UA83416C2 - Fused ring 4-oxopyrimidine derivative - Google Patents

Fused ring 4-oxopyrimidine derivative Download PDF

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UA83416C2
UA83416C2 UAA200609795A UAA200609795A UA83416C2 UA 83416 C2 UA83416 C2 UA 83416C2 UA A200609795 A UAA200609795 A UA A200609795A UA A200609795 A UAA200609795 A UA A200609795A UA 83416 C2 UA83416 C2 UA 83416C2
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aai
iabev
aza
oaize
iavev
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Тсуеси Нагасе
Нагааки САТО
Акио Канатани
Сигеру ТОКИТА
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Баниу Фармасьютикал Ко., Лтд.
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Abstract

Данное изобретение представляет соединение формулы (І), представленной ниже, или ее фармацевтически приемлемую соль, которая, имея активность антагониста или обратного агониста гистаминного рецептора Н3, является полезной для профилактики или лечения заболеваний обмена веществ, заболеваний системы кровообращения или заболеваний нервной системы,(I),где, например, Аr представляет собой бивалентную группу, образованную удалением двух атомов водорода из бензола, Xпредставляет собой атом азота, атом серы или атом кислорода, Rпредставляет собой 5-6-членную гетероарильную группу, кольцо А представляет собой 5-6- членное гетероарильное кольцо, Rи Rпредставляют собой аминогруппы или алкиламиногруппы, и Xпредставлен формулой (II)(II)(где Rи Rпредставляют собой низшие алкильные группы, и n представляет собой целое число, которое имеет значение от 2 до 4).
UAA200609795A 2004-02-13 2005-02-14 Fused ring 4-oxopyrimidine derivative UA83416C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2004037190 2004-02-13
PCT/JP2005/002664 WO2005077905A1 (ja) 2004-02-13 2005-02-14 縮環４－オキソ－ピリミジン誘導体

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UA83416C2 true UA83416C2 (en) 2008-07-10

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UAA200609795A UA83416C2 (en) 2004-02-13 2005-02-14 Fused ring 4-oxopyrimidine derivative

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US (2) US7521455B2 (ru)
EP (1) EP1717230B1 (ru)
JP (2) JP4102939B2 (ru)
KR (1) KR20070026385A (ru)
CN (1) CN1918128B (ru)
AU (1) AU2005212092B2 (ru)
BR (1) BRPI0507629A (ru)
CA (1) CA2555824C (ru)
EC (1) ECSP066760A (ru)
IL (1) IL177314A0 (ru)
MA (1) MA28463B1 (ru)
NO (1) NO20064089L (ru)
NZ (1) NZ549046A (ru)
RU (1) RU2358969C2 (ru)
UA (1) UA83416C2 (ru)
WO (1) WO2005077905A1 (ru)
ZA (1) ZA200606356B (ru)

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CA2569081A1 (en) * 2004-05-31 2005-12-08 Takashi Mizutani Quinazoline derivative
GB0412769D0 (en) 2004-06-08 2004-07-07 Novartis Ag Organic compounds
US9512125B2 (en) 2004-11-19 2016-12-06 The Regents Of The University Of California Substituted pyrazolo[3.4-D] pyrimidines as anti-inflammatory agents
WO2006085692A1 (ja) * 2005-02-14 2006-08-17 Banyu Pharmaceutical Co., Ltd ４（３ｈ）－キナゾリノン誘導体の結晶
EP1717235A3 (en) * 2005-04-29 2007-02-28 Bioprojet Phenoxypropylpiperidines and -pyrrolidines and their use as histamine H3-receptor ligands
EP1892241B1 (en) 2005-05-30 2016-03-30 Msd K.K. Novel piperidine derivative
EP1900733A4 (en) * 2005-06-07 2009-12-30 Banyu Pharma Co Ltd PROCESS FOR THE PRODUCTION OF 4 (3H) -QUINAZOLINONE DERIVATIVE
EP1903040A4 (en) * 2005-07-05 2010-08-04 Banyu Pharma Co Ltd PROCESS FOR PRODUCING 4 (3H) -QUINAZOLINONE DERIVATIVE
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