RU2005111256A - Производные фенола и их применение в качестве ингибиторов ротамаз - Google Patents
Производные фенола и их применение в качестве ингибиторов ротамаз Download PDFInfo
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- RU2005111256A RU2005111256A RU2005111256/04A RU2005111256A RU2005111256A RU 2005111256 A RU2005111256 A RU 2005111256A RU 2005111256/04 A RU2005111256/04 A RU 2005111256/04A RU 2005111256 A RU2005111256 A RU 2005111256A RU 2005111256 A RU2005111256 A RU 2005111256A
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- hydroxyphenyl
- chloro
- dichloro
- phenol
- urea
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C275/32—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
- C07C275/34—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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- C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02020987.0 | 2002-09-18 | ||
| EP20020020987 EP1402888A1 (en) | 2002-09-18 | 2002-09-18 | The use of substituted carbocyclic compounds as rotamases inhibitors |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2010136779/04A Division RU2010136779A (ru) | 2002-09-18 | 2010-09-02 | Производные фенола и их применение в качестве ингибиторов ротамаз |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| RU2005111256A true RU2005111256A (ru) | 2006-10-27 |
Family
ID=31970282
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2005111256/04A RU2005111256A (ru) | 2002-09-18 | 2003-09-18 | Производные фенола и их применение в качестве ингибиторов ротамаз |
| RU2010136779/04A RU2010136779A (ru) | 2002-09-18 | 2010-09-02 | Производные фенола и их применение в качестве ингибиторов ротамаз |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2010136779/04A RU2010136779A (ru) | 2002-09-18 | 2010-09-02 | Производные фенола и их применение в качестве ингибиторов ротамаз |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US20070054904A1 (https=) |
| EP (3) | EP1402888A1 (https=) |
| JP (2) | JP2005539072A (https=) |
| KR (1) | KR20050053673A (https=) |
| CN (1) | CN100546977C (https=) |
| AU (1) | AU2003271619A1 (https=) |
| BR (1) | BR0314544A (https=) |
| CA (1) | CA2498662A1 (https=) |
| MX (1) | MXPA05003084A (https=) |
| PL (1) | PL374846A1 (https=) |
| RU (2) | RU2005111256A (https=) |
| SG (1) | SG165995A1 (https=) |
| WO (1) | WO2004026815A2 (https=) |
| ZA (1) | ZA200501913B (https=) |
Families Citing this family (47)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2006518738A (ja) * | 2003-02-12 | 2006-08-17 | トランス テック ファーマ,インコーポレイテッド | 治療薬としての置換アゾール誘導体 |
| CA2520763A1 (en) * | 2003-04-03 | 2004-10-21 | The Regents Of The University Of California | Improved inhibitors for the soluble epoxide hydrolase |
| RS50589B (sr) * | 2003-12-23 | 2010-05-07 | H. Lundbeck A/S. | 2-(1h-indolilsulfanil)-benzil amin derivati kao ssri |
| US7304086B2 (en) * | 2004-02-05 | 2007-12-04 | Probiodrug Ag | Inhibitors of glutaminyl cyclase |
| EP1765311A4 (en) | 2004-03-16 | 2009-04-29 | Univ California | REDUCTION OF NEPHROPATHY WITH INHIBITORS OF SOLUBLE EPOXY HYDROLASE AND EPOXYEICOSANOIDS |
| US7550499B2 (en) | 2004-05-12 | 2009-06-23 | Bristol-Myers Squibb Company | Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions |
| WO2005113534A2 (en) * | 2004-05-12 | 2005-12-01 | Schering Corporation | Cxcr1 and cxcr2 chemokine antagonists |
| AR052308A1 (es) * | 2004-07-16 | 2007-03-14 | Lundbeck & Co As H | Derivados de 2-(1h-indolilsulfanil)-arilamina y una composicion farmaceutica que contiene al compuesto |
| US7662910B2 (en) * | 2004-10-20 | 2010-02-16 | The Regents Of The University Of California | Inhibitors for the soluble epoxide hydrolase |
| EP1954696B1 (en) | 2005-01-19 | 2011-02-23 | Bristol-Myers Squibb Company | 2-phenoxy-n-(1,3,4-thiadizol-2-yl)pyridin-3-amine derivatives and related compounds as p2y1 receptor inhibitors for the treatment of thromboembolic disorders |
| JP2008540571A (ja) * | 2005-05-12 | 2008-11-20 | ウィスコンシン・アルムニ・リサーチ・ファウンデーション | Pin1の遮断は活性化した免疫細胞によるサイトカイン産生を防ぐ |
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2002
- 2002-09-18 EP EP20020020987 patent/EP1402888A1/en not_active Withdrawn
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2003
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- 2003-09-18 SG SG200702382-3A patent/SG165995A1/en unknown
- 2003-09-18 US US10/528,139 patent/US20070054904A1/en not_active Abandoned
- 2003-09-18 MX MXPA05003084A patent/MXPA05003084A/es not_active Application Discontinuation
- 2003-09-18 JP JP2004537125A patent/JP2005539072A/ja not_active Withdrawn
- 2003-09-18 AU AU2003271619A patent/AU2003271619A1/en not_active Abandoned
- 2003-09-18 CA CA002498662A patent/CA2498662A1/en not_active Abandoned
- 2003-09-18 PL PL03374846A patent/PL374846A1/xx not_active Application Discontinuation
- 2003-09-18 WO PCT/EP2003/010406 patent/WO2004026815A2/en not_active Ceased
- 2003-09-18 RU RU2005111256/04A patent/RU2005111256A/ru not_active Application Discontinuation
- 2003-09-18 KR KR1020057004693A patent/KR20050053673A/ko not_active Ceased
- 2003-09-18 EP EP09007837A patent/EP2100876A3/en not_active Withdrawn
- 2003-09-18 EP EP03753427A patent/EP1539683A2/en not_active Ceased
- 2003-09-18 CN CNB038252651A patent/CN100546977C/zh not_active Expired - Fee Related
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- 2010-09-29 JP JP2010219856A patent/JP2011037869A/ja active Pending
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| KR20050053673A (ko) | 2005-06-08 |
| EP1402888A1 (en) | 2004-03-31 |
| JP2011037869A (ja) | 2011-02-24 |
| PL374846A1 (en) | 2005-11-14 |
| CA2498662A1 (en) | 2004-04-01 |
| AU2003271619A1 (en) | 2004-04-08 |
| WO2004026815A3 (en) | 2004-12-02 |
| EP2100876A3 (en) | 2010-02-24 |
| BR0314544A (pt) | 2005-08-16 |
| MXPA05003084A (es) | 2005-11-17 |
| US20110065760A1 (en) | 2011-03-17 |
| EP1539683A2 (en) | 2005-06-15 |
| EP2100876A2 (en) | 2009-09-16 |
| WO2004026815A2 (en) | 2004-04-01 |
| ZA200501913B (en) | 2005-07-27 |
| SG165995A1 (en) | 2010-11-29 |
| RU2010136779A (ru) | 2012-03-10 |
| CN100546977C (zh) | 2009-10-07 |
| JP2005539072A (ja) | 2005-12-22 |
| CN1701061A (zh) | 2005-11-23 |
| US20070054904A1 (en) | 2007-03-08 |
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