SE0301446D0 - New Compounds - Google Patents

New Compounds

Info

Publication number
SE0301446D0
SE0301446D0 SE0301446A SE0301446A SE0301446D0 SE 0301446 D0 SE0301446 D0 SE 0301446D0 SE 0301446 A SE0301446 A SE 0301446A SE 0301446 A SE0301446 A SE 0301446A SE 0301446 D0 SE0301446 D0 SE 0301446D0
Authority
SE
Sweden
Prior art keywords
compounds
new compounds
formula
preparation
new
Prior art date
Application number
SE0301446A
Other languages
English (en)
Swedish (sv)
Inventor
Yevgeni Besidski
Didier Rotticci
Andis Slaitas
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Priority to SE0301446A priority Critical patent/SE0301446D0/xx
Publication of SE0301446D0 publication Critical patent/SE0301446D0/xx
Priority to SE0400043A priority patent/SE0400043D0/xx
Priority to TW093113091A priority patent/TWI333950B/zh
Priority to PCT/SE2004/000738 priority patent/WO2004100865A2/fr
Priority to BRPI0410316-5A priority patent/BRPI0410316A/pt
Priority to RU2005136529/04A priority patent/RU2337098C2/ru
Priority to EP04732865A priority patent/EP1626964B1/fr
Priority to SG200717747-0A priority patent/SG171471A1/en
Priority to PT04732865T priority patent/PT1626964E/pt
Priority to DE602004019208T priority patent/DE602004019208D1/de
Priority to EP08171574A priority patent/EP2042490A3/fr
Priority to NZ543075A priority patent/NZ543075A/en
Priority to MXPA05012247A priority patent/MXPA05012247A/es
Priority to KR1020057021744A priority patent/KR101110404B1/ko
Priority to UAA200510093A priority patent/UA85842C2/uk
Priority to CNA2008101360511A priority patent/CN101328150A/zh
Priority to JP2006532186A priority patent/JP4762903B2/ja
Priority to CA2525628A priority patent/CA2525628C/fr
Priority to AT04732865T priority patent/ATE421506T1/de
Priority to ES04732865T priority patent/ES2319529T3/es
Priority to AU2004238177A priority patent/AU2004238177B2/en
Priority to US10/556,229 priority patent/US7645784B2/en
Priority to SG200717748-8A priority patent/SG164283A1/en
Priority to CNB2004800126199A priority patent/CN100413849C/zh
Priority to SI200431067T priority patent/SI1626964T1/sl
Priority to PL04732865T priority patent/PL1626964T3/pl
Priority to DK04732865T priority patent/DK1626964T3/da
Priority to ARP040101658A priority patent/AR044342A1/es
Priority to MYPI20041802A priority patent/MY140235A/en
Priority to CO05114671A priority patent/CO5631436A2/es
Priority to ZA200509241A priority patent/ZA200509241B/en
Priority to IS8180A priority patent/IS2656B/is
Priority to NO20055977A priority patent/NO20055977L/no
Priority to HK06105843.2A priority patent/HK1085735A1/xx
Priority to AU2008203305A priority patent/AU2008203305A1/en
Priority to CY20091100309T priority patent/CY1108894T1/el
Priority to HR20090167T priority patent/HRP20090167T1/xx
Priority to IL199668A priority patent/IL199668A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C215/04—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated
    • C07C215/06—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic
    • C07C215/16—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic the nitrogen atom of the amino group being further bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/52—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
    • C07C229/54—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C229/56—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring with amino and carboxyl groups bound in ortho-position
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/12—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
    • C07C233/15—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/46—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/47—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/16—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/14—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/26—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C317/32—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C317/34—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring
    • C07C317/36—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring with the nitrogen atoms of the amino groups bound to hydrogen atoms or to carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08—Radicals containing only hydrogen and carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30—Nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
SE0301446A 2003-05-16 2003-05-16 New Compounds SE0301446D0 (sv)

Priority Applications (38)

Application Number Priority Date Filing Date Title
SE0301446A SE0301446D0 (sv) 2003-05-16 2003-05-16 New Compounds
SE0400043A SE0400043D0 (sv) 2003-05-16 2004-01-12 New compounds
TW093113091A TWI333950B (en) 2003-05-16 2004-05-10 New benzimidazole derivatives
DK04732865T DK1626964T3 (da) 2003-05-16 2004-05-13 Nye benzimidazolderivater
AT04732865T ATE421506T1 (de) 2003-05-16 2004-05-13 Neue benzimidazolderivate
AU2004238177A AU2004238177B2 (en) 2003-05-16 2004-05-13 New benzimidazole derivatives
RU2005136529/04A RU2337098C2 (ru) 2003-05-16 2004-05-13 Новые производные бензимидазола и фармацевтическая композиция на их основе для использования в лечении расстройств, опосредованных vr1
EP04732865A EP1626964B1 (fr) 2003-05-16 2004-05-13 Nouveaux derives de benzimidazole
SG200717747-0A SG171471A1 (en) 2003-05-16 2004-05-13 New benzimidazole derivatives
PT04732865T PT1626964E (pt) 2003-05-16 2004-05-13 Novos derivados de benzimidazole
DE602004019208T DE602004019208D1 (de) 2003-05-16 2004-05-13 Neue benzimidazolderivate
EP08171574A EP2042490A3 (fr) 2003-05-16 2004-05-13 Dérivés du benzoimidazole comme antagonistes du recepteur Vanilloid
NZ543075A NZ543075A (en) 2003-05-16 2004-05-13 New benzimidazole derivatives
MXPA05012247A MXPA05012247A (es) 2003-05-16 2004-05-13 Derivados de bencimidazol nuevos.
KR1020057021744A KR101110404B1 (ko) 2003-05-16 2004-05-13 신규 벤즈이미다졸 유도체
UAA200510093A UA85842C2 (uk) 2003-05-16 2004-05-13 Похідні бензімідазолу як інгібітори ванілоїдного рецептора 1 (vr1)
CNA2008101360511A CN101328150A (zh) 2003-05-16 2004-05-13 新的苯并咪唑衍生物
JP2006532186A JP4762903B2 (ja) 2003-05-16 2004-05-13 新規のベンゾイミダゾール誘導体
CA2525628A CA2525628C (fr) 2003-05-16 2004-05-13 Nouveaux derives de benzimidazole
PCT/SE2004/000738 WO2004100865A2 (fr) 2003-05-16 2004-05-13 Nouveaux derives de benzimidazole
ES04732865T ES2319529T3 (es) 2003-05-16 2004-05-13 Nuevos derivados de bencimidazol.
BRPI0410316-5A BRPI0410316A (pt) 2003-05-16 2004-05-13 composto, composição farmacêutica, uso dos compostos, e, método de tratamento de distúrbios mediados por vr1 e para o tratamento de distúrbios de dores
US10/556,229 US7645784B2 (en) 2003-05-16 2004-05-13 Benzimidazole derivatives
SG200717748-8A SG164283A1 (en) 2003-05-16 2004-05-13 New benzimidazole derivatives
CNB2004800126199A CN100413849C (zh) 2003-05-16 2004-05-13 苯并咪唑衍生物
SI200431067T SI1626964T1 (sl) 2003-05-16 2004-05-13 Novi benzimidazolni derivati
PL04732865T PL1626964T3 (pl) 2003-05-16 2004-05-13 Nowe pochodne benzimidazolu
MYPI20041802A MY140235A (en) 2003-05-16 2004-05-14 New benzimidazole derivatives
ARP040101658A AR044342A1 (es) 2003-05-16 2004-05-14 Derivados de bencimidazol
CO05114671A CO5631436A2 (es) 2003-05-16 2005-11-10 Amidas y acidos derivados del bencimidazol para el tratamiento del dolor y la inflamacion
ZA200509241A ZA200509241B (en) 2003-05-16 2005-11-15 New benzimidazole derivatives
IS8180A IS2656B (is) 2003-05-16 2005-12-14 Nýjar besímídasólafleiður
NO20055977A NO20055977L (no) 2003-05-16 2005-12-15 Nye benzimidazolderivater
HK06105843.2A HK1085735A1 (en) 2003-05-16 2006-05-20 New benzimidazole derivatives
AU2008203305A AU2008203305A1 (en) 2003-05-16 2008-07-24 New benzimidazole derivatives
CY20091100309T CY1108894T1 (el) 2003-05-16 2009-03-19 Νεα παραγωγα βενζιμιδαζολης
HR20090167T HRP20090167T1 (en) 2003-05-16 2009-03-19 New benzimidazole derivatives
IL199668A IL199668A0 (en) 2003-05-16 2009-07-02 New benzimidazole derivatives

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
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Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2377484T3 (es) * 2003-09-03 2012-03-28 Pfizer, Inc. Compuestos de bencimidazolona que tiene actividad agonista del receptor 5-HT
SE0402284D0 (sv) * 2004-09-21 2004-09-21 Astrazeneca Ab New heterocyclic amides
CA2581335A1 (fr) * 2004-09-21 2006-03-30 Athersys, Inc. Acides benzimidazole acetiques presentant un antagonisme du recepteur crth2 et utilisations associees
TWI401254B (zh) * 2005-05-09 2013-07-11 Hydra Biosciences Inc 用於調節ｔｒｐｖ３功能之化合物
US8916550B2 (en) 2005-05-09 2014-12-23 Hydra Biosciences, Inc. Compounds for modulating TRPV3 function
KR20110093948A (ko) 2005-07-22 2011-08-18 모찌다 세이야쿠 가부시끼가이샤 신규 헤테로시클리덴 아세트아미드 유도체
RU2451014C2 (ru) * 2005-07-22 2012-05-20 Мотида Фармасьютикал Ко., Лтд. Новое производное гетероциклиден ацетамида
AU2006311036A1 (en) * 2005-11-08 2007-05-18 Msd Oss B.V. 2-(benzimidazol-1-yl)-N-(4-phenylthiazol-2-yl) acetamide derivatives useful in treatment of TRPV1 related disorders
WO2007054480A1 (fr) 2005-11-08 2007-05-18 N.V. Organon Derives bisarylique de 2-(benzimidazol-1-yl)-acetamide et leur utilisation comme inhibiteurs du recepteur trpv1
UY30048A1 (es) * 2005-12-23 2007-07-31 Astrazeneca Ab Derivados sustituidos de la n,2-(1h-benzimidazol-1-il) acetamida, composiciones farmacéuticas conteniéndolos, procesos de preparación y aplicaciones
WO2007091946A1 (fr) * 2006-02-07 2007-08-16 Astrazeneca Ab Utilisation de spiro[imidazolidine-4,3'-indole]2,2',5'(1h)triones pour le traitement de troubles associes au recepteur 1 de vanilloide
TW200801011A (en) 2006-02-07 2008-01-01 Astrazeneca Ab New compounds II
JP2009526044A (ja) * 2006-02-07 2009-07-16 アストラゼネカ・アクチエボラーグ 新規な化合物ｉ
TWI433839B (zh) 2006-08-11 2014-04-11 Neomed Inst 新穎的苯并咪唑衍生物290
EP2099444A4 (fr) 2006-12-14 2012-11-07 Nps Pharma Inc Utilisation de dérivés de la d-sérine pour le traitement de troubles de l'anxiété
PE20081692A1 (es) * 2007-01-24 2008-12-18 Mochida Pharm Co Ltd Nuevo derivado de heterocicliden acetamida
DE102007018151A1 (de) 2007-04-16 2008-10-23 Günenthal GmbH Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
CA2683461A1 (fr) * 2007-04-16 2008-10-23 Gruenenthal Gmbh Nouveaux ligands du recepteur vanilloide et leur utilisation pour la fabrication de medicaments
DE102007018149A1 (de) 2007-04-16 2008-10-23 Grünenthal GmbH Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
US10179761B2 (en) 2014-06-16 2019-01-15 Universite De Lille 2 Droit Et Sante Compounds, pharmaceutical composition and their use in treating neurodegenerative diseases
JP2018052817A (ja) * 2015-01-21 2018-04-05 大日本住友製薬株式会社 新規ベンズイミダゾール誘導体およびその医薬用途
WO2018051252A2 (fr) * 2016-09-15 2018-03-22 Insecticides (India) Limited Nouveau composé amide, son procédé de production et miticide
WO2020142842A1 (fr) * 2019-01-08 2020-07-16 Neomed Institute - Institut Neomed Formes cristallines de (s)-2-(7-cyano-1h-benzimidazol-1 yl)- n-{1-[4-(1-cyano-1-méthyléthyl)phényl]éthyl}acétamide
WO2022211518A1 (fr) * 2021-04-02 2022-10-06 파렌키마바이오텍 주식회사 Nouveau composé et son utilisation dans le traitement du psoriasis, de l'asthme ou du lupus érythémateux disséminé
DE102022104759A1 (de) 2022-02-28 2023-08-31 SCi Kontor GmbH Co-Kristall-Screening Verfahren, insbesondere zur Herstellung von Co-Kristallen

Family Cites Families (46)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1186504A (en) * 1966-10-15 1970-04-02 Fisons Pest Control Ltd Substituted Heterocyclic Compounds
IT1036004B (it) 1968-05-21 1979-10-30 Abc Ist Biolog Chem Spa Acidt 3 indolil adetoidrossamici
BE793718A (fr) 1972-01-07 1973-07-05 Merck & Co Inc Aminobenzimidazoles
DE3347290A1 (de) * 1983-12-28 1985-07-11 Dr. Karl Thomae Gmbh, 7950 Biberach Neue 2-phenyl-imidazole, ihre herstellung und diese verbindungen enthaltende arzneimittel
US4738981A (en) 1984-11-13 1988-04-19 Warner-Lambert Substituted trans-1,2-diaminocyclohexyl amide compounds
JPH06759B2 (ja) * 1989-09-22 1994-01-05 ファイザー製薬株式会社 新規なベンゾイミダゾール化合物
DE4309969A1 (de) * 1993-03-26 1994-09-29 Bayer Ag Substituierte heteroanellierte Imidazole
DE4491980B4 (de) * 1993-03-30 2006-05-11 Dainippon Ink And Chemicals, Inc. Härtbare Harzmasse, ihre Verwendung sowie Anstrichmittel
US5403851A (en) 1994-04-05 1995-04-04 Interneuron Pharmaceuticals, Inc. Substituted tryptamines, phenalkylamines and related compounds
HUT78019A (hu) * 1995-03-31 1999-05-28 András Horváth Eljárás szubsztituált nitrogéntartalmú, heterociklusos vegyületek szintézisére
WO1997012613A1 (fr) * 1995-10-05 1997-04-10 Warner-Lambert Company Procede de traitement et de prevention des inflammations et de l'atherosclerose
EA002357B1 (ru) 1995-12-28 2002-04-25 Фудзисава Фармасьютикал Ко., Лтд. Производные бензимидазола
CZ295468B6 (cs) 1996-04-12 2005-08-17 Warner-Lambert Company Polycyklické sloučeniny
GB9713484D0 (en) 1997-06-27 1997-09-03 Smithkline Beecham Plc Neuroprotective vanilloid compounds
JP2000095767A (ja) 1998-09-28 2000-04-04 Takeda Chem Ind Ltd 性腺刺激ホルモン放出ホルモン拮抗剤
KR20020060160A (ko) 1999-08-12 2002-07-16 파마시아 이탈리아 에스.피.에이. 3(5)-아미노-피라졸 유도체, 이의 제조 방법 및항종양제로서의 이의 용도
US6534651B2 (en) * 2000-04-06 2003-03-18 Inotek Pharmaceuticals Corp. 7-Substituted isoindolinone inhibitors of inflammation and reperfusion injury and methods of use thereof
WO2001085722A1 (fr) * 2000-05-05 2001-11-15 Cor Therapeutics, Inc. Sulfonamides heterobicycliques et utilisation de celles-ci comme inhibiteurs de recepteur adp des plaquettes
US6943174B2 (en) 2000-06-14 2005-09-13 Warner-Lambert Company 6,5-Fused bicyclic heterocycles
US6448281B1 (en) * 2000-07-06 2002-09-10 Boehringer Ingelheim (Canada) Ltd. Viral polymerase inhibitors
CA2420042A1 (fr) 2000-08-22 2003-02-18 Mikio Ogawa Derives d'acide carboxylique, procede de production de ceux-ci et medicaments contenant ceux-ci comme principe actif
GB0031315D0 (en) * 2000-12-21 2001-02-07 Glaxo Group Ltd Indole derivatives
ITTO20010110A1 (it) 2001-02-08 2002-08-08 Rotta Research Lab Nuovi derivati benzamidinici dotati di attivita' anti-infiammatoria ed immunosoppressiva.
GB0105895D0 (en) 2001-03-09 2001-04-25 Smithkline Beecham Plc Novel compounds
SE0101387D0 (sv) * 2001-04-20 2001-04-20 Astrazeneca Ab Novel compounds
GB0110901D0 (en) 2001-05-02 2001-06-27 Smithkline Beecham Plc Novel Compounds
EA008476B1 (ru) 2001-06-11 2007-06-29 Биовитрум Аб Замещенные сульфонамиды, способ их получения и их применение в качестве лечебного средства для лечения расстройств цнс, ожирения и диабета типа ii
TWI239942B (en) * 2001-06-11 2005-09-21 Dainippon Pharmaceutical Co N-arylphenylacetamide derivative and pharmaceutical composition containing the same
WO2003014064A1 (fr) 2001-07-31 2003-02-20 Bayer Healthcare Ag Derives amines
PE20030417A1 (es) 2001-09-13 2003-08-06 Smithkline Beecham Plc Derivados de urea como antagonistas del receptor vainilloide
TWI231757B (en) 2001-09-21 2005-05-01 Solvay Pharm Bv 1H-Imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity
CA2468544A1 (fr) 2001-12-10 2003-06-19 Amgen Inc. Ligands de recepteur vanilloide et utilisation de ceux-ci dans des traitements
GB0130550D0 (en) 2001-12-20 2002-02-06 Smithkline Beecham Plc Novel compounds
EP2033953A1 (fr) 2002-02-15 2009-03-11 Glaxo Group Limited Modulateurs des récepteurs vanilloides
US20030158188A1 (en) * 2002-02-20 2003-08-21 Chih-Hung Lee Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor
SG156524A1 (en) * 2002-06-20 2009-11-26 Biovitrum Ab Publ New compounds useful for the treatment of obesity, type ii diabetes and cns disorders
GB0221157D0 (en) 2002-09-12 2002-10-23 Glaxo Group Ltd Novel treatment
WO2004024710A1 (fr) 2002-09-13 2004-03-25 Glaxo Group Limited Composes a base d'uree, actifs en tant qu'antagonistes du recepteur de la vanilloide et utilises pour traiter les douleurs
US7582761B2 (en) * 2002-10-17 2009-09-01 Amgen Inc. Vanilloid receptor ligands and their use in treatments
SE0301701D0 (sv) * 2003-06-10 2003-06-10 Astrazeneca Ab Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof
ES2377484T3 (es) 2003-09-03 2012-03-28 Pfizer, Inc. Compuestos de bencimidazolona que tiene actividad agonista del receptor 5-HT
EP1736465A4 (fr) 2004-03-31 2009-06-17 Ajinomoto Kk Dérivés d'aniline
WO2006007851A2 (fr) 2004-07-19 2006-01-26 Novo Nordisk A/S Inhibition de l'activite du recepteur de la capsaicine dans le traitement de l'obesite ou de maladies et de troubles associe(e)s a l'obesite
SE0402284D0 (sv) 2004-09-21 2004-09-21 Astrazeneca Ab New heterocyclic amides
UY30048A1 (es) 2005-12-23 2007-07-31 Astrazeneca Ab Derivados sustituidos de la n,2-(1h-benzimidazol-1-il) acetamida, composiciones farmacéuticas conteniéndolos, procesos de preparación y aplicaciones
TWI433839B (zh) 2006-08-11 2014-04-11 Neomed Inst 新穎的苯并咪唑衍生物290

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AU2008203305A1 (en) 2008-08-14
SI1626964T1 (sl) 2009-06-30
UA85842C2 (uk) 2009-03-10
HK1085735A1 (en) 2006-09-01
RU2005136529A (ru) 2006-06-10
AU2004238177A1 (en) 2004-11-25
DE602004019208D1 (de) 2009-03-12
SG171471A1 (en) 2011-06-29
CY1108894T1 (el) 2014-07-02
KR101110404B1 (ko) 2012-02-17
EP2042490A2 (fr) 2009-04-01
PL1626964T3 (pl) 2009-06-30
US20060287377A1 (en) 2006-12-21
IS2656B (is) 2010-08-15
SG164283A1 (en) 2010-09-29
IL199668A0 (en) 2011-08-01
IS8180A (is) 2005-12-14
EP2042490A3 (fr) 2009-09-30
CO5631436A2 (es) 2006-04-28
CA2525628A1 (fr) 2004-11-25
US7645784B2 (en) 2010-01-12
MY140235A (en) 2009-12-31
CA2525628C (fr) 2012-03-06
CN100413849C (zh) 2008-08-27
HRP20090167T1 (en) 2009-05-31
TW200508207A (en) 2005-03-01
ZA200509241B (en) 2007-04-25
CN101328150A (zh) 2008-12-24
DK1626964T3 (da) 2009-04-20
JP4762903B2 (ja) 2011-08-31
WO2004100865A2 (fr) 2004-11-25
CN1784387A (zh) 2006-06-07
AU2004238177B2 (en) 2008-04-24
MXPA05012247A (es) 2006-02-10
ATE421506T1 (de) 2009-02-15
SE0400043D0 (sv) 2004-01-12
AR044342A1 (es) 2005-09-07
ES2319529T3 (es) 2009-05-08
NO20055977L (no) 2006-02-16
EP1626964A2 (fr) 2006-02-22
JP2006528971A (ja) 2006-12-28
BRPI0410316A (pt) 2006-05-23
RU2337098C2 (ru) 2008-10-27
KR20060009936A (ko) 2006-02-01
NZ543075A (en) 2009-03-31
EP1626964B1 (fr) 2009-01-21
TWI333950B (en) 2010-12-01
WO2004100865A3 (fr) 2005-01-20

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