1/en not_active Abandoned
- 2009-02-04 US US12/365,268 patent/US20090197933A1/en not_active Abandoned
-
2010
- 2010-07-01 IL IL206763A patent/IL206763A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP2238115B1 (de) | 2011-11-02 |
| EP2238115A1 (de) | 2010-10-13 |
| CA2711724A1 (en) | 2009-08-13 |
| BRPI0907495A2 (pt) | 2019-02-26 |
| US20090197933A1 (en) | 2009-08-06 |
| WO2009098133A1 (en) | 2009-08-13 |
| MX2010008019A (es) | 2010-08-10 |
| AU2009211503A1 (en) | 2009-08-13 |
| JP2011511023A (ja) | 2011-04-07 |
| CN101925579A (zh) | 2010-12-22 |
| IL206763A0 (en) | 2010-12-30 |
| KR20100096266A (ko) | 2010-09-01 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EA201390908A1 (ru) | Производные бицикло[3.2.1]октиламида и их применение | |
| MX390264B (es) | Antagonistas d2, metodos de sintesis y metodos de uso. | |
| EA201001724A1 (ru) | Производные изоксазола и их применение в качестве потенциирующих средств для метаботропных глутаматных рецепторов | |
| ATE517882T1 (de) | Chinolinderivate | |
| EA201390766A1 (ru) | БЕНЗОКСАЗЕПИНЫ КАК ИНГИБИТОРЫ PI3K/mTOR И СПОСОБЫ ИХ ИСПОЛЬЗОВАНИЯ И ПОЛУЧЕНИЯ | |
| NO20072978L (no) | Nye betuinderivater, preparat derav og anvendelse derav | |
| GEP20146146B (en) | Pyrrolopyrimidine compounds as inhibitors of cdk4/6 | |
| CY1119357T1 (el) | Φαρμακευτικες συνθεσεις που περιλαμβανουν συνδετες υποδοχεων σιγμα | |
| UA112317C2 (uk) | Похідні 2-(1,2,3-триазол-2-іл)бензаміду та 3-(1,2,3-триазол-2-іл)піколінаміду як антагоністи рецептора орексину | |
| DE602006006712D1 (de) | Thiazolylpiperidin-derivate nützlich als h3 rezeptor modulatoren | |
| EA200970341A1 (ru) | Пиразолиновые соединения в качестве антагонистов минералокортикоидных рецепторов | |
| EA201291217A1 (ru) | ФАРМАЦЕВТИЧЕСКИЕ КОМПОЗИЦИИ, СОДЕРЖАЩИЕ ПРОИЗВОДНЫЕ 1-(β-D-ГЛЮКОПИРАНОЗИЛ)-2-ТИЕНИЛМЕТИЛБЕНЗОЛА КАК ИНГИБИТОРЫ НЗПГ | |
| EA201390163A1 (ru) | Гетеробициклические производные в качетстве ингибиторов hcv | |
| UA109290C2 (uk) | Спільні кристали і солі інгібіторів ccr3 | |
| ATE552246T1 (de) | Substituierte aryloxy-n- bicyclomethylacetamidverbindungen als vr1- antagonisten | |
| EA201391524A1 (ru) | Производные гликозида и их применение | |
| EA201001566A1 (ru) | Новый класс спиропиперидинов для лечения нейродегенеративных заболеваний | |
| MA32479B1 (fr) | Compoés nouveaux actifs comme antagonistes des recepteurs muscariniques | |
| EA200901030A1 (ru) | Антагонист хроменового рецептора s1p1 | |
| ATE495159T1 (de) | Diaminocyclohexan- und diaminocyclopentanderivate | |
| EA201290534A1 (ru) | Бициклические тиазолы в качестве аллостерических модуляторов mglur5 рецепторов | |
| EA201270556A1 (ru) | Конденсированные тиазоло и оксазолопиримидиноны | |
| ATE525360T1 (de) | Neuartige imidazolinylmethyl-aryl-sulfonamide | |
| ATE546448T1 (de) | Urotensin-ii-rezeptorantagonisten | |
| EA201390488A1 (ru) | Новые агонисты gpr 119 |