RU2008143179A - Органические соединения - Google Patents

Органические соединения Download PDF

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Publication number
RU2008143179A
RU2008143179A RU2008143179/04A RU2008143179A RU2008143179A RU 2008143179 A RU2008143179 A RU 2008143179A RU 2008143179/04 A RU2008143179/04 A RU 2008143179/04A RU 2008143179 A RU2008143179 A RU 2008143179A RU 2008143179 A RU2008143179 A RU 2008143179A
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RU
Russia
Prior art keywords
optionally substituted
compound according
independently selected
halogen
disease
Prior art date
Application number
RU2008143179/04A
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English (en)
Russian (ru)
Inventor
Даниэль Каспар БЕШЛИН (CH)
Даниэль Каспар БЕШЛИН
Нильс ОСТЕРМАНН (DE)
Нильс Остерманн
Франсуа ЖЕССЬЕ (FR)
Франсуа Жессье
Фентон СИРОКЕН (FR)
Фентон СИРОКЕН
Кенджи НАМОТО (CH)
Кенджи Намото
Original Assignee
Новартис АГ (CH)
Новартис Аг
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Application filed by Новартис АГ (CH), Новартис Аг filed Critical Новартис АГ (CH)
Publication of RU2008143179A publication Critical patent/RU2008143179A/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Emergency Medicine (AREA)
  • Communicable Diseases (AREA)
RU2008143179/04A 2006-03-31 2007-03-29 Органические соединения RU2008143179A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78829406P 2006-03-31 2006-03-31
US60/788,294 2006-03-31

Publications (1)

Publication Number Publication Date
RU2008143179A true RU2008143179A (ru) 2010-05-10

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ID=38235160

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2008143179/04A RU2008143179A (ru) 2006-03-31 2007-03-29 Органические соединения

Country Status (11)

Country Link
US (2) US8097617B2 (cg-RX-API-DMAC7.html)
EP (1) EP2004643A1 (cg-RX-API-DMAC7.html)
JP (1) JP2009531390A (cg-RX-API-DMAC7.html)
KR (1) KR20080104351A (cg-RX-API-DMAC7.html)
CN (1) CN101410397A (cg-RX-API-DMAC7.html)
AU (1) AU2007233709A1 (cg-RX-API-DMAC7.html)
BR (1) BRPI0710110A2 (cg-RX-API-DMAC7.html)
CA (1) CA2644963A1 (cg-RX-API-DMAC7.html)
MX (1) MX2008012617A (cg-RX-API-DMAC7.html)
RU (1) RU2008143179A (cg-RX-API-DMAC7.html)
WO (1) WO2007113226A1 (cg-RX-API-DMAC7.html)

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US8710050B2 (en) 2011-03-08 2014-04-29 Sanofi Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
WO2012120053A1 (de) 2011-03-08 2012-09-13 Sanofi Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2683705B1 (de) 2011-03-08 2015-04-22 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
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