ATE232863T1 - Substituierte pyrido- oder pyrimidogruppen enthaltende 6,6- oder 6,7-bicyclische derivate - Google Patents

Substituierte pyrido- oder pyrimidogruppen enthaltende 6,6- oder 6,7-bicyclische derivate

Info

Publication number
ATE232863T1
ATE232863T1 AT97929472T AT97929472T ATE232863T1 AT E232863 T1 ATE232863 T1 AT E232863T1 AT 97929472 T AT97929472 T AT 97929472T AT 97929472 T AT97929472 T AT 97929472T AT E232863 T1 ATE232863 T1 AT E232863T1
Authority
AT
Austria
Prior art keywords
pyrimido
groups
derivatives containing
containing substituted
substituted pyrido
Prior art date
Application number
AT97929472T
Other languages
English (en)
Inventor
Yuhpyng Liang Chen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE232863T1 publication Critical patent/ATE232863T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/02Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Communicable Diseases (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Hematology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Pain & Pain Management (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
AT97929472T 1996-08-06 1997-07-23 Substituierte pyrido- oder pyrimidogruppen enthaltende 6,6- oder 6,7-bicyclische derivate ATE232863T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2345396P 1996-08-06 1996-08-06
PCT/IB1997/000918 WO1998005661A1 (en) 1996-08-06 1997-07-23 Substituted pyrido- or pyrimido-containing 6,6- or 6,7-bicyclic derivatives

Publications (1)

Publication Number Publication Date
ATE232863T1 true ATE232863T1 (de) 2003-03-15

Family

ID=21815208

Family Applications (1)

Application Number Title Priority Date Filing Date
AT97929472T ATE232863T1 (de) 1996-08-06 1997-07-23 Substituierte pyrido- oder pyrimidogruppen enthaltende 6,6- oder 6,7-bicyclische derivate

Country Status (40)

Country Link
US (1) US6492520B1 (de)
EP (1) EP0920429B1 (de)
JP (1) JP3345021B2 (de)
KR (1) KR20000029843A (de)
CN (1) CN1093130C (de)
AP (1) AP1096A (de)
AR (1) AR008829A1 (de)
AT (1) ATE232863T1 (de)
AU (1) AU709203B2 (de)
BG (1) BG103143A (de)
BR (1) BR9710808A (de)
CA (1) CA2262692C (de)
CO (1) CO4900060A1 (de)
CZ (1) CZ292806B6 (de)
DE (1) DE69719193T2 (de)
DK (1) DK0920429T3 (de)
DZ (1) DZ2289A1 (de)
EA (1) EA003188B1 (de)
ES (1) ES2191183T3 (de)
GT (1) GT199700089A (de)
HR (1) HRP970432B1 (de)
ID (1) ID17980A (de)
IL (1) IL128188A0 (de)
IS (1) IS4948A (de)
MA (1) MA24296A1 (de)
NO (1) NO313293B1 (de)
NZ (1) NZ333727A (de)
OA (1) OA10970A (de)
PA (1) PA8435201A1 (de)
PE (1) PE97098A1 (de)
PL (1) PL331602A1 (de)
SA (1) SA97180334A (de)
SK (1) SK14099A3 (de)
TN (1) TNSN97135A1 (de)
TR (1) TR199900228T2 (de)
TW (1) TW550265B (de)
UY (1) UY24655A1 (de)
WO (1) WO1998005661A1 (de)
YU (1) YU5399A (de)
ZA (1) ZA976954B (de)

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Also Published As

Publication number Publication date
HK1021734A1 (en) 2000-06-30
EA199900083A1 (ru) 1999-08-26
CO4900060A1 (es) 2000-03-27
ZA976954B (en) 1999-02-05
AU709203B2 (en) 1999-08-26
DE69719193D1 (de) 2003-03-27
SK14099A3 (en) 2000-05-16
AR008829A1 (es) 2000-02-23
ES2191183T3 (es) 2003-09-01
CN1093130C (zh) 2002-10-23
EP0920429B1 (de) 2003-02-19
JP3345021B2 (ja) 2002-11-18
PE97098A1 (es) 1999-01-12
BR9710808A (pt) 1999-08-17
IL128188A0 (en) 1999-11-30
CN1227552A (zh) 1999-09-01
JP2000501116A (ja) 2000-02-02
HRP970432B1 (en) 2002-10-31
YU5399A (sh) 2002-03-18
MA24296A1 (fr) 1998-04-01
PL331602A1 (en) 1999-08-02
TR199900228T2 (xx) 1999-03-22
HRP970432A2 (en) 1998-08-31
BG103143A (en) 1999-09-30
CZ41199A3 (cs) 2000-01-12
UY24655A1 (es) 2000-09-29
NO990544D0 (no) 1999-02-05
CZ292806B6 (cs) 2003-12-17
KR20000029843A (ko) 2000-05-25
DK0920429T3 (da) 2003-05-12
CA2262692A1 (en) 1998-02-12
AU3356397A (en) 1998-02-25
US6492520B1 (en) 2002-12-10
NO313293B1 (no) 2002-09-09
TNSN97135A1 (fr) 2005-03-15
DE69719193T2 (de) 2003-09-25
NZ333727A (en) 2000-09-29
IS4948A (is) 1999-01-19
AP1096A (en) 2002-08-26
AP9701052A0 (en) 1997-10-31
TW550265B (en) 2003-09-01
EA003188B1 (ru) 2003-02-27
NO990544L (no) 1999-03-31
PA8435201A1 (es) 1999-12-27
ID17980A (id) 1998-02-12
DZ2289A1 (fr) 2002-12-25
GT199700089A (es) 1999-01-26
OA10970A (en) 2001-11-05
WO1998005661A1 (en) 1998-02-12
CA2262692C (en) 2002-06-11
EP0920429A1 (de) 1999-06-09
SA97180334A (ar) 2005-12-03

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