SE9301916D0 - New peptides derivatives - Google Patents
New peptides derivativesInfo
- Publication number
- SE9301916D0 SE9301916D0 SE19939301916A SE9301916A SE9301916D0 SE 9301916 D0 SE9301916 D0 SE 9301916D0 SE 19939301916 A SE19939301916 A SE 19939301916A SE 9301916 A SE9301916 A SE 9301916A SE 9301916 D0 SE9301916 D0 SE 9301916D0
- Authority
- SE
- Sweden
- Prior art keywords
- new peptides
- peptides derivatives
- derivatives
- new
- therapy
- Prior art date
Links
- 102000004196 processed proteins & peptides Human genes 0.000 title 1
- 108090000765 processed proteins & peptides Proteins 0.000 title 1
- BSYNRYMUTXBXSQ-UHFFFAOYSA-N Aspirin Chemical compound CC(=O)OC1=CC=CC=C1C(O)=O BSYNRYMUTXBXSQ-UHFFFAOYSA-N 0.000 abstract 1
- 229960001138 acetylsalicylic acid Drugs 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D239/08—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
- C07D239/12—Nitrogen atoms not forming part of a nitro radical
- C07D239/14—Nitrogen atoms not forming part of a nitro radical with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to said nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/62—Compounds containing any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylcarbamates
- C07C271/64—Y being a hydrogen or a carbon atom, e.g. benzoylcarbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
- C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/26—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- C07K5/06165—Dipeptides with the first amino acid being heterocyclic and Pro-amino acid; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biochemistry (AREA)
- Pulmonology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Dermatology (AREA)
- Otolaryngology (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Psychiatry (AREA)
- Physical Education & Sports Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (59)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE19939301916A SE9301916D0 (sv) | 1993-06-03 | 1993-06-03 | New peptides derivatives |
UA95115078A UA65518C2 (en) | 1993-06-03 | 1994-02-06 | Peptide derivatives |
TW083104085A TW403731B (en) | 1993-06-03 | 1994-05-05 | New peptides derivatives |
IL123996A IL123996A (en) | 1993-06-03 | 1994-05-12 | Use of compounds as starting materials in synthesis of a serine protease inhibitor |
IL10963494A IL109634A (en) | 1993-06-03 | 1994-05-12 | Peptide derivatives their preparation and pharmaceutical compositions containing them |
IL12399594A IL123995A (en) | 1993-06-03 | 1994-05-12 | Peptide derivatives, their preparation and pharmaceutical compositions comprising them |
IS4166A IS1805B (is) | 1993-06-03 | 1994-05-16 | Aðferð til að framleiða nýjar peptíðafleiður sem eru þrombíntálmar |
HR940311A HRP940311B1 (en) | 1993-06-03 | 1994-05-17 | New peptide derivatives |
MX9404114A MX9404114A (es) | 1993-06-03 | 1994-06-01 | Nuevos derivados de peptidos. |
KR1019950705448A KR100339456B1 (ko) | 1993-06-03 | 1994-06-02 | 신규펩티드유도체 |
SG1996006171A SG48013A1 (en) | 1993-06-03 | 1994-06-02 | New peptide derivatives |
PL94311819A PL181968B1 (pl) | 1993-06-03 | 1994-06-02 | Nowe pochodne peptydowe, sposób wytwarzania pochodnych peptydowych oraz kompozycje farmaceutyczne zawierajace pochodne peptydowe PL |
AU69869/94A AU684086C (en) | 1993-06-03 | 1994-06-02 | New peptide derivatives |
PT94918636T PT701568E (pt) | 1993-06-03 | 1994-06-02 | Novos derivados de peptidos |
DK94918636T DK0701568T3 (da) | 1993-06-03 | 1994-06-02 | Nye peptidderivater |
EP94918636A EP0701568B1 (en) | 1993-06-03 | 1994-06-02 | New peptide derivatives |
DE69427150T DE69427150T2 (de) | 1993-06-03 | 1994-06-02 | Neuartige peptidderivate |
CA002162900A CA2162900C (en) | 1993-06-03 | 1994-06-02 | New peptide derivatives |
SK1454-95A SK283150B6 (sk) | 1993-06-03 | 1994-06-02 | Peptidové deriváty, spôsob ich prípravy, farmaceutický prípravok s ich obsahom a ich použitie |
MYPI94001423A MY119155A (en) | 1993-06-03 | 1994-06-02 | New peptide derivatives |
AT94918636T ATE200783T1 (de) | 1993-06-03 | 1994-06-02 | Neuartige peptidderivate |
JP50166595A JP3205558B2 (ja) | 1993-06-03 | 1994-06-02 | 新規ペプチド誘導体 |
PCT/SE1994/000535 WO1994029336A1 (en) | 1993-06-03 | 1994-06-02 | New peptide derivatives |
BR9406746A BR9406746A (pt) | 1993-06-03 | 1994-06-02 | Composto processo para sua preparaçao preparado farmacêutico uso de um composto processo para a obtençao da inibiçao de trombina em um organismo humano ou animale fragmento estrutural |
HU0103039A HU0103039D0 (en) | 1993-06-03 | 1994-06-02 | Use of para-amidinobenzylamine for the synthesis of peptide like serine protease inhibitors, and protected derivatives thereof |
HU9503445A HU226825B1 (en) | 1993-06-03 | 1994-06-02 | Peptide derivatives, process for prepearing them, pharmaceutical compositions containing them and use of them |
DE122004000045C DE122004000045I2 (de) | 1993-06-03 | 1994-06-02 | Neuartige peptidderivate |
EG32494A EG20671A (en) | 1993-06-03 | 1994-06-02 | New peptides derivatives |
DE0701568T DE701568T1 (de) | 1993-06-03 | 1994-06-02 | Neuartige peptidderivate |
SI9430365T SI0701568T1 (en) | 1993-06-03 | 1994-06-02 | New peptide derivatives |
CZ19953020A CZ290104B6 (cs) | 1993-06-03 | 1994-06-02 | Peptidový derivát, způsob jeho přípravy a použitía farmaceutický přípravek s jeho obsahem |
CN94192799A CN1099425C (zh) | 1993-06-03 | 1994-06-02 | 新的肽衍生物 |
EP00121659A EP1067136A1 (en) | 1993-06-03 | 1994-06-02 | New peptide derivatives |
RU96101161A RU2142469C1 (ru) | 1993-06-03 | 1994-06-02 | Пептидные производные, их стереоизомеры или физиологически приемлемые соли, обладающие противотромбозной, противосвертывающей или противовоспалительной активностью, способ их получения, фармацевтическая композиция, способ подавления тромбина, способ подавления кининогеназ, применение соединений в качестве исходных в синтезе ингибитора тромбина |
NZ267534A NZ267534A (en) | 1993-06-03 | 1994-06-02 | Trypsin-like serine protease inhibitors and compositions thereof, and precursor reagents |
ES94918636T ES2128277T3 (es) | 1993-06-03 | 1994-06-02 | Nuevos derivados de peptidos. |
LTIP1947A LT3768B (en) | 1993-06-03 | 1994-06-03 | Novel peptides derivatives, process for their preparation, pharmaceutical compositions and use starting materials in synthesis of a serine protease inhibitors |
YUP-336/94A RS49576B (sr) | 1993-06-03 | 1994-06-03 | Novi derivati peptida |
SA94150051A SA94150051B1 (ar) | 1993-06-03 | 1994-07-03 | مشتقات ببتيد جديدة |
EE9400456A EE03264B1 (et) | 1993-06-03 | 1994-11-23 | Peptiidi derivaadid, nende saamise protsess, neid sisaldavad ravimpreparaadid ja nende kasutamine |
US08/465,916 US5780631A (en) | 1993-06-03 | 1995-06-06 | Starting materials in the synthesis of thrombin and kininogenase inhibitors |
US08/468,046 US5602253A (en) | 1993-06-03 | 1995-06-06 | Peptides derivatives |
US08/470,277 US5723444A (en) | 1993-06-03 | 1995-06-06 | Starting materials in the synthesis of thrombin and kinogenase inhibitors |
US08/470,258 US5783563A (en) | 1993-06-03 | 1995-06-06 | Method for treatment or prophylaxis of venous thrombosis |
US08/484,427 US5856307A (en) | 1993-06-03 | 1995-06-07 | Peptide derivatives as kininogenase inhibitors |
US08/481,811 US5939392A (en) | 1993-06-03 | 1995-06-07 | Method of thrombin inhibition |
NO19954873A NO314406B1 (no) | 1993-06-03 | 1995-11-30 | Nye peptidderivater, farmasöytisk preparat inneholdende slike derivater, deres anvendelse, fremgangsmåter for deres fremstilling, ogmellomprodukter |
FI955828A FI119812B (fi) | 1993-06-03 | 1995-12-04 | Menetelmä uusien, terapeuttisesti käyttökelpoisten peptidijohdannaisten valmistamiseksi |
CNB991248597A CN1178905C (zh) | 1993-06-03 | 1999-11-15 | 新的肽衍生物 |
US09/566,403 US6984627B1 (en) | 1993-06-03 | 2000-05-08 | Peptide derivatives |
JP2001091958A JP2001322974A (ja) | 1993-06-03 | 2001-03-28 | 4−アミノメチル−1−アミジノベンゼン化合物 |
HK01102259A HK1031375A1 (en) | 1993-06-03 | 2001-03-28 | New peptide derivatives. |
JP2001158596A JP2002047264A (ja) | 1993-06-03 | 2001-05-28 | アミノアルキルベンゼン化合物 |
GR20010401107T GR3036258T3 (en) | 1993-06-03 | 2001-07-24 | New peptide derivatives |
NO2004009C NO2004009I1 (no) | 1993-06-03 | 2004-12-13 | Melagatran, stereoisomerer derav eller fysiologisksalter eller estrer derav |
NL300178C NL300178I2 (nl) | 1993-06-03 | 2005-03-03 | Nieuwe peptidederivaten. |
US11/090,786 US20050222395A1 (en) | 1993-06-03 | 2005-03-25 | New peptide derivatives |
LU91173C LU91173I2 (fr) | 1993-06-03 | 2005-05-11 | Ximelagatran, et les sels pharmaceutiquement acceptables de celui-ci (exanta). |
US12/222,604 US20090192137A1 (en) | 1993-06-03 | 2008-08-12 | Dialysis method |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE19939301916A SE9301916D0 (sv) | 1993-06-03 | 1993-06-03 | New peptides derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
SE9301916D0 true SE9301916D0 (sv) | 1993-06-03 |
Family
ID=20390165
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE19939301916A SE9301916D0 (sv) | 1993-06-03 | 1993-06-03 | New peptides derivatives |
Country Status (40)
Country | Link |
---|---|
US (4) | US5723444A (zh) |
EP (2) | EP0701568B1 (zh) |
JP (3) | JP3205558B2 (zh) |
KR (1) | KR100339456B1 (zh) |
CN (2) | CN1099425C (zh) |
AT (1) | ATE200783T1 (zh) |
BR (1) | BR9406746A (zh) |
CA (1) | CA2162900C (zh) |
CZ (1) | CZ290104B6 (zh) |
DE (3) | DE69427150T2 (zh) |
DK (1) | DK0701568T3 (zh) |
EE (1) | EE03264B1 (zh) |
EG (1) | EG20671A (zh) |
ES (1) | ES2128277T3 (zh) |
FI (1) | FI119812B (zh) |
GR (1) | GR3036258T3 (zh) |
HK (1) | HK1031375A1 (zh) |
HR (1) | HRP940311B1 (zh) |
HU (2) | HU226825B1 (zh) |
IL (2) | IL123996A (zh) |
IS (1) | IS1805B (zh) |
LT (1) | LT3768B (zh) |
LU (1) | LU91173I2 (zh) |
MX (1) | MX9404114A (zh) |
MY (1) | MY119155A (zh) |
NL (1) | NL300178I2 (zh) |
NO (2) | NO314406B1 (zh) |
NZ (1) | NZ267534A (zh) |
PL (1) | PL181968B1 (zh) |
PT (1) | PT701568E (zh) |
RS (1) | RS49576B (zh) |
RU (1) | RU2142469C1 (zh) |
SA (1) | SA94150051B1 (zh) |
SE (1) | SE9301916D0 (zh) |
SG (1) | SG48013A1 (zh) |
SI (1) | SI0701568T1 (zh) |
SK (1) | SK283150B6 (zh) |
TW (1) | TW403731B (zh) |
UA (1) | UA65518C2 (zh) |
WO (1) | WO1994029336A1 (zh) |
Families Citing this family (125)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5583146A (en) * | 1992-12-02 | 1996-12-10 | Bristol-Myers Squibb Company | Heterocyclic thrombin inhibitors |
SE9900043D0 (sv) * | 1999-01-11 | 1999-01-11 | Astra Ab | New use |
SE9301916D0 (sv) * | 1993-06-03 | 1993-06-03 | Ab Astra | New peptides derivatives |
US6984627B1 (en) * | 1993-06-03 | 2006-01-10 | Astrazeneca Ab | Peptide derivatives |
DE69416848T2 (de) * | 1993-10-21 | 1999-07-08 | Searle & Co | Amidino-derivate als no-synthetase inhibitoren |
JP4561696B2 (ja) * | 1994-01-27 | 2010-10-13 | 三菱化学株式会社 | プロリンアミド誘導体 |
CA2143533A1 (en) * | 1994-03-04 | 1995-09-05 | Kenneth D. Kurz | Antithrombotic agents |
ZA951617B (en) * | 1994-03-04 | 1997-02-27 | Lilly Co Eli | Antithrombotic agents. |
US5602101A (en) * | 1994-03-04 | 1997-02-11 | Eli Lilly And Company | Antithrombotic agents |
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2001
- 2001-03-28 JP JP2001091958A patent/JP2001322974A/ja active Pending
- 2001-03-28 HK HK01102259A patent/HK1031375A1/xx not_active IP Right Cessation
- 2001-05-28 JP JP2001158596A patent/JP2002047264A/ja active Pending
- 2001-07-24 GR GR20010401107T patent/GR3036258T3/el unknown
-
2004
- 2004-12-13 NO NO2004009C patent/NO2004009I1/no unknown
-
2005
- 2005-03-03 NL NL300178C patent/NL300178I2/nl unknown
- 2005-03-25 US US11/090,786 patent/US20050222395A1/en not_active Abandoned
- 2005-05-11 LU LU91173C patent/LU91173I2/fr unknown
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