TW200823227A - 3-aza-bicyclo[3.1.0]hexane derivatives - Google Patents

3-aza-bicyclo[3.1.0]hexane derivatives Download PDF

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Publication number
TW200823227A
TW200823227A TW096136490A TW96136490A TW200823227A TW 200823227 A TW200823227 A TW 200823227A TW 096136490 A TW096136490 A TW 096136490A TW 96136490 A TW96136490 A TW 96136490A TW 200823227 A TW200823227 A TW 200823227A
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TW
Taiwan
Prior art keywords
bicyclo
methyl
hex
carboxylic acid
nitro
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TW096136490A
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English (en)
Chinese (zh)
Inventor
Hamed Aissaoui
Christoph Boss
Markus Gude
Ralf Koberstein
David Lehmann
Thierry Sifferlen
Daniel Trachsel
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Actelion Pharmaceuticals Ltd
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Publication of TW200823227A publication Critical patent/TW200823227A/zh

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  • Diabetes (AREA)
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TW096136490A 2006-09-29 2007-09-28 3-aza-bicyclo[3.1.0]hexane derivatives TW200823227A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IB2006053570 2006-09-29

Publications (1)

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TW200823227A true TW200823227A (en) 2008-06-01

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TW096136490A TW200823227A (en) 2006-09-29 2007-09-28 3-aza-bicyclo[3.1.0]hexane derivatives

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Country Link
US (1) US20100016401A1 (OSRAM)
EP (1) EP2079690B1 (OSRAM)
JP (1) JP2010504957A (OSRAM)
KR (1) KR20090077051A (OSRAM)
CN (1) CN101522618A (OSRAM)
AR (1) AR063081A1 (OSRAM)
AT (1) ATE481383T1 (OSRAM)
CA (1) CA2662612A1 (OSRAM)
CL (1) CL2007002809A1 (OSRAM)
DE (1) DE602007009284D1 (OSRAM)
ES (1) ES2350460T3 (OSRAM)
TW (1) TW200823227A (OSRAM)
WO (1) WO2008038251A2 (OSRAM)

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CL2008000836A1 (es) * 2007-03-26 2008-11-07 Actelion Pharmaceuticals Ltd Compuestos derivados de tiazolidina, antagonistas del receptor de orexina; composicion farmaceutica que los comprende; y su uso en el tratamiento de neurosis emocional, depresion grave, trastornos psicoticos, alzheimer, parkinson, dolor, entre otras.
ES2379744T3 (es) 2007-05-23 2012-05-03 Merck Sharp & Dohme Corp. Antagonistas de piridil-piperidina de los receptores de orexinas
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KR20100046047A (ko) * 2007-07-27 2010-05-04 액테리온 파마슈티칼 리미티드 2-아자-비시클로[3.3.0]옥탄 유도체
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KR20120007061A (ko) 2009-04-24 2012-01-19 글락소 그룹 리미티드 오렉신 길항제로서 사용되는 3-아자비시클로［4.1.0］헵탄
EP2275421A1 (en) * 2009-07-15 2011-01-19 Rottapharm S.p.A. Spiro amino compounds suitable for the treatment of inter alia sleep disorders and drug addiction
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