SG11201609550PA - 1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor - Google Patents

1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor

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Publication number
SG11201609550PA
SG11201609550PA SG11201609550PA SG11201609550PA SG11201609550PA SG 11201609550P A SG11201609550P A SG 11201609550PA SG 11201609550P A SG11201609550P A SG 11201609550PA SG 11201609550P A SG11201609550P A SG 11201609550PA SG 11201609550P A SG11201609550P A SG 11201609550PA
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Singapore
Prior art keywords
methylpyrimidin
pyrazol
pyrrolidin
methoxyethyl
fluorophenyl
Prior art date
Application number
SG11201609550PA
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English (en)
Inventor
Shelley Allen
Steven W Andrews
Brian Baer
Zackary Crane
Weidong Liu
Daniel John Watson
Original Assignee
Array Biopharma Inc
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Publication date
Application filed by Array Biopharma Inc filed Critical Array Biopharma Inc
Publication of SG11201609550PA publication Critical patent/SG11201609550PA/en

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SG11201609550PA 2014-05-15 2015-05-14 1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor SG11201609550PA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201461993426P 2014-05-15 2014-05-15
PCT/US2015/030795 WO2015175788A1 (en) 2014-05-15 2015-05-14 1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor

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SG11201609550PA true SG11201609550PA (en) 2016-12-29

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SG10201903532XA SG10201903532XA (en) 2014-05-15 2015-05-14 1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor

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