ZA200409501B - [1,4]Diazepino[6,7,1,-ij]quinoline derivatives as antipsychotic and antiobesity agents - Google Patents

[1,4]Diazepino[6,7,1,-ij]quinoline derivatives as antipsychotic and antiobesity agents

Info

Publication number
ZA200409501B
ZA200409501B ZA200409501A ZA200409501A ZA200409501B ZA 200409501 B ZA200409501 B ZA 200409501B ZA 200409501 A ZA200409501 A ZA 200409501A ZA 200409501 A ZA200409501 A ZA 200409501A ZA 200409501 B ZA200409501 B ZA 200409501B
Authority
ZA
South Africa
Prior art keywords
diazepino
antipsychotic
quinoline derivatives
antiobesity agents
antiobesity
Prior art date
Application number
ZA200409501A
Other languages
English (en)
Inventor
Sivaramakrishnan P Ramamoorthy
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of ZA200409501B publication Critical patent/ZA200409501B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/22—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains four or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Anesthesiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA200409501A 2002-04-25 2004-11-24 [1,4]Diazepino[6,7,1,-ij]quinoline derivatives as antipsychotic and antiobesity agents ZA200409501B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US37559202P 2002-04-25 2002-04-25

Publications (1)

Publication Number Publication Date
ZA200409501B true ZA200409501B (en) 2007-04-25

Family

ID=29270669

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200409501A ZA200409501B (en) 2002-04-25 2004-11-24 [1,4]Diazepino[6,7,1,-ij]quinoline derivatives as antipsychotic and antiobesity agents

Country Status (28)

Country Link
US (2) US7129237B2 (xx)
EP (1) EP1497293B1 (xx)
JP (1) JP4537075B2 (xx)
KR (1) KR101009269B1 (xx)
CN (2) CN1955179B (xx)
AR (1) AR039669A1 (xx)
AT (1) ATE398127T1 (xx)
AU (1) AU2003234213C1 (xx)
BR (1) BR0309664A (xx)
CA (1) CA2481321C (xx)
CR (1) CR7510A (xx)
CY (1) CY1108286T1 (xx)
DE (1) DE60321559D1 (xx)
DK (1) DK1497293T3 (xx)
EC (1) ECSP045379A (xx)
ES (1) ES2307937T3 (xx)
HK (1) HK1069388A1 (xx)
IL (1) IL164806A0 (xx)
MX (1) MXPA04010372A (xx)
NO (1) NO329505B1 (xx)
NZ (1) NZ536115A (xx)
PT (1) PT1497293E (xx)
RU (1) RU2312866C2 (xx)
SI (1) SI1497293T1 (xx)
TW (1) TWI312781B (xx)
UA (1) UA79782C2 (xx)
WO (1) WO2003091250A1 (xx)
ZA (1) ZA200409501B (xx)

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Also Published As

Publication number Publication date
AU2003234213B2 (en) 2009-11-12
MXPA04010372A (es) 2005-02-03
US7129237B2 (en) 2006-10-31
US7687620B2 (en) 2010-03-30
TW200400038A (en) 2004-01-01
NO20044501L (no) 2005-01-18
CA2481321C (en) 2012-01-03
SI1497293T1 (sl) 2008-10-31
RU2312866C2 (ru) 2007-12-20
CR7510A (es) 2008-07-29
ECSP045379A (es) 2004-11-26
KR101009269B1 (ko) 2011-01-18
CN1955179B (zh) 2010-07-14
CN1662533A (zh) 2005-08-31
CY1108286T1 (el) 2014-02-12
CN100376575C (zh) 2008-03-26
DK1497293T3 (da) 2008-09-15
DE60321559D1 (de) 2008-07-24
JP2005529893A (ja) 2005-10-06
JP4537075B2 (ja) 2010-09-01
NO329505B1 (no) 2010-11-01
UA79782C2 (en) 2007-07-25
AU2003234213C1 (en) 2010-05-20
KR20050000405A (ko) 2005-01-03
EP1497293A1 (en) 2005-01-19
HK1069388A1 (en) 2005-05-20
CN1955179A (zh) 2007-05-02
ATE398127T1 (de) 2008-07-15
US20040009970A1 (en) 2004-01-15
TWI312781B (en) 2009-08-01
US20070004707A1 (en) 2007-01-04
CA2481321A1 (en) 2003-11-06
NZ536115A (en) 2007-11-30
PT1497293E (pt) 2008-09-05
EP1497293B1 (en) 2008-06-11
AR039669A1 (es) 2005-03-02
ES2307937T3 (es) 2008-12-01
AU2003234213A1 (en) 2003-11-10
RU2004134361A (ru) 2005-05-10
BR0309664A (pt) 2005-02-22
IL164806A0 (en) 2005-12-18
WO2003091250A1 (en) 2003-11-06

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