RU2005111256A - Производные фенола и их применение в качестве ингибиторов ротамаз - Google Patents

Производные фенола и их применение в качестве ингибиторов ротамаз Download PDF

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Publication number
RU2005111256A
RU2005111256A RU2005111256/04A RU2005111256A RU2005111256A RU 2005111256 A RU2005111256 A RU 2005111256A RU 2005111256/04 A RU2005111256/04 A RU 2005111256/04A RU 2005111256 A RU2005111256 A RU 2005111256A RU 2005111256 A RU2005111256 A RU 2005111256A
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Russia
Prior art keywords
hydroxyphenyl
chloro
dichloro
phenol
urea
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RU2005111256/04A
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English (en)
Russian (ru)
Inventor
Йохен КНОЛЛЕ (DE)
Йохен Кнолле
Мике ШУТКОВСКИ (DE)
Мике ШУТКОВСКИ
Герд ХУММЕЛЬ (DE)
Герд ХУММЕЛЬ
Томас ТРАДЛЕР (DE)
Томас ТРАДЛЕР
Лоранс ЖОБРОН (DE)
Лоранс ЖОБРОН
Клаудиа КРИСТНЕР (DE)
Клаудиа КРИСТНЕР
Дирк ШАРН (DE)
Дирк ШАРН
Роланд ШТРАГИС (DE)
Роланд ШТРАГИС
Кристоф ГИБСОН (DE)
Кристоф ГИБСОН
Франк ОСТЕРКАМП (DE)
Франк ОСТЕРКАМП
Original Assignee
Йерини Аг (De)
Йерини Аг
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Application filed by Йерини Аг (De), Йерини Аг filed Critical Йерини Аг (De)
Publication of RU2005111256A publication Critical patent/RU2005111256A/ru

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    • C07C275/00Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/28Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C275/32Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
    • C07C275/34Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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RU2005111256/04A 2002-09-18 2003-09-18 Производные фенола и их применение в качестве ингибиторов ротамаз RU2005111256A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP20020020987 EP1402888A1 (en) 2002-09-18 2002-09-18 The use of substituted carbocyclic compounds as rotamases inhibitors
EP02020987.0 2002-09-18

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RU2010136779/04A Division RU2010136779A (ru) 2002-09-18 2010-09-02 Производные фенола и их применение в качестве ингибиторов ротамаз

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RU2010136779/04A RU2010136779A (ru) 2002-09-18 2010-09-02 Производные фенола и их применение в качестве ингибиторов ротамаз

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US (2) US20070054904A1 (https=)
EP (3) EP1402888A1 (https=)
JP (2) JP2005539072A (https=)
KR (1) KR20050053673A (https=)
CN (1) CN100546977C (https=)
AU (1) AU2003271619A1 (https=)
BR (1) BR0314544A (https=)
CA (1) CA2498662A1 (https=)
MX (1) MXPA05003084A (https=)
PL (1) PL374846A1 (https=)
RU (2) RU2005111256A (https=)
SG (1) SG165995A1 (https=)
WO (1) WO2004026815A2 (https=)
ZA (1) ZA200501913B (https=)

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CA2514363A1 (en) * 2003-02-12 2004-08-26 Transtech Pharma, Inc. Substituted azole derivatives as therapeutic agents
US20050026844A1 (en) 2003-04-03 2005-02-03 Regents Of The University Of California Inhibitors for the soluble epoxide hydrolase
WO2005089380A2 (en) 2004-03-16 2005-09-29 The Regents Of The University Of California Reducing nephropathy with inhibitors of soluble epoxide hydrolase and epoxyeicosanoids
PL1701940T3 (pl) * 2003-12-23 2008-11-28 H Lundbeck As Pochodne 2-(1H-indolilosulfanylo)benzyloaminy jako SSRI
CA2554809C (en) * 2004-02-05 2014-04-29 Probiodrug Ag Novel n-alkyl thiourea- and thioamide-substituted imidazolyl inhibitors of glutaminyl cyclase
US7550499B2 (en) 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
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RU2010136779A (ru) 2012-03-10
EP2100876A3 (en) 2010-02-24
EP1402888A1 (en) 2004-03-31
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