UA79782C2 - [1,4]diazepino[6,7,1-ij]quinoline derivatives as anti psychotic and antiobesity agents - Google Patents
[1,4]diazepino[6,7,1-ij]quinoline derivatives as anti psychotic and antiobesity agents Download PDFInfo
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- UA79782C2 UA79782C2 UA20041109666A UA20041109666A UA79782C2 UA 79782 C2 UA79782 C2 UA 79782C2 UA 20041109666 A UA20041109666 A UA 20041109666A UA 20041109666 A UA20041109666 A UA 20041109666A UA 79782 C2 UA79782 C2 UA 79782C2
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Classifications
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-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/22—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains four or more hetero rings
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US37559202P | 2002-04-25 | 2002-04-25 | |
| PCT/US2003/012747 WO2003091250A1 (en) | 2002-04-25 | 2003-04-24 | [1,4]diazepino[6,7,1-ij]quinoline derivatives as anti psychotic and antiobesity agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA79782C2 true UA79782C2 (en) | 2007-07-25 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| UA20041109666A UA79782C2 (en) | 2002-04-25 | 2003-04-24 | [1,4]diazepino[6,7,1-ij]quinoline derivatives as anti psychotic and antiobesity agents |
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|---|---|
| US (2) | US7129237B2 (es) |
| EP (1) | EP1497293B1 (es) |
| JP (1) | JP4537075B2 (es) |
| KR (1) | KR101009269B1 (es) |
| CN (2) | CN100376575C (es) |
| AR (1) | AR039669A1 (es) |
| AT (1) | ATE398127T1 (es) |
| AU (1) | AU2003234213C1 (es) |
| BR (1) | BR0309664A (es) |
| CA (1) | CA2481321C (es) |
| CR (1) | CR7510A (es) |
| CY (1) | CY1108286T1 (es) |
| DE (1) | DE60321559D1 (es) |
| DK (1) | DK1497293T3 (es) |
| EC (1) | ECSP045379A (es) |
| ES (1) | ES2307937T3 (es) |
| HK (1) | HK1069388A1 (es) |
| IL (1) | IL164806A0 (es) |
| MX (1) | MXPA04010372A (es) |
| NO (1) | NO329505B1 (es) |
| NZ (1) | NZ536115A (es) |
| PT (1) | PT1497293E (es) |
| RU (1) | RU2312866C2 (es) |
| SI (1) | SI1497293T1 (es) |
| TW (1) | TWI312781B (es) |
| UA (1) | UA79782C2 (es) |
| WO (1) | WO2003091250A1 (es) |
| ZA (1) | ZA200409501B (es) |
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| TW200307682A (en) | 2002-04-25 | 2003-12-16 | Wyeth Corp | 1,2,3,4,7,8-Hexahydro-6H-[1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents |
| TW200307540A (en) | 2002-04-25 | 2003-12-16 | Wyeth Corp | [1, 4]Diazocino[7, 8, 1-hi] indole derivatives as antipsychotic and antiobesity agents |
| GB0306604D0 (en) * | 2003-03-21 | 2003-04-30 | Curidium Ltd | Second medical use |
| EP2248524A3 (en) | 2004-08-25 | 2011-03-09 | Takeda Pharmaceutical Company Limited | Preventives/remedies for stress urinary incontinence and method of screening the same |
| AR051946A1 (es) * | 2004-11-05 | 2007-02-21 | Wyeth Corp | Formulaciones de derivados de [1,4] diazepina [6,7,1-ij] quinolina |
| GT200500317A (es) * | 2004-11-05 | 2006-10-27 | Proceso para preparar compuestos de quinolina y productos obtenidos de los mismos | |
| TW200635926A (en) * | 2004-11-05 | 2006-10-16 | Wyeth Corp | Metabolites of ceratin [1,4]diazepino[6,7,1-ij]quinoline derivatives and methods of preparation and use thereof |
| US7576222B2 (en) | 2004-12-28 | 2009-08-18 | Wyeth | Alkynyl-containing tryptophan derivative inhibitors of TACE/matrix metalloproteinase |
| AR054849A1 (es) * | 2005-07-26 | 2007-07-18 | Wyeth Corp | Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas |
| WO2007025144A1 (en) * | 2005-08-24 | 2007-03-01 | University Of Illinois - Chicago | 5-ht2c receptor agonists as anorectic agents |
| AR056695A1 (es) * | 2005-10-17 | 2007-10-17 | Wyeth Corp | Tetrahidroquinolinas, su sintesis e intermediarios |
| TW200734334A (en) * | 2006-01-13 | 2007-09-16 | Wyeth Corp | Treatment of substance abuse |
| AR060324A1 (es) * | 2006-03-24 | 2008-06-11 | Wyeth Corp | Metodos para modular la funcion de la vejiga |
| CL2007000773A1 (es) * | 2006-03-24 | 2008-01-25 | Wyeth Corp | Uso de compuestos derivados de diazepina condensada para el tratamiento de un desorden cognitivo como add o adhd;o su uso para tratar spm o pmdd. |
| US20070238725A1 (en) * | 2006-03-24 | 2007-10-11 | Wyeth | Therapeutic combinations for the treatment or prevention of psychotic disorders |
| AU2007231011A1 (en) * | 2006-03-24 | 2007-10-04 | Wyeth | New therapeutic combinations for the treatment of depression |
| PE20081192A1 (es) * | 2006-03-24 | 2008-10-07 | Wyeth Corp | Tratamiento del dolor |
| US8158617B2 (en) | 2006-05-16 | 2012-04-17 | Takeda Pharmaceutical Company Limited | Fused heterocyclic compound and use thereof |
| EP2162135A4 (en) * | 2007-05-21 | 2012-02-22 | Reviva Pharmaceuticals Inc | COMPOSITIONS, SYNTHESIS AND METHOD FOR THE APPLICATION OF ATTAINED CHINOLINONE-BASED ANTIPSYCHOTICS |
| WO2008144981A1 (fr) * | 2007-05-25 | 2008-12-04 | Topharman Shanghai Co., Ltd. | Procédés et intermédiaires pour préparer une 4-acétyl-2,3,4,5-tétrahydro-1h-1,4-benzodiazépine |
| CL2008002777A1 (es) * | 2007-09-21 | 2010-01-22 | Wyeth Corp | Metodo de preparacion de compuestos diazepinoquinolinicos quirales por recristalizacion en un sistema de solvente ternario. |
| JP5520051B2 (ja) | 2007-11-15 | 2014-06-11 | 武田薬品工業株式会社 | 縮合ピリジン誘導体およびその用途 |
| JPWO2011071136A1 (ja) | 2009-12-11 | 2013-04-22 | アステラス製薬株式会社 | 線維筋痛症治療剤 |
| US20130267500A1 (en) | 2010-09-01 | 2013-10-10 | Arena Pharmaceuticals, Inc. | 5-ht2c receptor agonists in the treatment of disorders ameliorated by reduction of norepinephrine level |
| WO2013133325A1 (ja) * | 2012-03-06 | 2013-09-12 | 武田薬品工業株式会社 | 三環性化合物 |
| US20140080813A1 (en) | 2012-09-14 | 2014-03-20 | AbbVie Deutschland GmbH & Co. KG | Tricyclic quinoline and quinoxaline derivatives |
| AU2013314279B2 (en) * | 2012-09-14 | 2017-11-02 | AbbVie Deutschland GmbH & Co. KG | Tricyclic quinoline and quinoxaline derivatives |
| WO2015066344A1 (en) | 2013-11-01 | 2015-05-07 | Arena Pharmaceuticals, Inc. | 5-ht2c receptor agonists and compositions and methods of use |
| US9573950B2 (en) | 2014-03-14 | 2017-02-21 | Abbvie Deutschland Gmbh & Co Kg | Substituted [1,4]diazepino[6,7,1-ij]quinolines as serotonin 5-HT2C receptor modulators |
| WO2015136091A1 (en) | 2014-03-14 | 2015-09-17 | AbbVie Deutschland GmbH & Co. KG | Hexahydrodiazepinoquinolines carrying a substituted alkyl radical |
| JPWO2019131902A1 (ja) | 2017-12-27 | 2020-12-10 | 武田薬品工業株式会社 | 腹圧性尿失禁および便失禁の治療薬 |
| US11753419B2 (en) | 2019-12-11 | 2023-09-12 | Intra-Cellular Therapies, Inc. | 4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)phenyl)butan-1-one for treating conditions of the central nervous system and cardiac disorders |
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- 2003-04-22 TW TW092109349A patent/TWI312781B/zh not_active IP Right Cessation
- 2003-04-24 RU RU2004134361/04A patent/RU2312866C2/ru not_active IP Right Cessation
- 2003-04-24 AT AT03728523T patent/ATE398127T1/de active
- 2003-04-24 UA UA20041109666A patent/UA79782C2/uk unknown
- 2003-04-24 DE DE60321559T patent/DE60321559D1/de not_active Expired - Lifetime
- 2003-04-24 AU AU2003234213A patent/AU2003234213C1/en not_active Ceased
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- 2003-04-24 CN CNB038143380A patent/CN100376575C/zh not_active Expired - Fee Related
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- 2003-04-24 BR BR0309664-5A patent/BR0309664A/pt not_active IP Right Cessation
- 2003-04-24 WO PCT/US2003/012747 patent/WO2003091250A1/en active Application Filing
- 2003-04-24 KR KR1020047017062A patent/KR101009269B1/ko not_active IP Right Cessation
- 2003-04-24 IL IL16480603A patent/IL164806A0/xx not_active IP Right Cessation
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- 2003-04-24 AR ARP030101430A patent/AR039669A1/es not_active Application Discontinuation
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- 2003-04-24 CN CN2006101464653A patent/CN1955179B/zh not_active Expired - Fee Related
- 2003-04-24 SI SI200331291T patent/SI1497293T1/sl unknown
- 2003-04-24 DK DK03728523T patent/DK1497293T3/da active
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2004
- 2004-10-06 CR CR7510A patent/CR7510A/es unknown
- 2004-10-21 NO NO20044501A patent/NO329505B1/no not_active IP Right Cessation
- 2004-10-22 EC EC2004005379A patent/ECSP045379A/es unknown
- 2004-11-24 ZA ZA200409501A patent/ZA200409501B/xx unknown
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2005
- 2005-03-08 HK HK05101986A patent/HK1069388A1/xx not_active IP Right Cessation
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2006
- 2006-09-11 US US11/518,216 patent/US7687620B2/en not_active Expired - Fee Related
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2008
- 2008-08-25 CY CY20081100902T patent/CY1108286T1/el unknown
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