SG10201704858PA - Formulations and methods for vaginal delivery of antiprogestins - Google Patents

Formulations and methods for vaginal delivery of antiprogestins

Info

Publication number
SG10201704858PA
SG10201704858PA SG10201704858PA SG10201704858PA SG10201704858PA SG 10201704858P A SG10201704858P A SG 10201704858PA SG 10201704858P A SG10201704858P A SG 10201704858PA SG 10201704858P A SG10201704858P A SG 10201704858PA SG 10201704858P A SG10201704858P A SG 10201704858PA
Authority
SG
Singapore
Prior art keywords
antiprogestins
formulations
methods
vaginal delivery
vaginal
Prior art date
Application number
SG10201704858PA
Other languages
English (en)
Inventor
Joseph S Podolski
Kuang Hsu
Original Assignee
Repros Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48614182&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG10201704858P(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Repros Therapeutics Inc filed Critical Repros Therapeutics Inc
Publication of SG10201704858PA publication Critical patent/SG10201704858PA/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4816—Wall or shell material
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/02—Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
SG10201704858PA 2012-05-31 2013-05-30 Formulations and methods for vaginal delivery of antiprogestins SG10201704858PA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261653674P 2012-05-31 2012-05-31

Publications (1)

Publication Number Publication Date
SG10201704858PA true SG10201704858PA (en) 2017-07-28

Family

ID=48614182

Family Applications (2)

Application Number Title Priority Date Filing Date
SG10201704858PA SG10201704858PA (en) 2012-05-31 2013-05-30 Formulations and methods for vaginal delivery of antiprogestins
SG11201407397WA SG11201407397WA (en) 2012-05-31 2013-05-30 Formulations and methods for vaginal delivery of antiprogestins

Family Applications After (1)

Application Number Title Priority Date Filing Date
SG11201407397WA SG11201407397WA (en) 2012-05-31 2013-05-30 Formulations and methods for vaginal delivery of antiprogestins

Country Status (23)

Country Link
US (1) US10328022B2 (ko)
EP (1) EP2854763B1 (ko)
JP (1) JP6341910B2 (ko)
KR (1) KR102127348B1 (ko)
CN (1) CN104334158B (ko)
AU (1) AU2013267359C1 (ko)
BR (1) BR112014029131B1 (ko)
CA (1) CA2872644A1 (ko)
CL (1) CL2014003232A1 (ko)
CO (1) CO7141411A2 (ko)
CR (1) CR20140567A (ko)
EA (1) EA030444B1 (ko)
ES (1) ES2701400T3 (ko)
HK (1) HK1206622A1 (ko)
IL (1) IL235450B (ko)
IN (1) IN2014DN10548A (ko)
MX (2) MX363640B (ko)
NZ (1) NZ702467A (ko)
PH (1) PH12014502516A1 (ko)
SG (2) SG10201704858PA (ko)
UA (1) UA114106C2 (ko)
WO (1) WO2013181449A1 (ko)
ZA (1) ZA201408262B (ko)

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ES2885523T3 (es) 2011-11-23 2021-12-14 Therapeuticsmd Inc Formulaciones y terapias de reposición hormonal de combinación naturales
US9301920B2 (en) 2012-06-18 2016-04-05 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US20150196640A1 (en) 2012-06-18 2015-07-16 Therapeuticsmd, Inc. Progesterone formulations having a desirable pk profile
US20130338122A1 (en) 2012-06-18 2013-12-19 Therapeuticsmd, Inc. Transdermal hormone replacement therapies
US10806697B2 (en) 2012-12-21 2020-10-20 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10806740B2 (en) 2012-06-18 2020-10-20 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US10471072B2 (en) 2012-12-21 2019-11-12 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US11266661B2 (en) 2012-12-21 2022-03-08 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10568891B2 (en) 2012-12-21 2020-02-25 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US9180091B2 (en) 2012-12-21 2015-11-10 Therapeuticsmd, Inc. Soluble estradiol capsule for vaginal insertion
US10537581B2 (en) 2012-12-21 2020-01-21 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US11246875B2 (en) 2012-12-21 2022-02-15 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
CN111840246A (zh) 2014-05-05 2020-10-30 艾尔建制药国际有限公司 用于抗孕激素的阴道递送的制剂和方法
KR20170005819A (ko) 2014-05-22 2017-01-16 쎄러퓨틱스엠디, 인코퍼레이티드 천연 복합 호르몬 대체 제형 및 요법
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JP7222911B2 (ja) 2017-04-14 2023-02-15 カプスゲル・ベルギウム・ナムローゼ・フェンノートシャップ プルランを作製する方法

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Also Published As

Publication number Publication date
SG11201407397WA (en) 2014-12-30
EP2854763B1 (en) 2018-09-26
MX2019003467A (es) 2019-06-06
KR102127348B1 (ko) 2020-06-29
NZ702467A (en) 2016-07-29
EA030444B1 (ru) 2018-08-31
PH12014502516B1 (en) 2015-01-12
JP2015518052A (ja) 2015-06-25
PH12014502516A1 (en) 2015-01-12
CA2872644A1 (en) 2013-12-05
CN104334158B (zh) 2018-08-10
AU2013267359C1 (en) 2016-09-29
US20150111862A1 (en) 2015-04-23
AU2013267359B2 (en) 2016-05-26
CL2014003232A1 (es) 2015-03-13
MX2014014054A (es) 2015-02-12
ES2701400T3 (es) 2019-02-22
US10328022B2 (en) 2019-06-25
EP2854763A1 (en) 2015-04-08
IL235450B (en) 2020-02-27
KR20150014928A (ko) 2015-02-09
IN2014DN10548A (ko) 2015-08-21
IL235450A0 (en) 2014-12-31
CR20140567A (es) 2015-03-09
MX363640B (es) 2019-03-28
AU2013267359A1 (en) 2014-11-20
CN104334158A (zh) 2015-02-04
JP6341910B2 (ja) 2018-06-13
HK1206622A1 (en) 2016-01-15
WO2013181449A1 (en) 2013-12-05
EA201492290A1 (ru) 2015-03-31
CO7141411A2 (es) 2014-12-12
UA114106C2 (xx) 2017-04-25
BR112014029131A2 (pt) 2018-05-29
BR112014029131B1 (pt) 2021-03-09
ZA201408262B (en) 2015-12-23

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