TNSN97135A1 - Derives 6,6- ou 6,7 bicycliques a noyau pyrido ou pyrimido substitues - Google Patents

Derives 6,6- ou 6,7 bicycliques a noyau pyrido ou pyrimido substitues

Info

Publication number
TNSN97135A1
TNSN97135A1 TNTNSN97135A TNSN97135A TNSN97135A1 TN SN97135 A1 TNSN97135 A1 TN SN97135A1 TN TNSN97135 A TNTNSN97135 A TN TNSN97135A TN SN97135 A TNSN97135 A TN SN97135A TN SN97135 A1 TNSN97135 A1 TN SN97135A1
Authority
TN
Tunisia
Prior art keywords
pyrimido
pyrido
bicyclic derivatives
cores
substituted
Prior art date
Application number
TNTNSN97135A
Other languages
English (en)
Inventor
Liang Chen Yuhpyng
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of TNSN97135A1 publication Critical patent/TNSN97135A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones

Abstract

L'INVENTION CONCERNE DES PYRAZOLES PARASITICIDES NOUVEAUX DE FORMULE I .............................DANS LAQUELLE A, B, D, E, K, G, Z, R3 ET R5 REPRESENTENT DIVERS ATOMES OU RADICAUX . ELLE CONCERNE EGALEMENT UN PROCEDE POUR LEUR PREPARATION ET DES COMPOSITIONS PHARMACEUTIQUEMENT LES CONTENANT. APPLICATION: UTILISATION DE CES COMPOSES ET COMPOSITIONS POUR LE TRAITEMENT DE MALADIES QUI PEUT ETRE EFFECTUE OU FACILITE PAR ANTAGONISATION DU FACTEUR DE LIBERATION DE CORTICOTROPHINE
TNTNSN97135A 1996-08-06 1997-08-06 Derives 6,6- ou 6,7 bicycliques a noyau pyrido ou pyrimido substitues TNSN97135A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2345396P 1996-08-06 1996-08-06

Publications (1)

Publication Number Publication Date
TNSN97135A1 true TNSN97135A1 (fr) 2005-03-15

Family

ID=21815208

Family Applications (1)

Application Number Title Priority Date Filing Date
TNTNSN97135A TNSN97135A1 (fr) 1996-08-06 1997-08-06 Derives 6,6- ou 6,7 bicycliques a noyau pyrido ou pyrimido substitues

Country Status (41)

Country Link
US (1) US6492520B1 (fr)
EP (1) EP0920429B1 (fr)
JP (1) JP3345021B2 (fr)
KR (1) KR20000029843A (fr)
CN (1) CN1093130C (fr)
AP (1) AP1096A (fr)
AR (1) AR008829A1 (fr)
AT (1) ATE232863T1 (fr)
AU (1) AU709203B2 (fr)
BG (1) BG103143A (fr)
BR (1) BR9710808A (fr)
CA (1) CA2262692C (fr)
CO (1) CO4900060A1 (fr)
CZ (1) CZ292806B6 (fr)
DE (1) DE69719193T2 (fr)
DK (1) DK0920429T3 (fr)
DZ (1) DZ2289A1 (fr)
EA (1) EA003188B1 (fr)
ES (1) ES2191183T3 (fr)
GT (1) GT199700089A (fr)
HK (1) HK1021734A1 (fr)
HR (1) HRP970432B1 (fr)
ID (1) ID17980A (fr)
IL (1) IL128188A0 (fr)
IS (1) IS4948A (fr)
MA (1) MA24296A1 (fr)
NO (1) NO313293B1 (fr)
NZ (1) NZ333727A (fr)
OA (1) OA10970A (fr)
PA (1) PA8435201A1 (fr)
PE (1) PE97098A1 (fr)
PL (1) PL331602A1 (fr)
SA (1) SA97180334A (fr)
SK (1) SK14099A3 (fr)
TN (1) TNSN97135A1 (fr)
TR (1) TR199900228T2 (fr)
TW (1) TW550265B (fr)
UY (1) UY24655A1 (fr)
WO (1) WO1998005661A1 (fr)
YU (1) YU5399A (fr)
ZA (1) ZA976954B (fr)

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Also Published As

Publication number Publication date
ATE232863T1 (de) 2003-03-15
NO313293B1 (no) 2002-09-09
AP1096A (en) 2002-08-26
AP9701052A0 (en) 1997-10-31
CZ292806B6 (cs) 2003-12-17
WO1998005661A1 (fr) 1998-02-12
NO990544D0 (no) 1999-02-05
HRP970432B1 (en) 2002-10-31
CN1227552A (zh) 1999-09-01
MA24296A1 (fr) 1998-04-01
DE69719193D1 (de) 2003-03-27
EA003188B1 (ru) 2003-02-27
TR199900228T2 (xx) 1999-03-22
CA2262692A1 (fr) 1998-02-12
IL128188A0 (en) 1999-11-30
AU3356397A (en) 1998-02-25
NZ333727A (en) 2000-09-29
UY24655A1 (es) 2000-09-29
AR008829A1 (es) 2000-02-23
KR20000029843A (ko) 2000-05-25
TW550265B (en) 2003-09-01
HK1021734A1 (en) 2000-06-30
YU5399A (sh) 2002-03-18
SK14099A3 (en) 2000-05-16
GT199700089A (es) 1999-01-26
IS4948A (is) 1999-01-19
CA2262692C (fr) 2002-06-11
DZ2289A1 (fr) 2002-12-25
CZ41199A3 (cs) 2000-01-12
DE69719193T2 (de) 2003-09-25
JP3345021B2 (ja) 2002-11-18
CN1093130C (zh) 2002-10-23
HRP970432A2 (en) 1998-08-31
PE97098A1 (es) 1999-01-12
JP2000501116A (ja) 2000-02-02
BR9710808A (pt) 1999-08-17
US6492520B1 (en) 2002-12-10
NO990544L (no) 1999-03-31
EP0920429A1 (fr) 1999-06-09
EA199900083A1 (ru) 1999-08-26
CO4900060A1 (es) 2000-03-27
EP0920429B1 (fr) 2003-02-19
BG103143A (en) 1999-09-30
ID17980A (id) 1998-02-12
AU709203B2 (en) 1999-08-26
DK0920429T3 (da) 2003-05-12
ES2191183T3 (es) 2003-09-01
ZA976954B (en) 1999-02-05
SA97180334A (ar) 2005-12-03
OA10970A (en) 2001-11-05
PA8435201A1 (es) 1999-12-27
PL331602A1 (en) 1999-08-02

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TNSN00028A1 (fr) Derives de quinoleine -2-one a substituant heteroaryle nouveaux procede pour leur preparation et compositions pharmaceutiques les contenant.
TNSN98238A1 (fr) Macrolides nouveaux
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TNSN97192A1 (fr) Derives de pyrimidine bicycliques condenses, procede pour leur preparation et compositions pharmaceutiques les contenant.
TNSN99156A1 (fr) Derives d'acide hydroxypipecolate-hydroxamique nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant
TNSN97108A1 (fr) Analogues d'indazole nouveaux
TNSN99169A1 (fr) Derives de 4,4-biarylpiperidine nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant
TNSN99142A1 (fr) Derives de benzimidazole nouveaux, compositions pharmaceutiques les contenant et procede pour leur preparation.
TNSN97198A1 (fr) Derives de 6-phenylpyridyl-2- amine et compositions pharmaceutiques les contenant
TNSN98022A1 (fr) DERIVES DE N-HYDROXY-β-SULFONYLPROPIONAMIDE, PROCEDE POUR LEUR PREPARATION ET COMPOSITIONS PHARMACEUTIQUES LES CONTENANT.
TNSN98019A1 (fr) Derives d'acide arylsulfonylaminohydroxamique, procede pour leur preparation et compositions pharmaceutiques les contenant.
TNSN97197A1 (fr) Derives de pyrazole parasiticides, procede pour leur preparation et compositions les contenant.
TNSN00104A1 (fr) Derives d'isothiazole nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant
TNSN98194A1 (fr) Derives nouveaux de 6-o-methylerythromycine a, procede pour leur preparation et compositions pharmaceutiques les contenant
TNSN99039A1 (fr) Bicyclo [2.2.1] heptanes nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant